التفاصيل البيبلوغرافية
العنوان: |
Improved Binding Affinity and Pharmacokinetics Enable Sustained Degradation of BCL6 In Vivo |
المؤلفون: |
Huckvale, Rosemary, Harnden, Alice C., Cheung, Kwai-Ming J., Pierrat, Olivier A., Talbot, Rachel, Box, Gary M., Henley, Alan T., de Haven Brandon, Alexis K., Hallsworth, Albert E., Bright, Michael D., Akpinar, Hafize Aysin, Miller, Daniel S. J., Tarantino, Dalia, Gowan, Sharon, Hayes, Angela, Gunnell, Emma A., Brennan, Alfie, Davis, Owen A., Johnson, Louise D., de Klerk, Selby, McAndrew, Craig, Le Bihan, Yann-Vaï, Meniconi, Mirco, Burke, Rosemary, Kirkin, Vladimir, van Montfort, Rob L. M., Raynaud, Florence I., Rossanese, Olivia W., Bellenie, Benjamin R., Hoelder, Swen |
المساهمون: |
Cancer Research UK, Sixth Element Capital |
المصدر: |
Journal of Medicinal Chemistry ; volume 65, issue 12, page 8191-8207 ; ISSN 0022-2623 1520-4804 |
بيانات النشر: |
American Chemical Society (ACS) |
سنة النشر: |
2022 |
مصطلحات موضوعية: |
Drug Discovery, Molecular Medicine |
نوع الوثيقة: |
article in journal/newspaper |
اللغة: |
English |
DOI: |
10.1021/acs.jmedchem.1c02175 |
الإتاحة: |
https://doi.org/10.1021/acs.jmedchem.1c02175Test |
حقوق: |
https://creativecommons.org/licenses/by/4.0Test/ |
رقم الانضمام: |
edsbas.C2AFDF3E |
قاعدة البيانات: |
BASE |