المؤلفون: Stefania Butini, Uwe Grether, Kwang-Mook Jung, Alessia Ligresti, Marco Allarà, Annemarieke G. J. Postmus, Samuele Maramai, Simone Brogi, Alessandro Papa, Gabriele Carullo, David Sykes, Dmitry Veprintsev, Stefano Federico, Alessandro Grillo, Bruno Di Guglielmo, Anna Ramunno, Anna Floor Stevens, Dominik Heer, Stefania Lamponi, Sandra Gemma, Jörg Benz, Vincenzo Di Marzo, Mario van der Stelt, Daniele Piomelli, Giuseppe Campiani

مصطلحات موضوعية: Biochemistry, Medicine, Cell Biology, Pharmacology, Biotechnology, Cancer, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, ray analyses combined, high eudysmic ratio, >- glycerol levels, selective monoacylglycerol lipase, new magl inhibitors, ), 5v , potent irreversible inhibitors, inhibitors based, irreversible ligands, >)-< b, (±)-< b, vivo <, vitro <, sn <, r <, h <, therapeutic potential, structural analysis, serine hydrolases, selected analogues, results suggest

الوقت: 4

العلاقة: https://figshare.com/articles/journal_contribution/Development_of_Potent_and_Selective_Monoacylglycerol_Lipase_Inhibitors_SARs_Structural_Analysis_and_Biological_Characterization/25033752Test

الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c01278.s001Test
https://figshare.com/articles/journal_contribution/Development_of_Potent_and_Selective_Monoacylglycerol_Lipase_Inhibitors_SARs_Structural_Analysis_and_Biological_Characterization/25033752Test

المؤلفون: Lulić Ana-Marija, Katalinić Maja

المصدر: Arhiv za Higijenu Rada i Toksikologiju, Vol 74, Iss 2, Pp 75-89 (2023)

مصطلحات موضوعية: catalytic dyad, lipid droplets, patatin, phospholipases, serine hydrolases, fosfolipaze, katalitička dijada, lipidne kapljice, serinske hidrolaze, Toxicology. Poisons, RA1190-1270

وصف الملف: electronic resource

العلاقة: https://doaj.org/toc/1848-6312Test

الوصول الحر: https://doaj.org/article/40e320c51d6b4da8ad4a83fa86b45ef6Test

المؤلفون: Tiantian Zhang, Feng Zhang, Yani Zhang, Hongxin Li, Guanghao Zhu, Taotao Weng, Cheng Huang, Ping Wang, Yuqi He, Jing Hu, Guangbo Ge

المصدر: Frontiers in Pharmacology, Vol 14 (2023)

مصطلحات موضوعية: alisol B 23-acetate, alisol B, human serum albumin (hSA), serine hydrolases, farnesoid X receptor (FXR), Therapeutics. Pharmacology, RM1-950

وصف الملف: electronic resource

العلاقة: https://www.frontiersin.org/articles/10.3389/fphar.2023.1160665/fullTest; https://doaj.org/toc/1663-9812Test

الوصول الحر: https://doaj.org/article/624075f4c5e74f53948b2fc6bc3017b3Test

المؤلفون: Abreha, Kibrom B., Alexandersson, Erik, Resjö, Svante, Lankinen, Åsa, Sueldo, Daniela, Kaschani, Farnusch, Kaiser, Markus, van der Hoorn, Renier A.L., Levander, Fredrik, Andreasson, Erik

المصدر: International Journal of Molecular Sciences. 22(21)

مصطلحات موضوعية: ABPP, Apoplast, Field-omics, Potato, Proteomics, Serine hydrolases, β-glycosidases, Lantbruksvetenskap och veterinärmedicin, Lantbruksvetenskap, skogsbruk och fiske, Jordbruksvetenskap, Agricultural Sciences, Agricultural Science, Forestry and Fisheries

الوصول الحر: https://lup.lub.lu.se/record/b856f67c-c999-48aa-ba29-18aa17701573Test
http://dx.doi.org/10.3390/ijms222112033Test

المؤلفون: Yedji, Rodrigue, S, Sohm, Bénédicte, Salnot, Virginie, Guillonneau, François, Cossu-Leguille, Carole, Battaglia, Eric

المساهمون: Laboratoire Interdisciplinaire des Environnements Continentaux (LIEC), Institut Ecologie et Environnement - CNRS Ecologie et Environnement (INEE-CNRS), Centre National de la Recherche Scientifique (CNRS)-Centre National de la Recherche Scientifique (CNRS)-Institut national des sciences de l'Univers (INSU - CNRS)-Observatoire Terre et Environnement de Lorraine (OTELo), Institut national des sciences de l'Univers (INSU - CNRS)-Université de Lorraine (UL)-Centre National de la Recherche Scientifique (CNRS)-Institut national des sciences de l'Univers (INSU - CNRS)-Université de Lorraine (UL)-Centre National de la Recherche Scientifique (CNRS), Institut Cochin (IC UM3 (UMR 8104 / U1016)), Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité), Plateforme protéomique 3P5 Institut Cochin (3P5), Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité)

المصدر: ISSN: 1661-6596.

مصطلحات موضوعية: zebrafish larvae serine hydrolases dibutyl phthalate activity-based protein profiling proteomics, zebrafish larvae, serine hydrolases, dibutyl phthalate, activity-based protein profiling, proteomics, [SDE]Environmental Sciences

العلاقة: hal-04078318; https://hal.univ-lorraine.fr/hal-04078318Test; https://hal.univ-lorraine.fr/hal-04078318/documentTest; https://hal.univ-lorraine.fr/hal-04078318/file/YEDJI%20el%20al%202022%20fusionn%C3%A9.pdfTest

الإتاحة: https://doi.org/10.3390/ijms232416060Test
https://hal.univ-lorraine.fr/hal-04078318Test
https://hal.univ-lorraine.fr/hal-04078318/documentTest
https://hal.univ-lorraine.fr/hal-04078318/file/YEDJI%20el%20al%202022%20fusionn%C3%A9.pdfTest

المؤلفون: Rodrigue S. Yedji, Bénédicte Sohm, Virginie Salnot, François Guillonneau, Carole Cossu-Leguille, Eric Battaglia

المصدر: International Journal of Molecular Sciences, Vol 23, Iss 24, p 16060 (2022)

مصطلحات موضوعية: zebrafish larvae, serine hydrolases, dibutyl phthalate, activity-based protein profiling, proteomics, Biology (General), QH301-705.5, Chemistry, QD1-999

وصف الملف: electronic resource

العلاقة: https://www.mdpi.com/1422-0067/23/24/16060Test; https://doaj.org/toc/1661-6596Test; https://doaj.org/toc/1422-0067Test

الوصول الحر: https://doaj.org/article/f91d5af7e5264cb48ce29a99d849fa1dTest

المؤلفون: Alexander T. Bakker (14312845), Ioli Kotsogianni (9930187), Liza Mirenda (14312848), Verena M. Straub (6713687), Mariana Avalos (14312851), Richard J. B. H. N. van den Berg (14312854), Bogdan I. Florea (1330800), Gilles P. van Wezel (7838948), Antonius P. A. Janssen (7449809), Nathaniel I. Martin (847378), Mario van der Stelt (222751)

مصطلحات موضوعية: Biochemistry, Pharmacology, Sociology, Virology, Environmental Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, target interaction landscape, revealed several cysteine, resistant staphylococcus aureus, novel antibacterial chemotype, identify novel antibiotics, high antibacterial potency, comparative chemical proteomics, mrsa phenotypic screening, data showcase oxadiazolones, phenotypic screen, targets responsible, situ competitive, serine hydrolases, resistance studies, relevant targets, powerful approach, polypharmacological mode, ones identified, often challenging, central role, based probe, adhe play

العلاقة: https://figshare.com/articles/journal_contribution/Chemical_Proteomics_Reveals_Antibiotic_Targets_of_Oxadiazolones_in_MRSA/21799438Test

الإتاحة: https://doi.org/10.1021/jacs.2c10819.s001Test

المؤلفون: Natascha Berger, Hanna Allerkamp, Christian Wadsack

المصدر: International Journal of Molecular Sciences; Volume 23; Issue 12; Pages: 6851

مصطلحات موضوعية: serine hydrolases, lipases, placenta, placental metabolism, pregnancy disorders

جغرافية الموضوع: agris

وصف الملف: application/pdf

العلاقة: Molecular Biology; https://dx.doi.org/10.3390/ijms23126851Test

الإتاحة: https://doi.org/10.3390/ijms23126851Test

المؤلفون: Stefan Rudolph (10802320), Helmut Dahlhaus (10802323), Walburga Hanekamp (831443), Christian Albers (1672666), Maximilian Barth (9550733), Giulia Michels (10802326), Denise Friedrich (10802329), Matthias Lehr (537954)

مصطلحات موضوعية: Biochemistry, Medicine, Microbiology, Physiology, Pharmacology, Biotechnology, Hematology, Infectious Diseases, Chemical Sciences not elsewhere classified, plasma albumin, BuChE, chemical reactivity, inhibition, compound, solution, serine hydrolases, carbamate oxygen, porcine blood plasma, Amide Hydrolase, MAGL, Monoacylglycerol Lipase, alkyl spacers, carbamate group, carbamate reactivity, esterases, pseudo-esterase activity, FAAH, aryl moieties, porcine liver homogenate, acid amide hydrolase

العلاقة: https://figshare.com/articles/journal_contribution/Aryl_i_N_i_-_6-Fluoroindol-1-yl_alkyl_carbamates_as_Inhibitors_of_Fatty_Acid_Amide_Hydrolase_Monoacylglycerol_Lipase_and_Butyrylcholinesterase_Structure_Activity_Relationships_and_Hydrolytic_Stability/14597131Test

الإتاحة: https://doi.org/10.1021/acsomega.1c01699.s001Test

المؤلفون: Michael S. Malamas (2148259), Spiro Pavlopoulos (2409385), Shakiru O. Alapafuja (2259457), Shrouq I. Farah (10702329), Alexander Zvonok (334031), Khadijah A. Mohammad (5775539), Jay West (3623987), Nicholas Thomas Perry (10702332), Dimitrios N. Pelekoudas (10702335), Girija Rajarshi (1350981), Christina Shields (10702338), Honrao Chandrashekhar (10702341), Jodi Wood (10702344), Alexandros Makriyannis (32548)

مصطلحات موضوعية: Biophysics, Biochemistry, Physiology, Pharmacology, Biotechnology, Immunology, Science Policy, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, Information Systems not elsewhere classified, Amidase Inhibitors N, plasma stability, lipid molecules, NAAA, structure-activity relationship studies, hydrolyzes lipid palmitoylethanolamide, 2 h, Acylethanolamine acid amidase, drug addiction, isothiocyanate pharmacophore, role, inflammation, pain processes, cysteine peptidases, serine hydrolases, pathophysiological conditions, nanomolar inhibitors, hNAAA

العلاقة: https://figshare.com/articles/journal_contribution/Design_and_Structure_Activity_Relationships_of_Isothiocyanates_as_Potent_and_Selective_i_N_i_Acylethanolamine-Hydrolyzing_Acid_Amidase_Inhibitors/14488947Test

الإتاحة: https://doi.org/10.1021/acs.jmedchem.1c00076.s001Test