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1دورية أكاديمية
المؤلفون: Xiaowei Huang, Fengbo Wu, Jing Ye, Lian Wang, Xiaoyun Wang, Xiang Li, Gu He
المصدر: Acta Pharmaceutica Sinica B, Vol 14, Iss 6, Pp 2402-2427 (2024)
مصطلحات موضوعية: Targeted protein degradation, Proteolysis targeting chimera, Endocytosis, Autophagy, Proximity-inducing modality, Post-translational modification, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2211383524000133Test; https://doaj.org/toc/2211-3835Test
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2دورية أكاديمية
المؤلفون: Wang, Yuxin, Morisseau, Christophe, Takamura, Akihiro, Wan, Debin, Li, Dongyang, Sidoli, Simone, Yang, Jun, Wolan, Dennis W, Hammock, Bruce D, Kitamura, Seiya
المصدر: ACS Chemical Biology. 18(4)
مصطلحات موضوعية: Biochemistry and Cell Biology, Medicinal and Biomolecular Chemistry, Chemical Sciences, Biological Sciences, Biotechnology, Cytosol, Epoxide Hydrolases, Proteolysis Targeting Chimera, Endoplasmic Reticulum Stress, Organic Chemistry, Biological sciences, Chemical sciences
وصف الملف: application/pdf
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3دورية أكاديمية
المؤلفون: Pance, Katarina, Gramespacher, Josef A, Byrnes, James R, Salangsang, Fernando, Serrano, Juan-Antonio C, Cotton, Adam D, Steri, Veronica, Wells, James A
المصدر: Nature biotechnology. 41(2)
مصطلحات موضوعية: Cell Membrane, Receptors, Cytokine, Interleukin-2, Signal Transduction, Chemokine CXCL12, Proteolysis, Proteolysis Targeting Chimera, Biotechnology, Generic health relevance
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/1bd0b1dmTest
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4دورية أكاديمية
المؤلفون: Yulu Zhang, Annan Ming, Junyan Wang, Wenmin Chen, Zhiqing Fang
المصدر: Pharmacological Research, Vol 205, Iss , Pp 107234- (2024)
مصطلحات موضوعية: Proteolysis targeting chimera (PROTAC), Castration-resistant prostate cancer (CRPC), Androgen receptor (AR), Cancer therapy, Drug target, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S1043661824001798Test; https://doaj.org/toc/1096-1186Test
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5دورية أكاديمية
المؤلفون: André T. S. Vicente, Jorge A. R. Salvador
المصدر: MedComm, Vol 5, Iss 6, Pp n/a-n/a (2024)
مصطلحات موضوعية: bifunctional molecule, degrader, hematological malignancy, leukemia, PROteolysis‐TArgeting Chimera (PROTAC), targeted protein degradation, Medicine
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2688-2663Test
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6دورية أكاديمية
المؤلفون: Tran, Nathan L, Leconte, Georges A, Ferguson, Fleur M
المصدر: Current Protocols. 2(12)
مصطلحات موضوعية: Biochemistry and Cell Biology, Biological Sciences, Biotechnology, Generic health relevance, Proteolysis, Proteins, PROTAC, compound optimization, medicinal chemistry, proteolysis-targeting chimera, targeted protein degradation
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/4bz2v5qhTest
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7دورية أكاديمية
المؤلفون: Katharina Hilbig, Russell Towers, Marc Schmitz, Martin Bornhäuser, Petra Lennig, Yixin Zhang
المصدر: Molecules, Vol 29, Iss 12, p 2779 (2024)
مصطلحات موضوعية: cyclophilin A (CypA), cyclosporin A (CsA), protein degradation, protein–protein interactions, proteolysis targeting chimera (PROTAC), Organic chemistry, QD241-441
وصف الملف: electronic resource
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8دورية أكاديمية
المؤلفون: Deborah Grifagni, Elena Lenci, Alessia De Santis, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni
مصطلحات موضوعية: Biophysics, Biochemistry, Molecular Biology, Pharmacology, Immunology, Developmental Biology, Cancer, Mental Health, Infectious Diseases, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, Information Systems not elsewhere classified, reversible covalent bond, proteolysis targeting chimera, crystallographic data complemented, cellular studies showed, pro sup, peptidomimetic molecule able, 3 ‑ chymotrypsin, cov ‑ 2, 2 3, peptidomimetic protacs, protac molecule, sulfur atom, study paves, pomalidomide moiety, pomalidomide cereblon, like protease, high degree, future applicability
الإتاحة: https://doi.org/10.1021/acsmedchemlett.3c00498.s001Test
https://figshare.com/articles/journal_contribution/Development_of_a_GC-376_Based_Peptidomimetic_PROTAC_as_a_Degrader_of_3_Chymotrypsin-like_Protease_of_SARS-CoV_2/24975448Test -
9دورية أكاديمية
المؤلفون: Mengdie Hu, Xiaomei Li, Lin Wang, Yanping Zhang, Yujie Sun, Hui Hua, Huina Liu, Ting Cai, Dongsheng Zhu, Qiuping Xiang
مصطلحات موضوعية: Biochemistry, Cell Biology, Molecular Biology, Pharmacology, Cancer, Chemical Sciences not elsewhere classified, ubiquitin – proteasome, proteolysis targeting chimera, attractive therapeutic strategy, attractive intervention strategy, dependent lipid peroxidation, significantly degraded gpx4, 5i b, thereby inducing ferroptosis, gpx4 inducing ferroptosis, inducing ferroptosis, dependent manner, ferroptosis presents, study provides, related diseases, prostate cancer, novel form, molecule degrader, human diseases, ht1080 cells, efforts led, degraders using, cancer cells, breast cancer, biological evaluation
الإتاحة: https://doi.org/10.1021/acsmedchemlett.3c00571.s001Test
https://figshare.com/articles/journal_contribution/ZX703_A_Small-Molecule_Degrader_of_GPX4_Inducing_Ferroptosis_in_Human_Cancer_Cells/25225797Test -
10دورية أكاديمية
المؤلفون: Aishwarya Saraswat, Richa Vartak, Rehab Hegazy, Yige Fu, Trishaal Janardhanam Raghavendra Rao, Blase Billack, Ketan Patel
المصدر: Biomedicine & Pharmacotherapy, Vol 168, Iss , Pp 115754- (2023)
مصطلحات موضوعية: Vemurafenib-resistant melanoma, PROteolysis-TArgeting Chimera, Myc, Self-nanoemulsifying drug delivery system, ARV-825, Bromo domain 4, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S0753332223015524Test; https://doaj.org/toc/0753-3322Test