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1دورية أكاديمية
المؤلفون: Zeren Sun, Lanjie Li, Bingxin Zhai, Mengxuan Hu, Lei Huang, Shihui Huang, Liu Ye, Xiangying Kong, Jie Xu, Jie Bai, Jingjie Yan, Qichen Zhou, Zheqi Hu, Yuchen Zhang, Yuhan Jiang, Yan Zhang, Zhou Qiao, Yi Zou, Yungen Xu, Qihua Zhu
مصطلحات موضوعية: Biochemistry, Cell Biology, Molecular Biology, Pharmacology, Biotechnology, Cancer, Hematology, Infectious Diseases, Astronomical and Space Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, present study describes, hct116or xenograft models, current therapeutic challenge, 2 nm ), met inhibitor crizotinib, parp1 inhibitor olaparib, met dual inhibitors, 50 sub, 16 b, parp1 inhibitors poses, parp1 inhibitors, small molecules, novel strategies, findings highlight, either alone, 3 nm
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2دورية أكاديمية
المصدر: Drug Design, Development and Therapy, Vol Volume 17, Pp 761-769 (2023)
مصطلحات موضوعية: scc244, c-met inhibitor, food effect, pharmacokinetics, safety, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: https://www.dovepress.com/effect-of-food-on-the-pharmacokinetics-and-safety-of-a-novel-cTest-met-inh-peer-reviewed-fulltext-article-DDDT; https://doaj.org/toc/1177-8881Test
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3دورية أكاديمية
المؤلفون: Alessandro Inno, Giuseppe Bogina, Giulio Settanni, Matteo Salgarello, Giovanni Foti, Carlo Pomari, Vincenzo Picece, Stefania Gori
المصدر: Drug Target Insights, Vol 17, Iss 1 (2023)
مصطلحات موضوعية: Elderly, First-line treatment, MET 14-exon skipping mutation, MET inhibitor, Non-small cell lung cancer, Tepotinib, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: https://aboutscience.archicoop.it/index.php/dti/article/view/2626Test; https://doaj.org/toc/1177-3928Test
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4دورية أكاديمية
المؤلفون: Bahar Karayel, Sena Durgun, Orhan Öcalgiray
المصدر: STEMedicine, Vol 4, Iss 3 (2023)
مصطلحات موضوعية: c-MET inhibitor, DE605, sorafenib, hepatocellular carcinoma, Medicine (General), R5-920, Biology (General), QH301-705.5
وصف الملف: electronic resource
العلاقة: https://stemedicine.org/index.php/stem/article/view/183Test; https://doaj.org/toc/2705-1188Test
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5دورية أكاديمية
المؤلفون: Sebastian Kraus
المصدر: Current Problems in Cancer: Case Reports, Vol 10, Iss , Pp 100230- (2023)
مصطلحات موضوعية: Chemotherapy, Clinical effectiveness, Intolerability, MET inhibitor, Real-world evidence, Neoplasms. Tumors. Oncology. Including cancer and carcinogens, RC254-282
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2666621923000157Test; https://doaj.org/toc/2666-6219Test
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6دورية أكاديمية
المؤلفون: Yongfeng Yu, Jianya Zhou, Xingya Li, Koichi Goto, Xuhong Min, Kazumi Nishino, Jiuwei Cui, Lin Wu, Jun Sakakibara, Yongqian Shu, Xiaorong Dong, Lu Li, Yasuto Yoneshima, Chengzhi Zhou, Xiaoling Li, Yiping Zhang, Dingzhi Huang, Aimin Zang, Wei Zhang, Xiuwen Wang, Li Zhang, Chong Bai, Jian Fang, Lejie Cao, Yanqiu Zhao, Yan Yu, Meiqi Shi, Diansheng Zhong, Fugen Li, Meng Li, Qiuxia Wu, Jun Zhou, Minghui Sun, Shun Lu
المصدر: EClinicalMedicine, Vol 59, Iss , Pp 101952- (2023)
مصطلحات موضوعية: Lung cancer, MET mutation, MET inhibitor, Medicine (General), R5-920
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2589537023001293Test; https://doaj.org/toc/2589-5370Test
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7دورية أكاديمية
المؤلفون: Zhuo-Xun Wu, Qiu-Xu Teng, Yuqi Yang, Nikita Acharekar, Jing-Quan Wang, Min He, Sabesan Yoganathan, Jun Lin, Jian Wang, Zhe-Sheng Chen
المصدر: Acta Pharmaceutica Sinica B, Vol 12, Iss 5, Pp 2609-2618 (2022)
مصطلحات موضوعية: MET inhibitor, Tepotinib, Multidrug resistance, ABCG2 transporter, Reversal agent, Combination treatment, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2211383521004901Test; https://doaj.org/toc/2211-3835Test
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8دورية أكاديمية
المؤلفون: Xiaorong Dong, MD, PhD, Xingya Li, MD, Jianhua Chen, MD, Shenglin Ma, MD, Deguang Mu, MD, Jie Hu, MD, PhD, Shun Lu, MD
المصدر: JTO Clinical and Research Reports, Vol 4, Iss 2, Pp 100449- (2023)
مصطلحات موضوعية: c-Met inhibitor, Lung cancer, HS-10241, Phase I, Solid tumors, Tyrosine kinase, Neoplasms. Tumors. Oncology. Including cancer and carcinogens, RC254-282
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2666364322001734Test; https://doaj.org/toc/2666-3643Test
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9دورية أكاديمية
المؤلفون: Yuichi Kumaki, Goshi Oda, Sadakatsu Ikeda
المصدر: Cancers, Vol 15, Iss 18, p 4552 (2023)
مصطلحات موضوعية: MET amplification, polysomy, aneuploidy, acquired resistance, MET inhibitor, Neoplasms. Tumors. Oncology. Including cancer and carcinogens, RC254-282
وصف الملف: electronic resource
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10دورية أكاديمية
المؤلفون: Kathryn M. Pflug, Dong W. Lee, Ashutosh Tripathi, Vytas A. Bankaitis, Kevin Burgess, Raquel Sitcheran
مصطلحات موضوعية: Medicine, Cell Biology, Pharmacology, Biotechnology, Cancer, Space Science, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, preclinical rodent model, inducing kinase activity, highly aggressive form, glioma progression glioblastoma, heptamethine cyanine dye, blood brain barrier, observed increased ir, newly diagnosed gbm, limited treatment options, impaired tumor growth, met inhibitor crizotinib, tumor localization, novel inhibitor, infrared dye, gbm growth, brain cancer, vivo <, vitro <, unconjugated crizotinib, poor prognosis, poor penetration, nuclear factor
الإتاحة: https://doi.org/10.1021/acs.molpharmaceut.3c00496.s001Test
https://figshare.com/articles/journal_contribution/Cyanine_Dye_Conjugation_Enhances_Crizotinib_Localization_to_Intracranial_Tumors_Attenuating_NF-_B-Inducing_Kinase_Activity_and_Glioma_Progression/24528455Test