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1دورية أكاديمية
المؤلفون: Zhipeng Zeng, Runcheng Tan, Shi Chen, Haolin Chen, Zhijia Liu, Lixin Liu, Mingqiang Li, Yongming Chen
المصدر: Acta Pharmaceutica Sinica B, Vol 14, Iss 6, Pp 2761-2772 (2024)
مصطلحات موضوعية: Diabetes, Insulin, Therapeutic index, Hypoglycemia, PEGylation, Receptor-mediated clearance, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2211383524000753Test; https://doaj.org/toc/2211-3835Test
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2دورية أكاديمية
المؤلفون: Yusuke Oka, Kumi Abe-Sato, Hideaki Tabuse, Yoshifumi Yasukawa, Tohru Yahara, Tomohiro Nishimoto, Masafumi Kamitani, Takuya Fukunaga, Nagahiro Ochiai, Tomoko Kumasaka-Abe, Kosuke Hitaka, Emi Gunji, Hiroki Ohara, Takuya Takeda, Naoki Kojima, Taiji Asami
مصطلحات موضوعية: Biochemistry, Cell Biology, Physiology, Pharmacology, Cancer, Environmental Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, based drug design, tp0628103 (< b, mediated clearance designed, mediated hepatic uptake, ip values culminated, mediated clearance, uptake based, hepatic uptake, systemic clearance, vivo <, vitro <, substrate recognition, studies revealed, pathophysiological processes, novel approach, molecular hybridization, isoelectric point, important role, highly potent
الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c01967.s001Test
https://figshare.com/articles/journal_contribution/Discovery_of_TP0628103_A_Highly_Potent_and_Selective_MMP_7_Inhibitor_with_Reduced_OATP-Mediated_Clearance_Designed_by_Shifting_Isoelectric_Points/24991010Test -
3دورية أكاديمية
المؤلفون: Shishir Singh (14334351), Mateo Murillo-León (14334354), Niklas Sebastian Endres (14334357), Ailan Farid Arenas Soto (14334360), Jorge Enrique Gómez-Marín (7857968), Florence Melbert (14334363), Thirumala-Devi Kanneganti (62745), Masahiro Yamamoto (39398), Claudia Campos (8137581), Jonathan Charles Howard (14334366), Gregory Alan Taylor (14334369), Tobias Steinfeldt (154465)
مصطلحات موضوعية: Biochemistry, Microbiology, Immunology, Cancer, Infectious Diseases, Environmental Sciences not elsewhere classified, Physical Sciences not elsewhere classified, parasitophorous vacuolar membrane, inhibits homodimer formation, direct interaction partners, pvm integrity rescues, polymorphic rhoptry proteins, zoonotic apicomplexan parasite, irg resistance system, toxoplasma gondii <, specific parasite effector, irg proteins, specific inactivation, pvm ), gondii <, irg protein, yet unknown, vivo <, vitro <, study identifies, small rodents, related gtpases, overall reduction, one third, mediated clearance
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4دورية أكاديمية
المؤلفون: Shishir Singh (14334351), Mateo Murillo-León (14334354), Niklas Sebastian Endres (14334357), Ailan Farid Arenas Soto (14334360), Jorge Enrique Gómez-Marín (7857968), Florence Melbert (14334363), Thirumala-Devi Kanneganti (62745), Masahiro Yamamoto (39398), Claudia Campos (8137581), Jonathan Charles Howard (14334366), Gregory Alan Taylor (14334369), Tobias Steinfeldt (154465)
مصطلحات موضوعية: Biochemistry, Microbiology, Immunology, Cancer, Infectious Diseases, Environmental Sciences not elsewhere classified, Physical Sciences not elsewhere classified, parasitophorous vacuolar membrane, inhibits homodimer formation, direct interaction partners, pvm integrity rescues, polymorphic rhoptry proteins, zoonotic apicomplexan parasite, irg resistance system, toxoplasma gondii <, specific parasite effector, irg proteins, specific inactivation, pvm ), gondii <, irg protein, yet unknown, vivo <, vitro <, study identifies, small rodents, related gtpases, overall reduction, one third, mediated clearance
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5دورية أكاديمية
المؤلفون: Shishir Singh (14334351), Mateo Murillo-León (14334354), Niklas Sebastian Endres (14334357), Ailan Farid Arenas Soto (14334360), Jorge Enrique Gómez-Marín (7857968), Florence Melbert (14334363), Thirumala-Devi Kanneganti (62745), Masahiro Yamamoto (39398), Claudia Campos (8137581), Jonathan Charles Howard (14334366), Gregory Alan Taylor (14334369), Tobias Steinfeldt (154465)
مصطلحات موضوعية: Biochemistry, Microbiology, Immunology, Cancer, Infectious Diseases, Environmental Sciences not elsewhere classified, Physical Sciences not elsewhere classified, parasitophorous vacuolar membrane, inhibits homodimer formation, direct interaction partners, pvm integrity rescues, polymorphic rhoptry proteins, zoonotic apicomplexan parasite, irg resistance system, toxoplasma gondii <, specific parasite effector, irg proteins, specific inactivation, pvm ), gondii <, irg protein, yet unknown, vivo <, vitro <, study identifies, small rodents, related gtpases, overall reduction, one third, mediated clearance
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6دورية أكاديمية
المؤلفون: Shishir Singh (14334351), Mateo Murillo-León (14334354), Niklas Sebastian Endres (14334357), Ailan Farid Arenas Soto (14334360), Jorge Enrique Gómez-Marín (7857968), Florence Melbert (14334363), Thirumala-Devi Kanneganti (62745), Masahiro Yamamoto (39398), Claudia Campos (8137581), Jonathan Charles Howard (14334366), Gregory Alan Taylor (14334369), Tobias Steinfeldt (154465)
مصطلحات موضوعية: Biochemistry, Microbiology, Immunology, Cancer, Infectious Diseases, Environmental Sciences not elsewhere classified, Physical Sciences not elsewhere classified, parasitophorous vacuolar membrane, inhibits homodimer formation, direct interaction partners, pvm integrity rescues, polymorphic rhoptry proteins, zoonotic apicomplexan parasite, irg resistance system, toxoplasma gondii <, specific parasite effector, irg proteins, specific inactivation, pvm ), gondii <, irg protein, yet unknown, vivo <, vitro <, study identifies, small rodents, related gtpases, overall reduction, one third, mediated clearance
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7دورية أكاديمية
المؤلفون: Shishir Singh (14334351), Mateo Murillo-León (14334354), Niklas Sebastian Endres (14334357), Ailan Farid Arenas Soto (14334360), Jorge Enrique Gómez-Marín (7857968), Florence Melbert (14334363), Thirumala-Devi Kanneganti (62745), Masahiro Yamamoto (39398), Claudia Campos (8137581), Jonathan Charles Howard (14334366), Gregory Alan Taylor (14334369), Tobias Steinfeldt (154465)
مصطلحات موضوعية: Biochemistry, Microbiology, Immunology, Cancer, Infectious Diseases, Environmental Sciences not elsewhere classified, Physical Sciences not elsewhere classified, parasitophorous vacuolar membrane, inhibits homodimer formation, direct interaction partners, pvm integrity rescues, polymorphic rhoptry proteins, zoonotic apicomplexan parasite, irg resistance system, toxoplasma gondii <, specific parasite effector, irg proteins, specific inactivation, pvm ), gondii <, irg protein, yet unknown, vivo <, vitro <, study identifies, small rodents, related gtpases, overall reduction, one third, mediated clearance
العلاقة: https://figshare.com/articles/journal_contribution/Immunoreagents_used_in_this_study_/21824052Test
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8دورية أكاديمية
المؤلفون: Tina M. Tagmose (2715901), Karen-Margrethe Pedersen (12029890), Lone Pridal (2375119), Carsten E. Stidsen (9193879), Marie Ø. Pedersen (2245372), Zhaosheng Lin (12029893), Yuanyuan Zhang (101797), Zhe Wan (74018), Mercedes Ferreras (12029896), Helle Naver (10745027), Peter K. Nielsen (2684311), Zheng Cao (562710), Yi Wang (32470), Lennart Lykke (1766620), Josefine L. Christensen (12029899), Victoria S. Jensen (12029902), Valentina Manfè (9920942), Thomas Å. Pedersen (12029905), Eva Johansson (335751), Peter Madsen (2242984), János T. Kodra (2375125), Martin Münzel (1485277), Leonardo De Maria (416956), Erica Nishimura (197646), Thomas B. Kjeldsen (10745024)
مصطلحات موضوعية: Biophysics, Biochemistry, Genetics, Molecular Biology, Physiology, Pharmacology, Biotechnology, Immunology, Cancer, Virology, Computational Biology, Chemical Sciences not elsewhere classified, disulfide bond within, amino acid substitutions, long acting two, neonatal fc receptor, fc conjugation leads, long pharmacokinetic profile, insulin receptor affinity, describe molecular engineering, long pharmacokinetic, molecular engineering, fc molecule, fc element, fc conjugates, molecular size, pharmacodynamic profiles, mediated clearance, lysine residue, efficacious mono
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9دورية أكاديمية
المؤلفون: Andrew P. Degnan (1445947), Godwin K. Kumi (10168566), Christopher W. Allard (6240908), Erika V. Araujo (10168569), Walter L. Johnson (10168572), Kurt Zimmermann (327735), Bradley C. Pearce (2360980), Steven Sheriff (1601854), Alan Futran (9387879), Xin Li (51274), Gregory A. Locke (5941769), Dan You (1551370), John Morrison (91443), Karen E. Parrish (10168575), Caitlyn Stromko (10168578), Anwar Murtaza (6508505), Jinqi Liu (288494), Benjamin M. Johnson (1705429), Gregory D. Vite (1436365), Mark D. Wittman (2332546)
مصطلحات موضوعية: Biochemistry, Medicine, Cell Biology, Molecular Biology, Pharmacology, Immunology, Cancer, Infectious Diseases, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, T-cell receptor, Hematopoetic progenitor kinase 1, syngeneic tumor model, plasma protein binding, immune-mediated clearance, checkpoint inhibitors, compound 24, alternative mechanisms, Oral administration, colorectal cancer, TCR, serine-threonine kinase, response, Selective Inhibitors, structure-based discovery, HPK 1. Optimization, anti-PD 1 efficacy, anti-PD 1 antibody
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10صورة
المؤلفون: Shishir Singh (14334351), Mateo Murillo-León (14334354), Niklas Sebastian Endres (14334357), Ailan Farid Arenas Soto (14334360), Jorge Enrique Gómez-Marín (7857968), Florence Melbert (14334363), Thirumala-Devi Kanneganti (62745), Masahiro Yamamoto (39398), Claudia Campos (8137581), Jonathan Charles Howard (14334366), Gregory Alan Taylor (14334369), Tobias Steinfeldt (154465)
مصطلحات موضوعية: Biochemistry, Microbiology, Immunology, Cancer, Infectious Diseases, Environmental Sciences not elsewhere classified, Physical Sciences not elsewhere classified, parasitophorous vacuolar membrane, inhibits homodimer formation, direct interaction partners, pvm integrity rescues, polymorphic rhoptry proteins, zoonotic apicomplexan parasite, irg resistance system, toxoplasma gondii <, specific parasite effector, irg proteins, specific inactivation, pvm ), gondii <, irg protein, yet unknown, vivo <, vitro <, study identifies, small rodents, related gtpases, overall reduction, one third, mediated clearance