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1مؤتمر
المساهمون: CIRM - Centre Interdisciplinaire de Recherche sur le Médicament - ULiège
المصدر: CIRM Day, Liège, Belgium [BE], 2 février 2022
مصطلحات موضوعية: AMPA receptors, Alzeimer's disease, AMPA positive allosteric modulators, AMPA, Receptors, Glutamate, Alzeimer, Positive allosteric modulators, neurodegenerative diseases, BPAM344, Human health sciences, Pharmacy, pharmacology & toxicology, Sciences de la santé humaine, Pharmacie, pharmacologie & toxicologie
الوصول الحر: https://orbi.uliege.be/handle/2268/303008Test
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2دورية أكاديمية
المؤلفون: Genaro, K, Doan, B, Johnstone, T, Gee, Kelvin, Yoshimura, Ryan, Hogenkamp, Derk
مصطلحات موضوعية: Morphine-antinociceptive tolerance, Opioid, Opioid withdrawal symptoms, Positive allosteric modulators, δ-subunit GABA(A) receptor, Analgesics, Analgesics, Opioid, Animals, Dose-Response Relationship, Drug, Female, Humans, Male, Mice, Mice, Knockout, Morphine, Receptors, GABA-A, Receptors, Opioid, delta, Water, gamma-Aminobutyric Acid
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/9hp497vmTest
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3دورية أكاديمية
المؤلفون: Chunhao Zhu, Xiaobing Lan, Zhiqiang Wei, Jianqiang Yu, Jian Zhang
المصدر: Acta Pharmaceutica Sinica B, Vol 14, Iss 1, Pp 67-86 (2024)
مصطلحات موضوعية: Neuropathic pain, Allosteric modulators, G protein-coupled receptors, Analgesia, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2211383523002824Test; https://doaj.org/toc/2211-3835Test
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4دورية أكاديمية
المؤلفون: Robert J. Richardson, Steven Petrou, Alexander Bryson
المصدر: Frontiers in Pharmacology, Vol 15 (2024)
مصطلحات موضوعية: benzodiazepines, epilepsy, GABA A receptor, GABA allosteric modulators a, neurosteriod, antisense, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: https://www.frontiersin.org/articles/10.3389/fphar.2024.1341472/fullTest; https://doaj.org/toc/1663-9812Test
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5دورية أكاديمية
المؤلفون: Leonardo Brunetti, Fabio Francavilla, Marcello Leopoldo, Enza Lacivita
المصدر: Pharmaceuticals, Vol 17, Iss 6, p 695 (2024)
مصطلحات موضوعية: serotonin, GPCR, natural compounds, allosteric modulators, cannabinoids, Medicine, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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6رسالة جامعية
المؤلفون: Hilšer, Anna
المساهمون: Ladds, Graham
مصطلحات موضوعية: GPCR, pharmacology, diabetes, obesity, allosteric modulators, AR agonists, AR antagonists, GIPR
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7دورية أكاديمية
المؤلفون: Hoang Nguyen, Mary Hongying Cheng, Ji Young Lee, Shaili Aggarwal, Ole Valente Mortensen, Ivet Bahar
المصدر: Current Research in Physiology, Vol 7, Iss , Pp 100125- (2024)
مصطلحات موضوعية: Dopamine transporter, Serotonin transporter, Reuptake inhibitors, Allosteric modulators, Elastic network models, Ligand-binding sites, Physiology, QP1-981, Specialties of internal medicine, RC581-951
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2665944124000099Test; https://doaj.org/toc/2665-9441Test
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8دورية أكاديمية
المؤلفون: Chenxia Yang, Ying Meng, Xintong Wang, Xin Li, Tong Yu, Weiming Liao, Wenjun Xie, Qianchen Jiang, Han Wang, Cheng Shi, Wenxuan Jiao, Xiling Bian, Fang Hu, Xiaowei Wang, Yani Liu, Liangren Zhang, KeWei Wang, Qi Sun
مصطلحات موضوعية: Biochemistry, Medicine, Neuroscience, Physiology, Pharmacology, Biotechnology, Mental Health, Chemical Sciences not elsewhere classified, exhibits potent activation, representative atypical type, positive allosteric modulators, methyl group results, 100 μm ), 9 b, 7b b, 6p b, maximum activation effect, 50 sub, allosteric activation, xenopus <, typical type, max effect, amino group, 3 μm, α7 currents, therapeutic strategy, mouse schizophrenia, like model, cognitive disorders, cognitive deficits
الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c02323.s001Test
https://figshare.com/articles/journal_contribution/Allosteric_Activation_of_7_Nicotinic_Acetylcholine_Receptors_by_Novel_2_Arylamino-thiazole-5-carboxylic_Acid_Amide_Derivatives_for_the_Improvement_of_Cognitive_Deficits_in_Mice/25276604Test -
9دورية أكاديمية
المؤلفون: Balázs Krámos, Zsuzsa Hadady, Attila Makó, Gábor Szántó, Nóra Felföldi, Ildikó Magdó, Amrita Ágnes Bobok, Imre Bata, Viktor Román, András Visegrády, György M. Keserű, István Greiner, János Éles
مصطلحات موضوعية: Biophysics, Biochemistry, Genetics, Molecular Biology, Pharmacology, Immunology, Cancer, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, protein structure selecting, positive allosteric modulators, perfectly explained based, new protein structures, lead candidate offers, known hts hit, >] pyrimidine core, novel carboxyl feature, lipophilic ligand efficiency, b sub, receptor using, primary goal, physicochemical properties, pam pharmacophore, objective function, important element, binding mode, 5 -<
الإتاحة: https://doi.org/10.1021/acsmedchemlett.3c00560.s001Test
https://figshare.com/articles/journal_contribution/Novel-Type_GABA_sub_B_sub_PAMs_Structure_Activity_Relationship_in_Light_of_the_Protein_Structure/25324945Test -
10دورية أكاديمية
المؤلفون: Francotte, Pierre, Bay, Yasmin, Goffin, Eric, Colson, Thomas, Lesenfants, Cindy, Dorosz, Jerzy, Laulumaa, Saara, Fraikin, Pierre, De Tullio, Pascal, Beaufour, Caroline, Botez, Iuliana, Pickering, Darryl, Frydenvang, Karla, Danober, Laurence, Skov Kristensen, Anders, Sandholm Kastrup, Jette, Pirotte, Bernard
المصدر: European Journal of Medicinal Chemistry, 264, 116036 (2023-12-09)
مصطلحات موضوعية: Ionotropic glutamate receptors Positive allosteric modulators thieno[3, 2-e]-1, 2, 4-thiadiazine 1, 1-dioxides 1, 4-Benzothiadiazine 1, 1-dioxides X-ray crystallography Calcium-sensitive fluorescence-based assay, Organic Chemistry, Drug Discovery, Pharmacology, General Medicine, Human health sciences, Pharmacy, pharmacology & toxicology, Physical, chemical, mathematical & earth Sciences, Chemistry, Sciences de la santé humaine, Pharmacie, pharmacologie & toxicologie, Physique, chimie, mathématiques & sciences de la terre, Chimie
العلاقة: https://api.elsevier.com/content/article/PII:S0223523423010036?httpAccept=text/xmlTest; urn:issn:0223-5234; urn:issn:1768-3254
الوصول الحر: https://orbi.uliege.be/handle/2268/312961Test