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1دورية أكاديميةIdentification of New EGFR Inhibitors by Structure-Based Virtual Screening and Biological Evaluation
المؤلفون: Shuyi Wang, Xiaotian Xu, Chuxin Pan, Qian Guo, Qinlan Li, Shanhe Wan, Zhonghuang Li, Jiajie Zhang, Xiaoyun Wu
المصدر: International Journal of Molecular Sciences, Vol 25, Iss 3, p 1887 (2024)
مصطلحات موضوعية: epidermal growth factor receptor (EGFR), virtual screening, molecular dynamics, Biology (General), QH301-705.5, Chemistry, QD1-999
وصف الملف: electronic resource
العلاقة: https://www.mdpi.com/1422-0067/25/3/1887Test; https://doaj.org/toc/1661-6596Test; https://doaj.org/toc/1422-0067Test
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2دورية أكاديمية
المؤلفون: Ying Jiang, Chunhui Huang, Yaqi Huang, Lifan Long, Guowu Wu, Fengqiu Guo, Chuan Huang, Siming Liu, Zhengguang Zhu, Shaoyu Wu, Zhonghuang Li, Jiajie Zhang, Shanhe Wan
المصدر: Pharmaceutics, Vol 15, Iss 5, p 1501 (2023)
مصطلحات موضوعية: SMUZ106, epidermal growth factor receptor (EGFR), glioblastoma (GBM), EGFRvIII, temozolomide-resistance, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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3دورية أكاديميةCombined 3D-QSAR and Docking Modelling Study on Indolocarbazole Series Compounds as Tie-2 Inhibitors
المؤلفون: Yuanxin Tian, Jiajie Zhang, Zhengguang Zhu, Shuguang Wu, Jian Xu, Zhonghuang Li
المصدر: International Journal of Molecular Sciences, Vol 12, Iss 8, Pp 5080-5097 (2011)
مصطلحات موضوعية: Tie-2 kinase inhibitor, 3D-QSAR, CoMFA, CoMSIA, docking, Biology (General), QH301-705.5, Chemistry, QD1-999
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Yu Fu, Yuanyuan Wang, Shanhe Wan, Zhonghuang Li, Guangfa Wang, Jiajie Zhang, Xiaoyun Wu
المصدر: Molecules, Vol 22, Iss 4, p 542 (2017)
مصطلحات موضوعية: DFG-out, pan-RAF inhibitor, 1H-pyrazolo[3,4-d]pyrimidine derivatives, biological activities, molecular docking, molecular dynamics simulation, Organic chemistry, QD241-441
وصف الملف: electronic resource
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5دورية أكاديمية
المؤلفون: Yangcheng Ai (14394757), Zichao Yang (2002318), Zilong Yang (14394760), Shanhe Wan (3875341), Chunhui Huang (1505923), Chuan Huang (755258), Mingxia Li (547512), Zhonghuang Li (4382497), Jiajie Zhang (43131), Tingting Zhang (264633)
مصطلحات موضوعية: Biophysics, Biochemistry, Molecular Biology, Pharmacology, Biotechnology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, study could enhance, withdrawing substituents introduced, electrophilic group cyanoacrylamide, different electrophilic substituents, results might help, molecular dynamics simulations, reversible noncovalent inhibitors, α sub, withdrawing groups play, kinase assay experiment, reversible covalent inhibitors, withdrawing groups, electrophilic groups, covalent inhibitors, results suggested, molecular docking, egfr inhibitors, warheads reacting, structural information, steric complementarity, specific interactions, reverse β, olefin bond
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6
المؤلفون: Yangcheng Ai, Zichao Yang, Zilong Yang, Shanhe Wan, Chunhui Huang, Chuan Huang, Mingxia Li, Zhonghuang Li, Jiajie Zhang, Tingting Zhang
المصدر: Journal of Chemical Information and Modeling. 63:493-506
مصطلحات موضوعية: General Chemical Engineering, General Chemistry, Library and Information Sciences, Computer Science Applications
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::abc7afa735119debe6114d505eaa31a5Test
https://doi.org/10.1021/acs.jcim.2c00458Test -
7دورية أكاديمية
المؤلفون: Xiaoyun Wu (179670), Qian Guo (107009), Qinlan Li (9999324), Shanhe Wan (3875341), Zhonghuang Li (4382497), Jiajie Zhang (43131)
مصطلحات موضوعية: Biochemistry, Medicine, Cell Biology, Pharmacology, Biotechnology, Developmental Biology, Cancer, Hematology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, EGFR, allosteric inhibitor, EAI045, JBJ-04-125-02, molecular dynamics
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8
المؤلفون: Zichao, Yang, Yangcheng, Ai, Shanhe, Wan, Zilong, Yang, Honghao, Li, Zhonghuang, Li, Chunhui, Huang, Lishun, Zhang, Mingxia, Li, Jiajie, Zhang, Tingting, Zhang
المصدر: Bioorganic & Medicinal Chemistry. 74:117069
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Parkinson Disease, Biochemistry, Neuroblastoma, Neuroprotective Agents, Blood-Brain Barrier, Cell Line, Tumor, Benzamides, Drug Discovery, Animals, Humans, Molecular Medicine, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aed01af4f7abae77865052afa0176f94Test
https://doi.org/10.1016/j.bmc.2022.117069Test -
9
المؤلفون: Qinlan Li, Qian Guo, Shuyi Wang, Shanhe Wan, Zhonghuang Li, Jiajie Zhang, Xiaoyun Wu
المصدر: SSRN Electronic Journal.
مصطلحات موضوعية: Pharmacology, Acrylamides, History, Lung Neoplasms, Polymers and Plastics, Organic Chemistry, General Medicine, Industrial and Manufacturing Engineering, ErbB Receptors, Pyrimidines, Drug Resistance, Neoplasm, Carcinoma, Non-Small-Cell Lung, Cell Line, Tumor, Drug Discovery, Mutation, Proteolysis, Humans, Business and International Management, Protein Kinase Inhibitors, Cell Proliferation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::71ba1ea4873189c63613df8b707f06d3Test
https://doi.org/10.2139/ssrn.4051300Test -
10
المؤلفون: Yuanxin Tian, Jianxin Pang, Xinhua Chen, Jiajie Zhang, Jiajun Luo, Ting Wu, Zean Zhao, Shan Chang, Yudong Shen, Zhonghuang Li, Shanhe Wan
المصدر: Bioorganic chemistry. 117
مصطلحات موضوعية: Male, Scaffold, Organic Cation Transport Proteins, Organic Anion Transporters, Mice, Inbred Strains, Computational biology, Hyperuricemia, Biochemistry, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Docking (dog), In vivo, Drug Discovery, medicine, Animals, Medicine, Chinese Traditional, Molecular Biology, IC50, Virtual screening, Biological Products, Natural product, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, medicine.disease, Flavones, Gout, Molecular Docking Simulation, chemistry, Drugs, Chinese Herbal
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c87c7b8a32c8dc555a8a5a67ba873440Test
https://pubmed.ncbi.nlm.nih.gov/34775203Test