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1
المؤلفون: James C. Hershey, Youheng Shu, Cheng Wang, Julie A. O'Brien, Vanita Puri, Tracy L. Diamond, Shaei Huang, Antonella Converso, Brian C. Magliaro, Jason M. Uslaner, Victor N. Uebele, Kelly-Ann S. Schlegel
المصدر: Bioorganicmedicinal chemistry letters. 30(9)
مصطلحات موضوعية: High-throughput screening, Clinical Biochemistry, Allosteric regulation, Scopolamine, Pharmaceutical Science, Glutamic Acid, Receptors, Metabotropic Glutamate, Biochemistry, Mice, Structure-Activity Relationship, In vivo, Drug Discovery, Animals, Binding site, Amino Acids, Receptor, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Amphetamines, Glutamate receptor, Bridged Bicyclo Compounds, Heterocyclic, High-Throughput Screening Assays, Molecular Medicine, Metabotropic glutamate receptor 2, Antagonism, Neuroscience, Adjuvants, Anesthesia
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::60318faea5edce68a4bf4762b8f54575Test
https://pubmed.ncbi.nlm.nih.gov/32173198Test -
2
المؤلفون: William A. Kinney, Barry S. Selinsky, Youheng Shu, Stephen R Jones
المصدر: Steroids. 67:291-304
مصطلحات موضوعية: Staphylococcus aureus, Magnetic Resonance Spectroscopy, Stereochemistry, Clinical Biochemistry, Stigmasterol, Substituent, Spermine, Stereoisomerism, Biology, Hydroxylation, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Endocrinology, Anti-Infective Agents, Squalus acanthias, Candida albicans, Escherichia coli, Animals, Structure–activity relationship, Molecular Biology, Pharmacology, Cholestanes, Molecular Structure, Organic Chemistry, Antimicrobial, Anti-Bacterial Agents, chemistry, Dogfish, Squalamine, Pseudomonas aeruginosa, Cholestanols
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cad44dbb16504387f6816d09279c2f7bTest
https://doi.org/10.1016/s0039-128xTest(01)00161-1 -
3
المؤلفون: Wong Michael K C, Yueheng Jiang, Qingbei Zeng, Chung-Her Jenh, Stuart B. Rosenblum, De-Yi Yang, Yuefei Shao, Anilkumar G. Nair, Jingqi Duo, Doug W. Hobbs, Brian F. Mcguinness, Joseph A. Kozlowski, Lisa Guise Zawacki, Neng-Yang Shih, Carolyn DiIanni Carroll, Youheng Shu, Seong Heon Kim
المصدر: Bioorganicmedicinal chemistry letters. 24(4)
مصطلحات موضوعية: Receptors, CXCR3, Metabolite, Clinical Biochemistry, hERG, Pharmaceutical Science, CXCR3, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Heterocyclic Compounds, Amide, Drug Discovery, Animals, Humans, Molecular Biology, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Combinatorial chemistry, Amides, Ether-A-Go-Go Potassium Channels, Rats, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::126a3924ad6c61b713b4a73725849822Test
https://pubmed.ncbi.nlm.nih.gov/24486132Test -
4
المصدر: Bioorganicmedicinal chemistry letters. 23(11)
مصطلحات موضوعية: Stereochemistry, Spermidine, Clinical Biochemistry, Substituent, Phospholipid, Pharmaceutical Science, Spermine, Microbial Sensitivity Tests, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Escherichia coli, Molecular Biology, Vesicle, Organic Chemistry, Stereoisomerism, Sterol, Anti-Bacterial Agents, chemistry, Squalamine, Liposomes, Pseudomonas aeruginosa, Molecular Medicine, Polyamine, Cholestanols
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::94f5ab24849d3110e54482543a7011cdTest
https://pubmed.ncbi.nlm.nih.gov/23618624Test -
5
المؤلفون: Gopinadhan N. Anilkumar, Qingbei Zeng, Brian F. Mcguinness, Chung-Her Jenh, Guizhen Dong, Lisa Guise Zawacki, Inna Schulman, Yueheng Jiang, Seong Heon Kim, Yuefei Shao, Youheng Shu, Wong Michael K C, Doug W. Hobbs, Stuart B. Rosenblum, Neng-Yang Shih, James W. Hall, Carolyn DiIanni Carroll, Wensheng Yu, Joseph A. Kozlowski
المصدر: Bioorganicmedicinal chemistry letters. 21(5)
مصطلحات موضوعية: Receptors, CXCR3, Stereochemistry, medicine.drug_class, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CXCR3, Biochemistry, Piperazines, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, stomatognathic system, Piperidines, immune system diseases, Drug Discovery, medicine, Moiety, Humans, skin and connective tissue diseases, Receptor, Molecular Biology, IC50, Piperazine, Molecular Structure, Organic Chemistry, Antagonist, hemic and immune systems, In vitro, stomatognathic diseases, chemistry, Molecular Medicine, Piperidine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9894b320a60ce2053010ea1122688132Test
https://pubmed.ncbi.nlm.nih.gov/21277198Test -
6
المؤلفون: Cindy E. Nuss, John J. Renger, Thomas S. Reger, Jeanine E. Ballard, Thomayant Prueksaritanont, Susan L. Garson, Mark G. Bock, Youheng Shu, Yuxing Li, Zhi Qiang Yang, Richard L. Kraus, Scott M. Doran, Kenneth E. Rittle, Victor N. Uebele, Rowena V. Cube, Cuyue Tang, Phung Bondiskey, Schlegel Kelly-Ann, Yuhsin Kuo, Steven V. Fox, James C. Barrow, George D. Hartman
المصدر: Bioorganicmedicinal chemistry letters. 20(17)
مصطلحات موضوعية: medicine.medical_specialty, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Biological Availability, Biochemistry, Chemical synthesis, Calcium Channels, T-Type, Structure-Activity Relationship, In vivo, Internal medicine, Drug Discovery, medicine, Potency, Animals, Humans, Molecular Biology, Chromatography, High Pressure Liquid, Quinazolinones, Chemistry, Calcium channel, Organic Chemistry, T-type calcium channel, Antagonist, Biological activity, Haplorhini, Calcium Channel Blockers, Rats, Endocrinology, Anticonvulsant, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4ac8391014bf59598c5815986f43767Test
https://pubmed.ncbi.nlm.nih.gov/20673719Test -
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المؤلفون: Len Favreau, Chunli Huang, Guowei Zhou, Neng-Yang Shih, Waldemar Gonsiorek, R. William Hipkin, Charles A. Lunn, Ling Tong, Joseph A. Kozlowski, Joseph Kelly, Lei Chen, Brian J. Lavey, Asra Malikzay, Razia Rizvi, Eric J. Gilbert, Bandarpalle B. Shankar, Daniel Lundell, Wong Michael K C, Stuart W. McCombie, Youhao Dong, Youheng Shu
المصدر: Bioorganicmedicinal chemistry letters. 20(2)
مصطلحات موضوعية: Drug Inverse Agonism, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ring (chemistry), Biochemistry, Chemical synthesis, Sulfone, Receptor, Cannabinoid, CB2, chemistry.chemical_compound, Structure-Activity Relationship, Cytochrome P-450 Enzyme System, Piperidines, Drug Discovery, Moiety, Structure–activity relationship, Animals, Humans, Sulfones, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Aryl, Organic Chemistry, Sulfonamide, Rats, chemistry, Molecular Medicine, Piperidine, Calcium Channels
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dbdfe23991c9196dd275858b3d1c234Test
https://pubmed.ncbi.nlm.nih.gov/20005710Test -
8
المؤلفون: Guowei Zhou, Stuart W. McCombie, Neng-Yang Shih, De-Yi Yang, Bandarpalle B. Shankar, Youheng Shu, Razia Rizvi, Spitler James M, Brian J. Lavey, Michael K. C. Wong, Charles A. Lunn, Jie Wu, Joseph A. Kozlowski, Shing-Chun Wong, Ronald L. Wolin
المصدر: Bioorganicmedicinal chemistry letters. 17(13)
مصطلحات موضوعية: Cannabinoid receptor, Stereochemistry, medicine.medical_treatment, Chemistry, Pharmaceutical, Receptors, Drug, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Ligands, Biochemistry, Chemical synthesis, Sulfone, Receptor, Cannabinoid, CB2, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Inverse agonist, Structure–activity relationship, Animals, Sulfones, Molecular Biology, chemistry.chemical_classification, Organic Chemistry, Sodium, Sulfonamide, Rats, Kinetics, chemistry, Models, Chemical, Drug Design, Molecular Medicine, lipids (amino acids, peptides, and proteins), Cannabinoid, Selectivity, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ea56397b323077382995272baf1958eeTest
https://pubmed.ncbi.nlm.nih.gov/17466519Test -
9دورية أكاديمية
المؤلفون: Zhi-Qiang Yang, James C. Barrow, William D. Shipe, Kelly-Ann S. Schlegel, Youheng Shu, F. Vivien Yang, Craig W. Lindsley, Kenneth E. Rittle, Mark G. Bock, George D. Hartman, Victor N. Uebele, Cindy E. Nuss, Steve V. Fox, Richard L. Kraus, Scott M. Doran, Thomas M. Connolly, Cuyue Tang, Jeanine E. Ballard, Yuhsin Kuo, Emily D. Adarayan
المصدر: Journal of Medicinal Chemistry; Oct2008, Vol. 51 Issue 20, p6471-6477, 7p
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10دورية أكاديمية
المؤلفون: William D. Shipe, James C. Barrow, Zhi-Qiang Yang, Craig W. Lindsley, F. Vivien Yang, Kelly-Ann S. Schlegel, Youheng Shu, Kenneth E. Rittle, Mark G. Bock, George D. Hartman, Cuyue Tang, Jeanine E. Ballard, Yuhsin Kuo, Emily D. Adarayan, Thomayant Prueksaritanont, Matthew M. Zrada, Victor N. Uebele, Cindy E. Nuss, Thomas M. Connolly, Scott M. Doran
المصدر: Journal of Medicinal Chemistry; Jun2008, Vol. 51 Issue 13, p3692-3695, 4p