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1دورية أكاديمية
المؤلفون: Mohamed D. M. Traoré, Vincent Zwick, Claudia A. Simões-Pires, Alessandra Nurisso, Mark Issa, Muriel Cuendet, Marjorie Maynadier, Sharon Wein, Henri Vial, Helene Jamet, Yung-Sing Wong
المصدر: ACS Omega, Vol 2, Iss 4, Pp 1550-1562 (2017)
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2470-1343Test
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المؤلفون: Claudia A. Simões-Pires, Yung-Sing Wong, Mohamed Dit Mady Traoré, Vincent Zwick, Sharon Wein, Muriel Cuendet, Marjorie Maynadier, Mark E. Issa, Alessandra Nurisso, Henri Vial, Hélène Jamet
المساهمون: Université des Sciences, des Techniques et des Technologies de Bamako (USTTB), School of Pharmaceutical Sciences, University of Geneva [Switzerland]-Université de Lausanne (UNIL), Dynamique des interactions membranaires normales et pathologiques (DIMNP), Centre National de la Recherche Scientifique (CNRS)-Université de Montpellier (UM)-Université Montpellier 2 - Sciences et Techniques (UM2)-Université Montpellier 1 (UM1), Département de Chimie Moléculaire - Chimie Inorganique Redox Biomimétique (DCM - CIRE ), Département de Chimie Moléculaire (DCM), Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes [2016-2019] (UGA [2016-2019])-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes [2016-2019] (UGA [2016-2019]), Département de pharmacochimie moléculaire (DPM ), Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes [2016-2019] (UGA [2016-2019])
المصدر: ACSOmega
ACS Omega
ACS Omega, Vol. 2, No 4 (2017) pp. 1550-1562
ACS Omega, Vol 2, Iss 4, Pp 1550-1562 (2017)
ACS Omega, ACS Publications, 2017, 2 (4), pp.1550-1562. ⟨10.1021/acsomega.6b00481⟩مصطلحات موضوعية: 0301 basic medicine, Gene isoform, Ketone, Molecular model, Stereochemistry, General Chemical Engineering, 01 natural sciences, Article, lcsh:Chemistry, 03 medical and health sciences, [CHIM]Chemical Sciences, ComputingMilieux_MISCELLANEOUS, chemistry.chemical_classification, ddc:615, 010405 organic chemistry, Chemistry, General Chemistry, HDAC6, HDAC1, 3. Good health, 0104 chemical sciences, 030104 developmental biology, lcsh:QD1-999, Histone deacetylase, Selectivity, Linker
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6d7e042e3b919823a01ddf17b882dc4bTest
http://pubs.acs.org/doi/abs/10.1021/acsomega.6b00481Test -
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المؤلفون: Claudia A. Simões-Pires, PM Allard, Muriel Cuendet, Vincent Zwick, J-L Wolfender, L Ory
المصدر: Planta Medica. 81:S1-S381
مصطلحات موضوعية: Pharmacology, Chromatography, Complementary and alternative medicine, Chemistry, Organic Chemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Uhplc ms ms, Analytical Chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::b746350a3cbc20fa9d38f3d51bcf15c4Test
https://doi.org/10.1055/s-0036-1596682Test -
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المؤلفون: Laurence Marcourt, Vincent Zwick, Pierre-Marie Allard, Katia Gindro, Lucie Ory, Jean-Luc Wolfender, Claudia A. Simões-Pires, Muriel Cuendet
المصدر: Phytochemical Analysis. 28:93-100
مصطلحات موضوعية: 0301 basic medicine, Penicillium griseofulvum, Plant Science, Pharmacology, Biochemistry, Analytical Chemistry, Romidepsin, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Panobinostat, Drug Discovery, medicine, Vorinostat, biology, General Medicine, Trypsin, Enzyme assay, 030104 developmental biology, Complementary and alternative medicine, chemistry, 030220 oncology & carcinogenesis, biology.protein, Molecular Medicine, Histone deacetylase, Belinostat, Food Science, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::02b2a031951c1cb9a72525fb8c2df044Test
https://doi.org/10.1002/pca.2652Test -
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المؤلفون: Vincent Zwick, Giuseppe Marco Randazzo, Claudia A. Simões-Pires, Muriel Cuendet, Philippe Bertrand, Carolina dos Santos Passos, Nadine Martinet, Charlotte Petit, Alessandra Nurisso
المصدر: Bioorganic & Medicinal Chemistry Letters
Bioorganic & Medicinal Chemistry Letters, Vol. 26, No 20 (2016) pp. 4955-4959مصطلحات موضوعية: 0301 basic medicine, In silico, Clinical Biochemistry, Cell, Pharmaceutical Science, Pharmacology, Histone Deacetylase 6, Blood–brain barrier, Biochemistry, Histone Deacetylases, 03 medical and health sciences, 0302 clinical medicine, Neuroblast, Cell Line, Tumor, Drug Discovery, medicine, Humans, Molecular Biology, IC50, Chromatography, High Pressure Liquid, Neurons, ddc:615, Chemistry, Organic Chemistry, Neurodegeneration, HDAC6, medicine.disease, In vitro, 3. Good health, Histone Deacetylase Inhibitors, 030104 developmental biology, medicine.anatomical_structure, Blood-Brain Barrier, Molecular Medicine, 030217 neurology & neurosurgery
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dc7b299e25e2702caf3f9cfc48225296Test
https://doi.org/10.1016/j.bmcl.2016.09.011Test -
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المصدر: Journal of Visualized Experiments, No 126 (2017) P. e55878
مصطلحات موضوعية: 0301 basic medicine, Gene isoform, General Chemical Engineering, Cell, Drug Evaluation, Preclinical, Histone Deacetylase 1, Histone Deacetylase 6, Hydroxamic Acids, General Biochemistry, Genetics and Molecular Biology, Mass Spectrometry, Romidepsin, HeLa, 03 medical and health sciences, Depsipeptides, Methods, medicine, Humans, Chromatography, High Pressure Liquid, Pharmacology, ddc:615, Chromatography, biology, General Immunology and Microbiology, General Neuroscience, biology.organism_classification, Molecular biology, Preclinical, Histone Deacetylase Inhibitors, Chemistry, Metabolism, 030104 developmental biology, Trichostatin A, medicine.anatomical_structure, Cell culture, Acetylation, High Pressure Liquid, Drug Evaluation, Histone deacetylase, Analysis, medicine.drug, HeLa Cells
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4854cbf93cb10640955a0abba8333b9fTest
https://pubmed.ncbi.nlm.nih.gov/28829415Test -
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المؤلفون: Yung-Sing Wong, Flaviane F. Hilário, Marjorie Maynadier, Vincent Zwick, Henri Vial, Rossimiriam Pereira de Freitas, Claudia A. Simões-Pires, Mohamed Dit Mady Traoré, Laurence Berry, Nicolas Fantozzi, Sharon Wein, Muriel Cuendet
المصدر: Organic Letters, Vol. 19, No 3 (2017) pp. 612-615
مصطلحات موضوعية: Scaffold, Cell, Triazole, Nanotechnology, 010402 general chemistry, 01 natural sciences, Biochemistry, Peptides, Cyclic, chemistry.chemical_compound, medicine, Physical and Theoretical Chemistry, ddc:615, Natural product, biology, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Cell Membrane, biology.organism_classification, Fluorescence, Transmembrane protein, 0104 chemical sciences, Membrane, medicine.anatomical_structure, chemistry, Biophysics, Tetra
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::499374aa90a4159699fff4c66596e28fTest
https://archive-ouverte.unige.ch/unige:94968Test -
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المؤلفون: Vincent, Zwick, Pierre-Marie, Allard, Lucie, Ory, Claudia A, Simões-Pires, Laurence, Marcourt, Katia, Gindro, Jean-Luc, Wolfender, Muriel, Cuendet
المصدر: Phytochemical Analysis, Vol. 28, No 2 (2017) pp. 93-100
مصطلحات موضوعية: ddc:615, Chromatography, Fungi/metabolism, Tandem Mass Spectrometry, High Pressure Liquid/methods, Fungi, Histone Deacetylases/metabolism, Tandem Mass Spectrometry/methods, Chromatography, High Pressure Liquid, Histone Deacetylases
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::7d23d944ae6a405da182e153d0412746Test
https://archive-ouverte.unige.ch/unige:94971Test -
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المؤلفون: Muriel Cuendet, Claudia A. Simões-Pires, Vincent Zwick
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol. 31, No sup1 (2016) pp. 209-214
مصطلحات موضوعية: 0301 basic medicine, Spectrometry, Mass, Electrospray Ionization, High-throughput screening, Cell, Drug Evaluation, Preclinical, Molecular Conformation, Histone Deacetylase 1, Pharmacology, Histone Deacetylase 6, Histone Deacetylases, Dose-Response Relationship, 03 medical and health sciences, Structure-Activity Relationship, Histone Deacetylase Inhibitors/analysis/chemistry/pharmacology, Drug Discovery, medicine, Humans, Chromatography, High Pressure Liquid, chemistry.chemical_classification, Histone Deacetylase 1/antagonists & inhibitors/metabolism, ddc:615, Chromatography, Dose-Response Relationship, Drug, biology, Drug discovery, Spectrometry, Electrospray Ionization, Cancer, General Medicine, HDAC6, Mass, medicine.disease, Histone Deacetylase Inhibitors, 030104 developmental biology, medicine.anatomical_structure, Histone, Enzyme, chemistry, Preclinical/methods, High Pressure Liquid, biology.protein, Drug Evaluation, Histone deacetylase, Histone Deacetylases/metabolism, Drug, HeLa Cells
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::883ab462cbcd9a7751ca36c6ff377bbeTest
https://archive-ouverte.unige.ch/unige:94975Test -
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المؤلفون: Judit Ovádi, Claudia A. Simões-Pires, Attila Lehotzky, Alessandra Nurisso, Philippe Bertrand, Muriel Cuendet, Nadine Martinet, Samuel Bouchet, Vincent Zwick, Christophe Blanquart
المساهمون: School of Pharmaceutical Sciences, Université de Lausanne (UNIL)-University of Geneva [Switzerland], Réseau épigénétique, Cancéropôle Grand-Ouest, Institut de Chimie des Milieux et Matériaux de Poitiers (IC2MP), Université de Poitiers-Institut national des sciences de l'Univers (INSU - CNRS)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Institut de Chimie de Nice (ICN), Université Nice Sophia Antipolis (... - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Côte d'Azur (UCA), Institute of Enzymology [Budapest], Research Centre for Natural Sciences, Hungarian Academy of Sciences (MTA)-Hungarian Academy of Sciences (MTA), Centre de Recherche en Cancérologie Nantes-Angers (CRCNA), Centre Hospitalier Universitaire d'Angers (CHU Angers), PRES Université Nantes Angers Le Mans (UNAM)-PRES Université Nantes Angers Le Mans (UNAM)-Hôtel-Dieu de Nantes-Institut National de la Santé et de la Recherche Médicale (INSERM)-Hôpital Laennec-Centre National de la Recherche Scientifique (CNRS)-Faculté de Médecine d'Angers-Centre hospitalier universitaire de Nantes (CHU Nantes), Authors thank the Centre National de la Recherche Scientifique– France, University of Poitiers, Region Poitou-Charentes (S.B. financial support), the Ligue Contre le Cancer: Committees of Vendée, et Charente-Maritime – France, ARSMeso44 – France, COST Actions CM1406 and CM1106 – Belgium and Hungarian OTKA Founds K-101039 and K-112144 for financial support. A.N. thanks the Excellence programme of the University of Geneva –Switzerland for financial support., Bernardo, Elizabeth, Université de Lausanne = University of Lausanne (UNIL)-Université de Genève = University of Geneva (UNIGE), Université Nice Sophia Antipolis (1965 - 2019) (UNS)
المصدر: Bioorganic and Medicinal Chemistry Letters
Bioorganic and Medicinal Chemistry Letters, Elsevier, 2016, ⟨10.1016/j.bmcl.2015.11.011⟩
Bioorganic and Medicinal Chemistry Letters, 2016, ⟨10.1016/j.bmcl.2015.11.011⟩
Bioorganic & Medicinal Chemistry Letters, Vol. 26, No 1 (2016) pp. 154-159مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Intrinsic activity, Formic Acid Esters, Stereochemistry, Clinical Biochemistry, Convergent synthesis, Pharmaceutical Science, [SDV.CAN]Life Sciences [q-bio]/Cancer, Alkenes, Hydroxamic Acids, Metathesis, Biochemistry, Histone Deacetylases, Catalysis, Dose-Response Relationship, Formic Acid Esters/chemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, [SDV.CAN] Life Sciences [q-bio]/Cancer, Models, Drug Discovery, Humans, Structure–activity relationship, Benzamides/chemistry, Benzamide, Molecular Biology, ddc:615, Dose-Response Relationship, Drug, Molecular Structure, biology, Organic Chemistry, Molecular, Alkenes/chemistry, 3. Good health, Histone Deacetylase Inhibitors, 030104 developmental biology, Tubulin, Histone Deacetylase Inhibitors/chemistry/pharmacology, Hydroxamic Acids/chemistry, chemistry, Benzamides, biology.protein, Molecular Medicine, Histone Deacetylases/metabolism, Drug, Selectivity
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::acc9fefa73c13b45a09cef22d951db0cTest
https://www.hal.inserm.fr/inserm-01299475/documentTest