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1
المؤلفون: A A Seymour, William N. Washburn, Dorothy Slusarchyk, P.J. McCann, B.E. Abboa-Offei, Minsheng Zhang, G.T. Allen, Ravindar N. Girotra, B.H. Frohlich, Michael Cap, Jollie D. Godfrey, Peter T. W. Cheng, R.J. George, C. Shao, Anita D. Russell, S. Skwish, Philip M. Sher, Jon J. Hangeland, A.V. Gavai, T.L. Waldron, Belay Tesfamariam, Yolanda Caringal, T.W. Harper, Tamara Dejneka, Kenneth E.J. Dickinson, Ginger Wu, Syed Z. Ahmed, Amarendra B. Mikkilineni, Hongwei Zhang
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:4290-4296
مصطلحات موضوعية: Agonist, β3 adrenergic receptor, Alkylation, medicine.drug_class, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Adrenergic beta-3 Receptor Agonists, Oxidative phosphorylation, Adrenergic beta-Agonists, Pharmacology, Biochemistry, Propanolamines, Structure-Activity Relationship, Drug Discovery, medicine, Molecular Medicine, Adrenergic agonist, β adrenergic receptor, Oxidation-Reduction, Molecular Biology, Drug metabolism
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::db28be835bfadb1da0ebd09bad48db49Test
https://doi.org/10.1016/j.bmcl.2007.05.030Test -
2
المؤلفون: Kenneth E.J. Dickinson, J. Buote, Denis E. Ryono, John Lloyd, Diane E. Normandin, J.E. Bird, Tamara Dejneka, Suzanne Moreland, E.R. Spitzmiller, Carol L. Delaney, Thomas L. Waldron, S. Skwish
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:195-200
مصطلحات موضوعية: Angiotensin receptor, medicine.medical_specialty, Lagomorpha, Angiotensin II receptor type 1, biology, Chemistry, Organic Chemistry, Clinical Biochemistry, Quinoline, Pharmaceutical Science, Pharmacology, biology.organism_classification, Biochemistry, Chemical synthesis, Angiotensin II, In vitro, chemistry.chemical_compound, Endocrinology, In vivo, Internal medicine, Drug Discovery, medicine, Molecular Medicine, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::1bc4ab930ac2965fffc9bb7323eb0c1fTest
https://doi.org/10.1016/s0960-894xTest(01)81146-x -
3
المؤلفون: Denis E. Ryono, Richard A. Morrison, Parker D. Mathers, James R. Powell, Zhengxiang Gu, J. Buote, John Lloyd, T. R. Schaeffer, S. Chong, Suzanne Moreland, Ronald E. White, E.R. Spitzmiller, Edward W. Petrillo, Kenneth E.J. Dickinson, J.E. Bird, Michael A. Poss, Tamara Dejneka
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:201-206
مصطلحات موضوعية: chemistry.chemical_classification, Angiotensin receptor, Carboxylic acid, Organic Chemistry, Clinical Biochemistry, Quinoline, Pharmaceutical Science, Angiotensin II receptor antagonist, Prodrug, Pharmacology, Biochemistry, Angiotensin II, chemistry.chemical_compound, chemistry, Oral administration, Drug Discovery, Molecular Medicine, Tetrazole, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::4d82e90d9b6bfaaede1fa290caa8ca24Test
https://doi.org/10.1016/s0960-894xTest(01)81147-1 -
4
المؤلفون: Carol L. Delaney, Suzanne Moreland, Zhengxiang Gu, Tamara Dejneka, Ellen Sieber-McMaster, Thomas L. Waldron, Michael A. Poss, J.Eileen Bird, Edward W. Petrillo, Ervin R. Spitzmiller, Denis E. Ryono, Sharon B. Williams, T. R. Schaeffer, S.Anders Hedberg, Kenneth E.J. Dickinson, Joyce A. Reid
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:145-150
مصطلحات موضوعية: Long lasting, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biological activity, Biochemistry, Angiotensin II, Orally active, Oral administration, Drug Discovery, Molecular Medicine, Receptor, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::c4b64c7596c17948cdb55858a7fa1fabTest
https://doi.org/10.1016/s0960-894xTest(01)81137-9 -
5
المؤلفون: Joyce A. Reid, Edward W. Petrillo, Maria P. Cimarusti, Harold N. Weller, Michael A. Poss, Russell J. Brittain, W. Lynn Rogers, Charles A. Free, Tamara Dejneka, Denis E. Ryono, Thomas L. Waldron, Helen Weber, Jack M. DeForrest
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:2739-2744
مصطلحات موضوعية: chemistry.chemical_classification, biology, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Sulfonamide (medicine), Diol, Pharmaceutical Science, Biological activity, Biochemistry, Chemical synthesis, Human renin, chemistry.chemical_compound, Enzyme, Enzyme inhibitor, Drug Discovery, Renin–angiotensin system, medicine, biology.protein, Molecular Medicine, Molecular Biology, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::024853216931a5b28419ff1637c4ec96Test
https://doi.org/10.1016/s0960-894xTest(01)80755-1 -
6
المؤلفون: Diane E. Normandin, Kenneth E.J. Dickinson, Denis E. Ryono, J.E. Bird, Thomas L. Waldron, Suzanne Moreland, Tamara Dejneka, Carol L. Delaney, J. Buote, John Lloyd, E.R. Spitzmiller, S. Skwish
المصدر: ChemInform. 25
مصطلحات موضوعية: chemistry.chemical_compound, Angiotensin receptor, Chemistry, In vivo, Quinoline, General Medicine, Aortic strips, Pharmacology, Affinities, Functional antagonism
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::fc28a15727d2dd7db1d3131e17d28538Test
https://doi.org/10.1002/chin.199426182Test -
7
المؤلفون: Tamara Dejneka, Jay Stevenson, Peter T. W. Cheng, Chongqing Sun, Baerbel R. Brown, Jeffrey A. Robl, Michael A. Poss, Tammy C. Wang
المصدر: ChemInform. 33
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, General method, Chemistry, Sequence (biology), General Medicine, Prodrug, Phosphonate, Combinatorial chemistry, Alkyl
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::4d767058d8658388ba42fcae15367857Test
https://doi.org/10.1002/chin.200221090Test -
8
المؤلفون: Konrad F. Koehler, Todd J. Friends, Marlena Grynfarb, Pratik Devasthale, Arthur M. Doweyko, Bolette Husman, Howard Einspahr, Jon J. Hangeland, John S. Sack, Tamara Dejneka, Jan Ljunggren, Cheryl M. Sheppard, Karin Mellström, Johnny Sandberg, Denis E. Ryono, Mathias Färnegårdh, Johan Malm
المصدر: Bioorganicmedicinal chemistry letters. 14(13)
مصطلحات موضوعية: Agonist, Steric effects, Thyroid Hormones, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Ligands, Biochemistry, Cell Line, Thyroid hormone receptor beta, 2-Propanol, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Amide, Drug Discovery, medicine, Side chain, Moiety, Structure–activity relationship, Amino Acids, Molecular Biology, Thyroid hormone receptor, Binding Sites, Chemistry, Organic Chemistry, Thyroid Hormone Receptors beta, Drug Design, Molecular Medicine, Triiodothyronine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::25aa20583081ad8d56e2722e4902c73cTest
https://pubmed.ncbi.nlm.nih.gov/15177471Test -
9
المؤلفون: Z. Merchant, S. Skwish, Dorothy Slusarchyk, P.J. McCann, D.A. Young, M. Morella, Kenneth E.J. Dickinson, Michael Cap, Ravindar N. Girotra, Anita D. Russell, B.E. Abboa-Offei, William N. Washburn, G.T. Allen, A.V. Gavai, Belay Tesfamariam, Peter T. W. Cheng, G. S. Bisacchi, Tammy C. Wang, A A Seymour, T.W. Harper, C.M. Arbeeny, Tamara Dejneka, Amarendra B. Mikkilineni, Poss Kathleen M, Chongqing Sun, Philip M. Sher, T.L. Waldron, R.J. George, B.H. Frohlich, Ginger Wu, Denis E. Ryono
المصدر: Bioorganicmedicinal chemistry letters. 14(13)
مصطلحات موضوعية: Agonist, Beta-3 adrenergic receptor, medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Glycine, Pharmaceutical Science, Adrenergic beta-3 Receptor Agonists, Pharmacology, Biochemistry, Methylation, Structure-Activity Relationship, In vivo, Drug Discovery, medicine, Animals, Humans, Molecular Biology, β3 adrenergic receptor, Dose-Response Relationship, Drug, Chemistry, digestive, oral, and skin physiology, Organic Chemistry, Biological activity, Stereoisomerism, Haplorhini, Adrenergic beta-Agonists, In vitro, Safety profile, Receptors, Adrenergic, beta-3, Molecular Medicine, Clinical evaluation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8c4e6c1a53153c8278f43697b1fe4710Test
https://pubmed.ncbi.nlm.nih.gov/15177466Test -
10
المؤلفون: Kenneth E.J. Dickinson, Michael Cap, Peter T. W. Cheng, A.V. Gavai, Arvind Mathur, Belay Tesfamariam, G.T. Allen, T.W. Harper, D.E. Hillyer, Tamara Dejneka, Dorothy Slusarchyk, S. Skwish, P.J. McCann, Chongqing Sun, Richard E. Gregg, D.A. Young, Carl P. Ciosek, Tammy C. Wang, Ravindar N. Girotra, Philip M. Sher, B.E. Abboa-Offei, A A Seymour, William N. Washburn, C.M. Arbeeny, Amarendra B. Mikkilineni, Poss Kathleen M, T.L. Waldron, R.J. George, B.H. Frohlich, Anita D. Russell, Denis E. Ryono
المصدر: Bioorganicmedicinal chemistry letters. 11(23)
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Biological Availability, Adrenergic beta-3 Receptor Agonists, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Ethanolamine, Drug Discovery, Chlorocebus aethiops, medicine, Structure–activity relationship, Animals, Humans, Anilides, Beta (finance), Molecular Biology, Aryl, Organic Chemistry, Adrenergic beta-Agonists, Rats, chemistry, Ethanolamines, Benzyl group, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3a03ede478701d49831f880574ab7cfbTest
https://pubmed.ncbi.nlm.nih.gov/11714605Test