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المؤلفون: Béatrice Quiclet-Sire, Samir Z. Zard, Stuart W. McCombie
المصدر: Organic Reactions. :1-257
مصطلحات موضوعية: chemistry, Radical, chemistry.chemical_element, Photochemistry, Nitrogen
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::b4de6fb8a593382ca3515816bab0fba3Test
https://doi.org/10.1002/0471264180.or108.01Test -
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المؤلفون: Samir Z. Zard, Stuart W. McCombie, Béatrice Quiclet-Sire
المساهمون: Merck Research Laboratories, Laboratoire de synthèse organique (DCSO), École polytechnique (X)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)
المصدر: Tetrahedron
Tetrahedron, Elsevier, 2018, 74 (38), pp.4969-4979. ⟨10.1016/j.tet.2018.03.042⟩مصطلحات موضوعية: Xanthates, [CHIM.ORGA]Chemical Sciences/Organic chemistry, 010405 organic chemistry, Chemistry, Radical, Organic Chemistry, Nitrogen-centered radicals, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Barton-McCombie deoxygenation, Barton–McCombie deoxygenation, Computational chemistry, Mechanism (philosophy), Drug Discovery, Barton decarboxylation, Deoxygenation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a50914839f5f46743d084ef402bd70e5Test
https://doi.org/10.1016/j.tet.2018.03.042Test -
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المؤلفون: William F. Berkowitz, Stuart W. McCombie
المصدر: Organic Reactions
مصطلحات موضوعية: Indole test, 010405 organic chemistry, Carbazole, Nitrene, Aryl, Thermal decomposition, 010402 general chemistry, Ring (chemistry), 01 natural sciences, 0104 chemical sciences, Catalysis, chemistry.chemical_compound, chemistry, Organic chemistry, Pyrrole
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::4ef539baa15210f81eb2dbab7c566104Test
https://doi.org/10.1002/0471264180.or092.02Test -
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المؤلفون: Stuart W. McCombie, Thomas P. Sakmar, Tatjana Dragic, Fotini Tsamis, Bahige M. Baroudy, Christoph Seibert, John W. Clader, John P. Moore, Anandan Palani, Svetlana Gavrilov, Shawn E. Kuhmann, Jayaram R. Tagat, Steven O. Smith, Weiwen Ying
المصدر: Virology. 349(1):41-54
مصطلحات موضوعية: Models, Molecular, Receptors, CCR5, Pyridines, viruses, Biology, Protein Structure, Secondary, Cell Line, Cyclic N-Oxides, 03 medical and health sciences, GPCR, Protein structure, Piperidines, HIV Fusion Inhibitors, Viral entry, Virology, Oximes, Humans, CCR5 inhibitors, SCH-C, Homology modeling, TAK-779, 030304 developmental biology, G protein-coupled receptor, chemistry.chemical_classification, 0303 health sciences, Binding Sites, Molecular Structure, 030302 biochemistry & molecular biology, AD101, Rational design, virus diseases, Amides, Small molecule, 3. Good health, Amino acid, Quaternary Ammonium Compounds, Biochemistry, chemistry, Chemokine binding, Mutagenesis, Site-Directed, HIV-1, CCR5
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::37bf7b55794ac5ea33b739e547cfe2a9Test
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المؤلفون: E. J. Remarque, Chuan-Chu Chou, B. A. ‘t Hart, Jayaram R. Tagat, Michel P.M. Vierboom, Julie M. Strizki, Catherine Pugliese-Sivo, Steensma Ruo, Paul J. Zavodny, Margreet Jonker, Satwant K. Narula, Stuart W. McCombie, Liesbeth Celebi-Paul
المصدر: Arthritis & Rheumatism. 52:627-636
مصطلحات موضوعية: Autoimmune disease, medicine.medical_specialty, Pathology, business.industry, medicine.medical_treatment, Cartilage, Immunology, Type II collagen, Antagonist, Arthritis, Inflammation, medicine.disease, Endocrinology, medicine.anatomical_structure, Rheumatology, Rheumatoid arthritis, Internal medicine, medicine, Immunology and Allergy, Pharmacology (medical), medicine.symptom, business, Saline
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::6c4058f0b9e8df37959f63d244776a49Test
https://doi.org/10.1002/art.20850Test -
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المؤلفون: Marc A. Labroli, Geoffrey B. Varty, Dennis V. Nazareno, Stuart W. McCombie, Steensma Ruo, Julie M. Strizki, Bahige M. Baroudy, Jayaram R. Tagat, Kathleen Cox, Robert W. Watkins, Jean E. Lachowicz, Yushi Xiao
المصدر: Journal of Medicinal Chemistry. 47:2405-2408
مصطلحات موضوعية: Potassium Channels, Anti-HIV Agents, medicine.drug_class, Stereochemistry, Substituent, Administration, Oral, Biological Availability, Carboxamide, CCR5 receptor antagonist, In Vitro Techniques, Chemical synthesis, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Drug Discovery, polycyclic compounds, medicine, Animals, Humans, Structure–activity relationship, heterocyclic compounds, Cation Transport Proteins, Trifluoromethyl, organic chemicals, Brain, Stereoisomerism, Ether-A-Go-Go Potassium Channels, Rats, Macaca fascicularis, Piperazine, Pyrimidines, chemistry, Potassium Channels, Voltage-Gated, CCR5 Receptor Antagonists, HIV-1, Leukocytes, Mononuclear, Molecular Medicine, Selectivity, Digestive System
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bb2f7d87ed1298266b41ff938e8e90d6Test
https://doi.org/10.1021/jm0304515Test -
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المؤلفون: William J. Greenlee, William Billard, Herbert Binch, Lian-Yong Chen, Ruth A. Duffy, Charles Liu, Gordon Crosby, Stuart W. McCombie, John W. Clader, Jennifer Ford, Shengjian Li, Joseph A. Kozlowski, Gowei Zhou, Vice Susan F, Jean E. Lachowicz
المصدر: Bioorganic & Medicinal Chemistry. 12:319-326
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Biological Availability, Pharmaceutical Science, Carboxamide, CHO Cells, Muscarinic Antagonists, Pharmacology, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Piperidines, In vivo, Cricetinae, Drug Discovery, Muscarinic acetylcholine receptor, Avoidance Learning, medicine, Animals, Structure–activity relationship, ortho-Aminobenzoates, Molecular Biology, Receptor, Muscarinic M2, Dose-Response Relationship, Drug, Chemistry, Organic Chemistry, Antagonist, In vitro, Rats, Bioavailability, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e7fb6725ef949509463e302ecb37ec1fTest
https://doi.org/10.1016/j.bmc.2003.11.005Test -
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المؤلفون: Tom Ketas, Jayaram R. Tagat, John W. Clader, Thomas P. Sakmar, Bahige M. Baroudy, Alexandra Trkola, Fotini Tsamis, Christoph Seibert, Svetlana Gavrilov, Francis Kajumo, Anadan Palani, John P. Moore, Shawn E. Kuhmann, Tatjana Dragic, Stuart W. McCombie
المصدر: Journal of Virology. 77:5201-5208
مصطلحات موضوعية: CD4-Positive T-Lymphocytes, Models, Molecular, Receptors, CCR5, Pyridines, viruses, Molecular Sequence Data, Immunology, Mutagenesis (molecular biology technique), HIV Envelope Protein gp120, Biology, Virus Replication, Membrane Fusion, Microbiology, Epitope, Cyclic N-Oxides, Piperidines, Viral entry, Virology, Vaccines and Antiviral Agents, Oximes, medicine, Humans, Amino Acid Sequence, Peptide sequence, Cells, Cultured, Antibodies, Monoclonal, virus diseases, Envelope glycoprotein GP120, Molecular biology, Transmembrane domain, Mechanism of action, Viral replication, Insect Science, CCR5 Receptor Antagonists, HIV-1, biology.protein, medicine.symptom
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2f00b025062d7674338c9a7ff16a42b5Test
https://doi.org/10.1128/jvi.77.9.5201-5208.2003Test -
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المؤلفون: Lisa Wojcik, Sherry Shapiro, Shawn E. Kuhmann, John W. Clader, Serena Xu, Stuart W. McCombie, Gregory R. Reyes, Julie M. Strizki, Jayaram R. Tagat, Tom Ketas, Elizabeth S. Maxwell, John P. Moore, Thomas Hunt Morgan, Bahige M. Baroudy, Alexandra Trkola, Pavel Pugach, Anandan Palani
المصدر: Proceedings of the National Academy of Sciences. 99:395-400
مصطلحات موضوعية: Multidisciplinary, viruses, Mutant, virus diseases, Transfection, CCR5 receptor antagonist, Biology, Virology, Peripheral blood mononuclear cell, Virus, Entry inhibitor, medicine, Vicriviroc, Receptor, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::855b983b32ab7ba68835b7674012511aTest
https://doi.org/10.1073/pnas.012519099Test -
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المؤلفون: Stuart W. McCombie, Bahige M. Baroudy, Anandan Palani, Mary E. Moreno, David D. Ho, Matthias Endres, Sherry Shapiro, Cheryl A. Stoddart, Liza Davies, Gregory R. Reyes, Chuan-Chu Chou, Julie M. Strizki, Yan Hou, Lisa Wojcik, Nicole Wagner, Serena Xu, Jia Liu, Catherine Pugliese-Sivo, Alexandra Trkola, John P. Moore, John W. Clader, Ahmad Fawzi, Jayaram R. Tagat, Kathleen Cox, William J. Greenlee
المصدر: Proceedings of the National Academy of Sciences. 98:12718-12723
مصطلحات موضوعية: Male, Anti-HIV Agents, Pyridines, Chemokine receptor CCR5, Aplaviroc, Mice, SCID, CCR5 receptor antagonist, Pharmacology, Cyclic N-Oxides, Rats, Sprague-Dawley, Mice, Piperidines, In vivo, Oximes, polycyclic compounds, medicine, Animals, Humans, heterocyclic compounds, Chemokine CCL5, Acquired Immunodeficiency Syndrome, Multidisciplinary, biology, Antagonist, virus diseases, Biological Sciences, Rats, Macaca fascicularis, Mechanism of action, CCR5 Receptor Antagonists, HIV-1, biology.protein, Vicriviroc, medicine.symptom, Astroglioma, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e9db017ab14a6d1c4985c63a00e570dcTest
https://doi.org/10.1073/pnas.221375398Test