المؤلفون: Durcik, Martina, Nyerges, Ákos, Skok, Žiga, Skledar, Darja Gramec, Trontelj, Jurij, Zidar, Nace, Ilaš, Janez, Zega, Anamarija, Cruz, Cristina D., Tammela, Päivi, Welin, Martin, Kimbung, Yengo R., Focht, Dorota, Benek, Ondřej, Révész, Tamás, Draskovits, Gábor, Szili, Petra Éva, Daruka, Lejla, Pal, Csaba, Kikelj, Danijel, Peterlin Mašič, Lucija, Tomašič, Tihomir

المساهمون: Bioactivity Screening Group, Division of Pharmaceutical Biosciences, Drug Research Program, Divisions of Faculty of Pharmacy

مصطلحات موضوعية: Antibacterial, Benzothiazole, DNA gyrase, Dual inhibitor, Topoisomerase IV, 317 Pharmacy

وصف الملف: application/pdf

العلاقة: The study was funded by the Slovenian Research Agency (Grant No. P1-0208, J1-9192 and BI-HU/19-20-008) and supported by the following research grants: European Research Council H2020-ERC-2014-CoG 648364 ? Resistance Evolution (C.P.); ?C?lzott Lend?let? Programme of the Hungarian Academy of Sciences LP-2017?10/2017(C.P.); ??lvonal? KKP 126506 (C.P.); GINOP-2.3.2?15?2016?00014 (EVOMER, to C.P.), GINOP-2.3.2?15?2016?00020 (MolMedEx TUMORDNS), and GINOP-2.3.3?15?2016?00001; EFOP 3.6.3-VEKOP-16-406 2017?00009 (P.Sz, T.R.); UNKP-19-3 New National Excellence Program of the Ministry for Innovation and Technology (P.Sz.); and a PhD Fellowship from the Boehringer Ingelheim Funds (A.N.). The authors thank Chris Berrie for editing the manuscript.; Durcik , M , Nyerges , Á , Skok , Ž , Skledar , D G , Trontelj , J , Zidar , N , Ilaš , J , Zega , A , Cruz , C D , Tammela , P , Welin , M , Kimbung , Y R , Focht , D , Benek , O , Révész , T , Draskovits , G , Szili , P É , Daruka , L , Pal , C , Kikelj , D , Peterlin Mašič , L & Tomašič , T 2021 , ' New dual ATP-competitive inhibitors of bacterial DNA gyrase and topoisomerase IV active against ESKAPE pathogens ' , European Journal of Medicinal Chemistry , vol. 213 , 113200 . https://doi.org/10.1016/j.ejmech.2021.113200Test; ORCID: /0000-0003-4697-8066/work/92285098; ORCID: /0000-0003-4655-8563/work/92286479; b2bee7cc-4b08-4fc0-a74f-4c22fc4c4085; http://hdl.handle.net/10138/353356Test; 000629626600053

الإتاحة: http://hdl.handle.net/10138/353356Test

المؤلفون: Skledar, Darja Gramec, Carino, Adriana, Trontelj, Jurij, Troberg, Johanna, Distrutti, Eleonora, Marchiano, Silvia, Tornasic, Tihomir, Zega, Anamarija, Finel, Moshe, Fiorucci, Stefano, Maisic, Lucija Peterlin

المساهمون: Faculty of Pharmacy, Division of Pharmaceutical Chemistry and Technology, Pharmaceutical Design and Discovery group, Drug Research Program, Moshe Finel / Principal Investigator

مصطلحات موضوعية: Bisphenol AF, Bisphenol AF glucuronide, Glucuronidation, Endocrine activities, Lipid accumulation, IN-VITRO, SEWAGE-SLUDGE, ANALOGS, CELLS, TOXICITY, GAMMA, IDENTIFICATION, PREADIPOCYTES, ANTAGONIST, Biochemistry, cell and molecular biology

وصف الملف: application/pdf

العلاقة: The authors thank OpenEye Scientific Software, Santa Fe, NM, USA, for free academic licenses for the use of their software, and Johanna Mosorin for skillful assistance in recombinant UGT preparations. Financial support of the Slovenian Research Agency (Grant No. P1-0208) and the Sigrid Juseliuksen Saatio, Finland (grant no. 4704583) are acknowledged.; Skledar , D G , Carino , A , Trontelj , J , Troberg , J , Distrutti , E , Marchiano , S , Tornasic , T , Zega , A , Finel , M , Fiorucci , S & Maisic , L P 2019 , ' Endocrine activities and adipogenic effects of bisphenol AF and its main metabolite ' , Chemosphere , vol. 215 , pp. 870-880 . https://doi.org/10.1016/j.chemosphere.2018.10.129Test; ORCID: /0000-0003-3886-4771/work/51564915; http://hdl.handle.net/10138/325049Test; f063b300-8d14-4568-8375-b75ca2da9adc; 85055983814; 000450383400096

الإتاحة: http://hdl.handle.net/10138/325049Test

المؤلفون: Skledar, Darja Gramec, Mašič, Lucija Peterlin

المصدر: https://www.intechopen.com/books/6891Test.

مصطلحات موضوعية: Estrogen

العلاقة: https://mts.intechopen.com/articles/show/title/the-role-of-metabolism-in-the-estrogenic-activity-of-endocrine-disrupting-chemicalsTest

الإتاحة: https://doi.org/10.5772/intechopen.81918Test
https://mts.intechopen.com/articles/show/title/the-role-of-metabolism-in-the-estrogenic-activity-of-endocrine-disrupting-chemicalsTest

المؤلفون: Skledar, Darja Gramec, Trontelj, Jurij, Troberg, Johanna, Tomašič, Tihomir, Zega, Anamarija, Finel, Moshe, Mašič, Lucija Peterlin

المساهمون: Divisions of Faculty of Pharmacy, Faculty of Pharmacy, Division of Pharmaceutical Chemistry and Technology, Drug Research Program, Pharmaceutical Design and Discovery group, Moshe Finel / Principal Investigator

مصطلحات موضوعية: ANTAGONIST, BINDING, ESTROGEN, RECEPTOR, 317 Pharmacy

وصف الملف: application/pdf

العلاقة: Skledar , D G , Trontelj , J , Troberg , J , Tomašič , T , Zega , A , Finel , M & Mašič , L P 2019 , ' Data on biosynthesis of BPAF glucuronide, enzyme kinetics of BPAF glucuronidation, and molecular modeling ' , Data in Brief , vol. 22 , pp. 977-986 . https://doi.org/10.1016/j.dib.2018.12.033Test; RIS: urn:94545CA9C581F6027C7252DE6976C546; ORCID: /0000-0003-3886-4771/work/57799882; 85060500571; 5e0a2ace-9bb8-48d7-aa38-589fcda55710; http://hdl.handle.net/10138/302049Test; 000458114600133

الإتاحة: http://hdl.handle.net/10138/302049Test

المؤلفون: Durcik, Martina, Skledar, Darja Gramec, Tomašič, Tihomir, Trontelj, Jurij, Peterlin Masic, Lucija

المصدر: SSRN Electronic Journal ; ISSN 1556-5068

الإتاحة: https://doi.org/10.2139/ssrn.4081145Test

المؤلفون: Durcik, Martina, Nyerges, Ákos, Skok, Žiga, Skledar, Darja Gramec, Trontelj, Jurij, Zidar, Nace, Ilaš, Janez, Zega, Anamarija, Cruz, Cristina D., Tammela, Päivi, Welin, Martin, Kimbung, Yengo R., Focht, Dorota, Benek, Ondřej, Révész, Tamás, Draskovits, Gábor, Szili, Petra Éva, Daruka, Lejla, Pál, Csaba, Kikelj, Danijel, Mašič, Lucija Peterlin, Tomašič, Tihomir

المساهمون: Boehringer Ingelheim Fonds, Magyar Tudományos Akadémia, Javna Agencija za Raziskovalno Dejavnost RS, Innovációs és Technológiai Minisztérium, European Research Council

المصدر: European Journal of Medicinal Chemistry ; volume 213, page 113200 ; ISSN 0223-5234

مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Pharmacology, General Medicine

الإتاحة: https://doi.org/10.1016/j.ejmech.2021.113200Test
https://api.elsevier.com/content/article/PII:S0223523421000490?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S0223523421000490?httpAccept=text/plainTest

المؤلفون: Skledar, Darja Gramec, Mašič, Lucija Peterlin

المساهمون: Slovenian Research Agency

المصدر: Science of The Total Environment ; volume 707, page 135211 ; ISSN 0048-9697

مصطلحات موضوعية: Pollution, Waste Management and Disposal, Environmental Chemistry, Environmental Engineering

الإتاحة: https://doi.org/10.1016/j.scitotenv.2019.135211Test
https://api.elsevier.com/content/article/PII:S0048969719352039?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S0048969719352039?httpAccept=text/plainTest

المؤلفون: Skledar, Darja Gramec, Carino, Adriana, Trontelj, Jurij, Troberg, Johanna, Distrutti, Eleonora, Marchianò, Silvia, Tomašič, Tihomir, Zega, Anamarija, Finel, Moshe, Fiorucci, Stefano, Mašič, Lucija Peterlin

المساهمون: Sigrid Juséliuksen Säätiö, Javna Agencija za Raziskovalno Dejavnost RS

المصدر: Chemosphere ; volume 215, page 870-880 ; ISSN 0045-6535

مصطلحات موضوعية: General Medicine, General Chemistry, Environmental Chemistry, Environmental Engineering, Pollution, Health, Toxicology and Mutagenesis, Public Health, Environmental and Occupational Health

الإتاحة: https://doi.org/10.1016/j.chemosphere.2018.10.129Test
https://api.elsevier.com/content/article/PII:S0045653518319908?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S0045653518319908?httpAccept=text/plainTest

المؤلفون: Skledar, Darja Gramec, Carino, Adriana, Trontelj, Jurij, Finel, Moshe, Troberg, Johanna, Fiorucci, Stefano, Mašič, Lucija Peterlin

المصدر: Toxicology Letters ; volume 280, page S111 ; ISSN 0378-4274

مصطلحات موضوعية: Toxicology, General Medicine

الإتاحة: https://doi.org/10.1016/j.toxlet.2017.07.310Test
https://api.elsevier.com/content/article/PII:S0378427417305477?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S0378427417305477?httpAccept=text/plainTest

المؤلفون: Skledar, Darja Gramec, Schmidt, Jan, Fic, Anja, Klopčič, Ivana, Trontelj, Jurij, Dolenc, Marija Sollner, Finel, Moshe, Mašič, Lucija Peterlin

المساهمون: Slovenian Research Agency, Academy of Finland

المصدر: Chemosphere ; volume 157, page 152-159 ; ISSN 0045-6535

مصطلحات موضوعية: General Medicine, General Chemistry, Environmental Chemistry, Environmental Engineering, Pollution, Health, Toxicology and Mutagenesis, Public Health, Environmental and Occupational Health

الإتاحة: https://doi.org/10.1016/j.chemosphere.2016.05.027Test
https://api.elsevier.com/content/article/PII:S004565351630666X?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S004565351630666X?httpAccept=text/plainTest