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1
المؤلفون: Thomas Wein, Sonja Sichler, Horst Thiermann, Franz Worek, Thomas Seeger, Karin V. Niessen, Sebastian Rappenglück, Klaus T. Wanner
المصدر: Current Computer-Aided Drug Design. 15:104-109
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Synaptic cleft, Stereochemistry, Drug Evaluation, Preclinical, Pyridinium Compounds, Receptors, Nicotinic, Ligands, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Organophosphate Poisoning, Drug Discovery, medicine, Computer Simulation, Acetylcholine receptor, Virtual screening, General Medicine, Acetylcholinesterase, Nicotinic acetylcholine receptor, 030104 developmental biology, Nicotinic agonist, chemistry, Molecular Medicine, Pharmacophore, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dd461f920c1b9a6f2d3b873866bb5536Test
https://doi.org/10.2174/1573409914666180703120201Test -
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المؤلفون: Sebastian Rappenglück, Horst Thiermann, Karin V. Niessen, Franz F. Paintner, Franz Worek, Thomas Seeger, Georg Höfner, Klaus T. Wanner, Thomas Wein, Sonja Sichler
المصدر: ChemMedChem. 13:2653-2663
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Stereochemistry, In silico, Pyridinium Compounds, Receptors, Nicotinic, Neurotransmission, Torpedo, 010402 general chemistry, 01 natural sciences, Biochemistry, Neuromuscular junction, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, General Pharmacology, Toxicology and Pharmaceutics, Binding site, Pharmacology, Binding Sites, Molecular Structure, Organic Chemistry, Acetylcholinesterase, 0104 chemical sciences, Nicotinic acetylcholine receptor, 030104 developmental biology, medicine.anatomical_structure, chemistry, Molecular Medicine, Pyridinium, Hydrophobic and Hydrophilic Interactions, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::647280789ea527f5bf6b9d7153ee7e7dTest
https://doi.org/10.1002/cmdc.201800539Test -
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المؤلفون: Karin V. Niessen, Thomas Seeger, Georg Höfner, Horst Thiermann, Franz Worek, Klaus T. Wanner, Thomas Wein, Sebastian Rappenglück
المصدر: Toxicology Letters. 293:190-197
مصطلحات موضوعية: Male, 0301 basic medicine, Obidoxime, Pyridines, Antidotes, Diaphragm, Soman, Pyridinium Compounds, Muscarinic Antagonists, Receptors, Nicotinic, Pharmacology, Toxicology, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Organophosphate Poisoning, 0302 clinical medicine, medicine, Animals, Chemical Warfare Agents, Nicotinic Agonists, Rats, Wistar, Nerve agent, Chemistry, Stereoisomerism, General Medicine, Bridged Bicyclo Compounds, Heterocyclic, Receptors, Muscarinic, Acetylcholinesterase, Rats, Nicotinic acetylcholine receptor, 030104 developmental biology, Nicotinic agonist, Epibatidine, Cholinergic, Cholinesterase Inhibitors, 030217 neurology & neurosurgery, Acetylcholine, Muscle Contraction, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ae7671cbcf2f717eb13a2528cb07f378Test
https://doi.org/10.1016/j.toxlet.2017.10.009Test -
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المؤلفون: Sebastian Rappenglück, Georg Höfner, Sonja Sichler, Klaus T. Wanner, Thomas Wein, Thomas Seeger, Franz Worek, Karin V. Niessen, Horst Thiermann
المصدر: Toxicology Letters. 293:184-189
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Cholinesterase Reactivators, Synaptic cleft, Protein Conformation, Stereochemistry, Pyridinium Compounds, Receptors, Nicotinic, Torpedo, Toxicology, 03 medical and health sciences, Acetylcholine binding, Organophosphate Poisoning, 0302 clinical medicine, medicine, Animals, Computer Simulation, Binding site, Acetylcholine receptor, Binding Sites, Molecular Structure, Chemistry, General Medicine, Acetylcholine, Molecular Docking Simulation, Nicotinic acetylcholine receptor, 030104 developmental biology, Nicotinic agonist, Docking (molecular), 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::914026e186285b7d585dda5c7e393f8dTest
https://doi.org/10.1016/j.toxlet.2017.10.024Test -
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المؤلفون: Thomas Seeger, Franz Worek, Georg Höfner, Sebastian Rappenglück, Franz F. Paintner, Thomas Wein, Sonja Sichler, Karin V. Niessen, Horst Thiermann, Klaus T. Wanner
المصدر: Toxicology Letters. 293:172-183
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Cholinesterase Reactivators, Spectrometry, Mass, Electrospray Ionization, Phencyclidine, Pyridinium Compounds, Receptors, Nicotinic, Torpedo, Toxicology, Tandem mass spectrometry, Binding, Competitive, Mass Spectrometry, law.invention, Radioligand Assay, 03 medical and health sciences, Tandem Mass Spectrometry, Liquid chromatography–mass spectrometry, law, Muscarinic acetylcholine receptor M5, Animals, Binding site, Chromatography, High Pressure Liquid, Binding Sites, Chemistry, Reproducibility of Results, General Medicine, Ligand (biochemistry), Nicotinic acetylcholine receptor, 030104 developmental biology, Biochemistry, Carbachol
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::33676eb184af9dbb14b0d18454f80bb8Test
https://doi.org/10.1016/j.toxlet.2017.11.013Test -
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المؤلفون: Franz F. Paintner, Franz Worek, Thomas Wein, Sebastian Rappenglück, Sonja Sichler, Karin V. Niessen, Klaus T. Wanner, Horst Thiermann, Georg Höfner, Thomas Seeger
المصدر: ChemMedChem. 13:1806-1816
مصطلحات موضوعية: 0301 basic medicine, Steric effects, Stereochemistry, Pyridinium Compounds, Receptors, Nicotinic, Torpedo, 010402 general chemistry, 01 natural sciences, Biochemistry, law.invention, Structure-Activity Relationship, 03 medical and health sciences, Organophosphate Poisoning, law, Drug Discovery, Animals, General Pharmacology, Toxicology and Pharmaceutics, Binding site, Binding affinities, Pharmacology, Binding Sites, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Ligand binding assay, Organic Chemistry, Affinities, 0104 chemical sciences, Nicotinic acetylcholine receptor, 030104 developmental biology, Molecular Medicine, Linker
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::491b129484f63b220eb89aa840d96e93Test
https://doi.org/10.1002/cmdc.201800325Test -
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المؤلفون: Franz Worek, Klaus T. Wanner, Thomas Seeger, Sebastian Rappenglück, Horst Thiermann, Karin V. Niessen
المصدر: Synthesis. 49:4055-4064
مصطلحات موضوعية: chemistry.chemical_classification, Nucleophilic addition, Nitrile, 010405 organic chemistry, Organic Chemistry, Aromatization, Alkyne, Regioselectivity, 010402 general chemistry, 01 natural sciences, Medicinal chemistry, Catalysis, 0104 chemical sciences, chemistry.chemical_compound, chemistry, Reagent, Amide, Pyridine, Organic chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::7b1c631637ed7474ab1a08538e80aa2bTest
https://doi.org/10.1055/s-0036-1589025Test -
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المؤلفون: Thomas Seeger, Corinna Scheffel, Karin V. Niessen, Klaus T. Wanner, Franz Worek, Horst Thiermann, Sebastian Rappenglück
المصدر: Toxicology letters. 293
مصطلحات موضوعية: 0301 basic medicine, Agonist, Allosteric modulator, Patch-Clamp Techniques, alpha7 Nicotinic Acetylcholine Receptor, medicine.drug_class, Pyridinium Compounds, CHO Cells, Pharmacology, Toxicology, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, 0302 clinical medicine, Cricetulus, Cricetinae, Muscarinic acetylcholine receptor, medicine, Animals, Nicotinic Agonists, Receptor, Acetylcholine receptor, Dose-Response Relationship, Drug, Chemistry, Phenylurea Compounds, General Medicine, Isoxazoles, Acetylcholinesterase, Electrophysiological Phenomena, 030104 developmental biology, Nicotinic agonist, 030217 neurology & neurosurgery, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2e390b55cc845e8864de88507b6594b8Test
https://pubmed.ncbi.nlm.nih.gov/29191791Test -
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المصدر: ChemPlusChem. 77:877-888
مصطلحات موضوعية: chemistry.chemical_classification, Aqueous solution, Sodium, Inorganic chemistry, chemistry.chemical_element, Salt (chemistry), General Chemistry, Oxime, Chloride, chemistry.chemical_compound, Hydroxylamine, chemistry, Nitric acid, Hydroxylammonium chloride, medicine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::a026704a328352252cbd358f9211c1baTest
https://doi.org/10.1002/cplu.201200136Test -
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المصدر: Chemistry - A European Journal. 18:4051-4062
مصطلحات موضوعية: Propellant, Chemistry, Isochoric process, Detonation velocity, Organic Chemistry, Analytical chemistry, Detonation, General Chemistry, Catalysis, symbols.namesake, Differential scanning calorimetry, symbols, Specific energy, Specific impulse, Raman spectroscopy
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::770ca9eb5fa9b7ca11d044c30acaa472Test
https://doi.org/10.1002/chem.201103737Test