المؤلفون: Creighton, Samantha D. (ORCID 0000-0002-3463-2394), Jardine, Kristen H., Desimone, Alexa, Zmetana, Megan, Castellano, Sabrina, Milite, Ciro, Sbardella, Gianluca (ORCID 0000-0003-0748-1145), Winters, Boyer D.

المصدر: Learning & Memory. Mar 2022 29(3):71-76.

تمت مراجعته من قبل الزملاء: Y

Page Count: 6

الواصفات: Alzheimers Disease, Animals, Research, Spatial Ability, Memory, Age Differences, Intervention, Biochemistry

المؤلفون: Auberson, Yves, P, Arimondo, Paola, B, Duca, Maria, Essig, Sebastian, Grether, Uwe, Rufer, Arne, Sbardella, Gianluca, Schopfer, Ulrich, Torrens, Antoni, van der Stelt, Mario, Vauzeilles, Boris, Vázquez, Olalla, Zhang, Andrew

المساهمون: Novartis Institutes for BioMedical Research (NIBR), Chimie biologique épigénétique - Epigenetic Chemical Biology (EpiCBio), Institut Pasteur Paris (IP)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité), Institut de Chimie de Nice (ICN), Université Nice Sophia Antipolis (1965 - 2019) (UNS)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)-Université Côte d'Azur (UniCA), Bayer AG Wuppertal, Germany, F. Hoffmann-La Roche Basel, Università degli Studi di Salerno = University of Salerno (UNISA), ABAC Therapeutics Barcelona, Universiteit Leiden = Leiden University, Institut de Chimie des Substances Naturelles (ICSN), Institut de Chimie - CNRS Chimie (INC-CNRS)-Université Paris-Saclay-Centre National de la Recherche Scientifique (CNRS), Philipps Universität Marburg = Philipps University of Marburg, AstraZeneca US Waltham, USA, AstraZeneca Cambridge, UK

المصدر: ISSN: 1439-4227.

مصطلحات موضوعية: [CHIM.THER]Chemical Sciences/Medicinal Chemistry

العلاقة: info:eu-repo/semantics/altIdentifier/pmid/36704975; hal-04278306; https://hal.science/hal-04278306Test; https://hal.science/hal-04278306/documentTest; https://hal.science/hal-04278306/file/EFMC%20trends%20in%20MCCB.pdfTest; PUBMED: 36704975

الإتاحة: https://doi.org/10.1002/cbic.202200690Test
https://hal.science/hal-04278306Test
https://hal.science/hal-04278306/documentTest
https://hal.science/hal-04278306/file/EFMC%20trends%20in%20MCCB.pdfTest

المؤلفون: Fiorentino, Francesco, Sementilli, Sara, Menna, Martina, Turrisi, Federica, Tomassi, Stefano, Pellegrini, Francesca Romana, Iuzzolino, Angela, D’Acunzo, Francesca, Feoli, Alessandra, Wapenaar, Hannah, Taraglio, Sophie, Fraschetti, Caterina, Del Bufalo, Donatella, Sbardella, Gianluca, Dekker, Frank J., Paiardini, Alessandro, Trisciuoglio, Daniela, Mai, Antonello, Rotili, Dante

المصدر: Fiorentino , F , Sementilli , S , Menna , M , Turrisi , F , Tomassi , S , Pellegrini , F R , Iuzzolino , A , D’Acunzo , F , Feoli , A , Wapenaar , H , Taraglio , S , Fraschetti , C , Del Bufalo , D , Sbardella , G , Dekker , F J , Paiardini , A , Trisciuoglio , D , Mai , A & Rotili , D 2023 , ' First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8 ' , Journal of Medicinal Chemistry , vol. 66 , ....

وصف الملف: application/pdf

العلاقة: https://research.rug.nl/en/publications/7ca47a3f-7ab9-4c7b-a739-7961d690ede8Test

الإتاحة: https://doi.org/10.1021/acs.jmedchem.2c01937Test
https://hdl.handle.net/11370/7ca47a3f-7ab9-4c7b-a739-7961d690ede8Test
https://research.rug.nl/en/publications/7ca47a3f-7ab9-4c7b-a739-7961d690ede8Test
https://pure.rug.nl/ws/files/688529096/acs.jmedchem.2c01937.pdfTest
http://www.scopus.com/inward/record.url?scp=85159627845&partnerID=8YFLogxKTest

المؤلفون: Cipriano, Alessandra, Viviano, Monica, Feoli, Alessandra, Milite, Ciro, Sarno, Giuliana, Castellano, Sabrina, Sbardella, Gianluca

المساهمون: Ministero dell'Universit? e della Ricerca

المصدر: Journal of Medicinal Chemistry ; volume 66, issue 17, page 11632-11655 ; ISSN 0022-2623 1520-4804

الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c00770Test

المؤلفون: Feoli, Alessandra, Iannelli, Giulia, Cipriano, Alessandra, Milite, Ciro, Shen, Lei, Wang, Zhihao, Hadjikyriacou, Andrea, Lowe, Troy L., Safaeipour, Cyrus, Viviano, Monica, Sarno, Giuliana, Morretta, Elva, Monti, Maria Chiara, Yang, Yanzhong, Clarke, Steven G., Cosconati, Sandro, Castellano, Sabrina, Sbardella, Gianluca

المساهمون: Division of Molecular and Cellular Biosciences, Ministero dell’Istruzione, dell’Università e della Ricerca, Associazione Italiana per la Ricerca sul Cancro, Università degli Studi di Salerno, National Institute of General Medical Sciences, Regione Campania

المصدر: Journal of Medicinal Chemistry ; volume 66, issue 19, page 13665-13683 ; ISSN 0022-2623 1520-4804

مصطلحات موضوعية: Drug Discovery, Molecular Medicine

الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c01030Test

المؤلفون: Viviano, Monica, Cipriano, Alessandra, Fabbrizi, Emanuele, Feoli, Alessandra, Castellano, Sabrina, Sbardella, Gianluca, Mai, Antonello, Milite, Ciro, Rotili, Dante

المساهمون: Viviano, Monica, Cipriano, Alessandra, Fabbrizi, Emanuele, Feoli, Alessandra, Castellano, Sabrina, Sbardella, Gianluca, Mai, Antonello, Milite, Ciro, Rotili, Dante

مصطلحات موضوعية: BD1, BET, Epigenetic, bromodomain, cancer, selective inhibition, small molecule modulators

العلاقة: info:eu-repo/semantics/altIdentifier/pmid/38465537; firstpage:1; lastpage:17; numberofpages:17; journal:EXPERT OPINION ON THERAPEUTIC PATENTS; https://hdl.handle.net/11386/4859652Test

الإتاحة: https://doi.org/10.1080/13543776.2024.2327300Test
https://hdl.handle.net/11386/4859652Test

المؤلفون: Feoli, Alessandra, Sarno, Giuliana, Castellano, Sabrina, Sbardella, Gianluca

المساهمون: Feoli, Alessandra, Sarno, Giuliana, Castellano, Sabrina, Sbardella, Gianluca

مصطلحات موضوعية: DMSO, DMSO effect, biophysical characterization, epigenetic, ligand affinity

العلاقة: info:eu-repo/semantics/altIdentifier/pmid/38205880; info:eu-repo/semantics/altIdentifier/wos/WOS:001148333600001; volume:25; firstpage:e202300809; lastpage:e202300809; numberofpages:11; journal:CHEMBIOCHEM; https://hdl.handle.net/11386/4853735Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85183041993

الإتاحة: https://doi.org/10.1002/cbic.202300809Test
https://hdl.handle.net/11386/4853735Test

المؤلفون: Milite, Ciro, Sarno, Giuliana, Pacilio, Ida, Cianciulli, Agostino, Viviano, Monica, Iannelli, Giulia, Gazzillo, Erica, Feoli, Alessandra, Cipriano, Alessandra, Giovanna Chini, Maria, Castellano, Sabrina, Bifulco, Giuseppe, Sbardella, Gianluca

المصدر: ChemMedChem ; ISSN:1860-7187

مصطلحات موضوعية: Arginine mimics, Bioisosterism, PRMT4 inhibitors, Prodrugs, pyrrole

العلاقة: https://doi.org/10.1002/cmdc.202400139Test; https://pubmed.ncbi.nlm.nih.gov/38752332Test

الإتاحة: https://doi.org/10.1002/cmdc.202400139Test
https://pubmed.ncbi.nlm.nih.gov/38752332Test

المؤلفون: Cipriano, Alessandra, Milite, Ciro, Feoli, Alessandra, Viviano, Monica, Pepe, Giacomo, Campiglia, Pietro, Sarno, Giuliana, Picaud, Sarah, Imaide, Satomi, Makukhin, Nikolai, Filippakopoulos, Panagis, Ciulli, Alessio, Castellano, Sabrina, Sbardella, Gianluca

المصدر: Cipriano , A , Milite , C , Feoli , A , Viviano , M , Pepe , G , Campiglia , P , Sarno , G , Picaud , S , Imaide , S , Makukhin , N , Filippakopoulos , P , Ciulli , A , Castellano , S & Sbardella , G 2022 , ' Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain ' , ChemMedChem , vol. 17 , no. 20 , e202200343 . https://doi.org/10.1002/cmdc.202200343Test

مصطلحات موضوعية: Benzimidazole-6-sulfonamide, Bromodomain, Bioisosteres, Selectivity, Structure-activity relationships

وصف الملف: application/pdf

العلاقة: https://discovery.dundee.ac.uk/en/publications/9262919b-076d-4f3a-b6e8-482a936747cdTest

الإتاحة: https://doi.org/10.1002/cmdc.202200343Test
https://discovery.dundee.ac.uk/en/publications/9262919b-076d-4f3a-b6e8-482a936747cdTest
https://discovery.dundee.ac.uk/ws/files/86582869/ChemMedChem_2022_Cipriano_Discovery_of_Benzo_d_imidazole_6_sulfonamides_as_Bromodomain_and_Extra_Terminal_Domain_BET.pdfTest
http://www.scopus.com/inward/record.url?scp=85138079605&partnerID=8YFLogxKTest

المؤلفون: Iannelli, Giulia, Milite, Ciro, Marechal, Nils, Cura, Vincent, Bonnefond, Luc, Troffer-Charlier, Nathalie, Feoli, Alessandra, Rescigno, Donatella, Wang, Yalong, Cipriano, Alessandra, Viviano, Monica, Bedford, Mark, Cavarelli, Jean, Castellano, Sabrina, Sbardella, Gianluca

المساهمون: Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), Université de Strasbourg (UNISTRA)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)

المصدر: ISSN: 0022-2623.

مصطلحات موضوعية: [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology

العلاقة: hal-04116086; https://hal.science/hal-04116086Test; https://hal.science/hal-04116086/documentTest; https://hal.science/hal-04116086/file/islandora_163785.pdfTest

الإتاحة: https://doi.org/10.1021/acs.jmedchem.2c00252Test
https://hal.science/hal-04116086Test
https://hal.science/hal-04116086/documentTest
https://hal.science/hal-04116086/file/islandora_163785.pdfTest