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1دورية أكاديمية
المؤلفون: Na Meng (215412), Wensheng Yu (2124583), Takao Suzuki (401012), Maofen Chen (10499243), Zhiqi Qi (8815358), Bin Hu (122268), Jianming Bao (2125180), John S. Debenham (2295976), Robert Mazzola (2452012), Joseph L. Duffy (1601548)
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Evolutionary Biology, Sociology, Cancer, Environmental Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, Physical Sciences not elsewhere classified, Methanol, charge, heterocyclic groups, methanol derivatives, nitrogen atom, deoxygenation, pyridyl
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المؤلفون: Mckittrick Brian A, Mihirbaran Mandal, Jared N. Cumming, Andrew Brunskill, Andrew Stamford, Hongwu Wang, Xiaoxiang Liu, Alexei V. Buevich, Robert Mazzola, Peter Orth, Zhaoning Zhu, John P. Caldwell
المصدر: European Journal of Organic Chemistry. 2021:5073-5079
مصطلحات موضوعية: Chemistry, Organic Chemistry, Regioselectivity, Organic chemistry, Amine gas treating, Physical and Theoretical Chemistry, Interception, Curtius rearrangement
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::df583a27443bdf99ebdd82d44726c381Test
https://doi.org/10.1002/ejoc.202101056Test -
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المؤلفون: Wensheng Yu, Maofen Chen, Takao Suzuki, Zhiqi Qi, Bin Hu, Jianming Bao, John S. Debenham, Na Meng, Joseph L. Duffy, Robert Mazzola
المصدر: The Journal of Organic Chemistry. 86:5560-5567
مصطلحات موضوعية: 010405 organic chemistry, Organic Chemistry, 010402 general chemistry, 01 natural sciences, Medicinal chemistry, 0104 chemical sciences, chemistry.chemical_compound, chemistry, Nitrogen atom, Negative charge, Imidazole, Methanol, Tertiary alcohols, Deoxygenation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b6e46bfea57fcf3b5d4f09671845422eTest
https://doi.org/10.1021/acs.joc.1c00067Test -
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المؤلفون: Wenping, Li, Yuchuan, Wang, Talakad G, Lohith, Zhizhen, Zeng, Ling, Tong, Robert, Mazzola, Kerry, Riffel, Patricia, Miller, Mona, Purcell, Marie, Holahan, Hyking, Haley, Liza, Gantert, David, Hesk, Sumei, Ren, John, Morrow, Jason, Uslaner, Arie, Struyk, Jenny Miu-Chun, Wai, Michael T, Rudd, David M, Tellers, Thomas, McAvoy, Guy, Bormans, Michel, Koole, Koen, Van Laere, Kim, Serdons, Jan, de Hoon, Ruben, Declercq, Inge, De Lepeleire, Maria B, Pascual, Paolo, Zanotti-Fregonara, Meixiang, Yu, Victoria, Arbones, Joseph C, Masdeu, Amy, Cheng, Azher, Hussain, Tjerk, Bueters, Matt S, Anderson, Eric D, Hostetler, Anthony S, Basile
المصدر: Science translational medicine. 14(627)
مصطلحات موضوعية: Alzheimer Disease, Positron-Emission Tomography, Acetylcholinesterase, Animals, Humans, Macaca mulatta, Receptors, Muscarinic
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::d4a48387c373777e91d8509feb8c9c29Test
https://pubmed.ncbi.nlm.nih.gov/35020407Test -
5
المؤلفون: Wenping Li, Yuchuan Wang, Talakad G. Lohith, Zhizhen Zeng, Ling Tong, Robert Mazzola, Kerry Riffel, Patricia Miller, Mona Purcell, Marie Holahan, Hyking Haley, Liza Gantert, David Hesk, Sumei Ren, John Morrow, Jason Uslaner, Arie Struyk, Jenny Miu-Chun Wai, Michael T. Rudd, David M. Tellers, Thomas McAvoy, Guy Bormans, Michel Koole, Koen Van Laere, Kim Serdons, Jan de Hoon, Ruben Declercq, Inge De Lepeleire, Maria B. Pascual, Paolo Zanotti-Fregonara, Meixiang Yu, Victoria Arbones, Joseph C. Masdeu, Amy Cheng, Azher Hussain, Tjerk Bueters, Matt S. Anderson, Eric D. Hostetler, Anthony S. Basile
مصطلحات موضوعية: General Medicine
وصف الملف: Print-Electronic
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1e44197a5317a5a2a9f28fb0766d601bTest
https://lirias.kuleuven.be/handle/20.500.12942/688229Test -
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المؤلفون: John A. Morrow, Robert Mazzola, Cristian Salinas, Eric D. Hostetler, Stefania Risso, Fiona Thomson, Tjerk Bueters, Nicholas B. Hastings, Jenny Wai, Sony Agrawal, Liza Gantert, Brian C. Magliaro, Paul McQuade, Zhizhen Zeng, Marie A. Holahan, David Hesk, Melissa Egbertson, Jeffrey W. Schubert, Ling Tong, Robert Gomez, Jongrock Kong, Aniket Joshi, Frederick J. Monsma, David M. Tellers, Kristen L.G. Jones, Jason M. Uslaner, Jing Liao, Patricia Miller, Michelle Smith, Oleg Selyutin, Kerry Riffel, Xiaolei Gao, Scott T. Harrison, Zhaoyang Meng, James Mulhearn, Michael Man-Chu Lo, Wenping Li, Michael T. Rudd, Barbara Hanney, Mona Purcell, Jianming Bao, Hyking Haley
المصدر: Journal of Medicinal Chemistry. 63:2411-2425
مصطلحات موضوعية: Agonist, 0303 health sciences, Carbachol, medicine.diagnostic_test, Chemistry, medicine.drug_class, Allosteric regulation, Pharmacology, 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, In vivo, Positron emission tomography, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Molecular Medicine, Receptor, Preclinical imaging, 030304 developmental biology, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::949c4dbede58ed2de44d27f608635d36Test
https://doi.org/10.1021/acs.jmedchem.9b01406Test -
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المؤلفون: Hongwu Wang, Leonard Favreau, Jairam Palamanda, Xinjie Lin, Diane Rindgen, John P. Caldwell, Zhaoning Zhu, Pramila Kumari, Alexei V. Buevich, Reshma Kuvelkar, Edward C. Sherer, Andrew Stamford, Kathleen Cox, Jared N. Cumming, Diane Grotz, Matthew E. Kennedy, Xiaoxang Liu, Mihir Mandal, Lynn A. Hyde, Kaushik Mitra, Eric M. Parker, Xia Chen, Robert Mazzola
المصدر: Journal of Medicinal Chemistry. 61:10700-10708
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Metabolite, Oxidative phosphorylation, 030226 pharmacology & pharmacy, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Cytochrome P-450 CYP3A, Animals, Humans, Moiety, Structure–activity relationship, Tissue Distribution, Cytochrome P-450 CYP3A Inhibitors, CYP3A4, Rats, Kinetics, Pyrimidines, 030104 developmental biology, chemistry, Reactive metabolite, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::39ff6cf8405739a6779b4176b25e3536Test
https://doi.org/10.1021/acs.jmedchem.8b01326Test -
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المؤلفون: Lili Zhang, Li Xiao, Diane Rindgen, Mihirbaran Mandal, John P. Caldwell, Xiaoxiang Liu, Anandan Palani, Zhaoning Zhu, Alexei V. Buevich, Dmitri A. Pissarnitski, Eric M. Parker, Robert Mazzola, Lynn A. Hyde, Xianhai Huang, Mckittrick Brian A
المصدر: Journal of medicinal chemistry. 63(15)
مصطلحات موضوعية: chemistry.chemical_classification, Oxadiazoles, Amyloid beta-Peptides, Binding Sites, Double bond, Stereochemistry, Alkenes, In vitro, Peptide Fragments, Rats, chemistry.chemical_compound, Structure-Activity Relationship, HEK293 Cells, chemistry, Nucleophile, Drug Discovery, Molecular Medicine, Moiety, Structure–activity relationship, Animals, Humans, Reactivity (chemistry), γ secretase, Azepine, Amyloid Precursor Protein Secretases
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3c49d382e7dab42ef6f306cb076a3f72Test
https://pubmed.ncbi.nlm.nih.gov/32786237Test -
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المؤلفون: Ling, Tong, Wenping, Li, Michael Man-Chu, Lo, Xiaolei, Gao, Jenny Miu-Chen, Wai, Michael, Rudd, David, Tellers, Aniket, Joshi, Zhizhen, Zeng, Patricia, Miller, Cristian, Salinas, Kerry, Riffel, Hyking, Haley, Mona, Purcell, Marie, Holahan, Liza, Gantert, Jeffrey W, Schubert, Kristen, Jones, James, Mulhearn, Melissa, Egbertson, Zhaoyang, Meng, Barbara, Hanney, Robert, Gomez, Scott T, Harrison, Paul, McQuade, Tjerk, Bueters, Jason, Uslaner, John, Morrow, Fiona, Thomson, Jongrock, Kong, Jing, Liao, Oleg, Selyutin, Jianming, Bao, Nicholas B, Hastings, Sony, Agrawal, Brian C, Magliaro, Frederick J, Monsma, Michelle D, Smith, Stefania, Risso, David, Hesk, Eric, Hostetler, Robert, Mazzola
المصدر: Journal of medicinal chemistry. 63(5)
مصطلحات موضوعية: Cricetulus, Allosteric Regulation, Receptor, Muscarinic M4, Pyridines, Positron-Emission Tomography, Animals, Humans, Neurodegenerative Diseases, CHO Cells, Carbon Radioisotopes, Muscarinic Agonists, Macaca mulatta
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::cd3ef3c047c980065bd64efde0a0b7e9Test
https://pubmed.ncbi.nlm.nih.gov/32101422Test -
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المؤلفون: Ying Zhai, De-Yi Yang, Ernest Asante-Appiah, Lei Chen, Haiqun Tang, Paul Ingravallo, Amin A. Nomeir, John P. Caldwell, Ling Tong, Guowei Zhou, Wensheng Yu, Yueheng Jiang, Oleg Selyutin, Anilkumar G. Nair, Seong Heon Kim, Rong Liu, Joseph A. Kozlowski, Qingbei Zeng, Stuart B. Rosenblum, Michael P. Dwyer, Rong Kong, Ellen Xia, Sony Agrawal, Robert Mazzola, Bandarpalle B. Shankar, Kerry Keertikar
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:1954-1957
مصطلحات موضوعية: 0301 basic medicine, Genotype, Proline, Silylation, viruses, Clinical Biochemistry, Pharmaceutical Science, Hepacivirus, Viral Nonstructural Proteins, Pharmacology, Virus Replication, Antiviral Agents, Heterocyclic Compounds, 4 or More Rings, Biochemistry, 03 medical and health sciences, Dogs, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Pharmacokinetics, Drug Discovery, Animals, Humans, Potency, NS5A, Molecular Biology, Chemistry, Organic Chemistry, virus diseases, Haplorhini, biochemical phenomena, metabolism, and nutrition, digestive system diseases, In vitro, Rats, Regimen, 030104 developmental biology, Molecular Medicine, 030211 gastroenterology & hepatology, Half-Life
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dd2480c8ed858188f3382243eccdd83Test
https://doi.org/10.1016/j.bmcl.2018.03.049Test