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1دورية أكاديمية
المؤلفون: Mani Suresh, Raju Rajesh, Arumugam Natarajan, Almansour Abdulrahman I., Suresh Kumar Raju, Perumal Karthikeyan
المصدر: Green Processing and Synthesis, Vol 12, Iss 1, Pp 527-92 (2023)
مصطلحات موضوعية: tandem multicomponent reaction, eco-friendly protocol, solid state melt reaction, pyrrolo[3,2-c]quinolinone/pyrrolizino[2,3-c]quinolinone, Chemistry, QD1-999
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2191-9550Test
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2دورية أكاديمية
المؤلفون: Faisal Aziz, Kanamata Reddy, Virneliz Fernandez Vega, Raja Dey, Katherine A. Hicks, Sumitha Rao, Luis Ortiz Jordan, Emery Smith, Justin Shumate, Louis Scampavia, Nicholas Carpino, Timothy P. Spicer, Jarrod B. French
مصطلحات موضوعية: Biochemistry, Medicine, Microbiology, Cell Biology, Genetics, Pharmacology, Immunology, Developmental Biology, Cancer, Infectious Diseases, Virology, Chemical Sciences not elsewhere classified, reveals key interactions, provide foundational tools, poor cell permeability, crystal structure confirmed, cell receptor signaling, histidine phosphatase activity, sar analysis indicates, >)- quinolinone derivative, 000 compound high, 50 sub, 1 enzyme activity, sts phosphatase activity, phosphatase activity, 1h <, throughput screen, studies demonstrate, small library, significant resistance
الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c01763.s001Test
https://figshare.com/articles/journal_contribution/Rebamipide_and_Derivatives_are_Potent_Selective_Inhibitors_of_Histidine_Phosphatase_Activity_of_the_Suppressor_of_T_Cell_Receptor_Signaling_Proteins/25043322Test -
3دورية أكاديمية
المؤلفون: Chongqing Pan, Hongwei Sun, Yonglei Du, Wenbin Wang, Lingling Xu, Yu Hu, Manzhou Zhu
مصطلحات موضوعية: Biochemistry, Cell Biology, Biotechnology, Ecology, Infectious Diseases, Virology, Chemical Sciences not elsewhere classified, tedious synthetic routes, fused quinolinone products, fused heterocyclic catalysts, fused heterocycles represent, paracyclophanecarboxamide substrates, important scaffold, good yields, concise protocol, 84 %)
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4دورية أكاديمية
المصدر: Drug Design, Development and Therapy, Vol Volume 16, Pp 1495-1514 (2022)
مصطلحات موضوعية: alzheimer’s disease, cholinesterase, monoamine oxidase, 4-dihydro-2(1h)-quinolinone, dithiocarbamate, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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5دورية أكاديمية
المؤلفون: Wennan Zhao, Mingxia Song, Yi Hua, Yangnv Zhu, Wenli Liu, Qishan Xia, Xianqing Deng, Yushan Huang
المصدر: Molecules; Volume 28; Issue 4; Pages: 1987
مصطلحات موضوعية: quinolinone, triazole, antidepressant, antiseizure, anticonvulsant, forced swim test, GABA, maximal electroshock seizure
جغرافية الموضوع: agris
وصف الملف: application/pdf
العلاقة: Medicinal Chemistry; https://dx.doi.org/10.3390/molecules28041987Test
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6دورية أكاديمية
المؤلفون: Manzoor, Shoaib, Gabr, Moustafa T, Nafie, Mohamed S, Raza, Md Kausar, Khan, Ashma, Nayeem, Shahid M, Arafa, Reem K, Hoda, Nasimul
المصدر: ACS Chem Neurosci ; ISSN:1948-7193 ; Volume:15 ; Issue:3
مصطلحات موضوعية: Alzheimer’s disease, acetylcholinesterase, amyloid-beta, quinolinone hybrids
العلاقة: https://doi.org/10.1021/acschemneuro.3c00588Test; https://pubmed.ncbi.nlm.nih.gov/38149821Test
الإتاحة: https://doi.org/10.1021/acschemneuro.3c00588Test
https://pubmed.ncbi.nlm.nih.gov/38149821Test -
7دورية أكاديمية
المؤلفون: Jhesua Valencia, Vivian Rubio, Gloria Puerto, Luisa Vasquez, Anthony Bernal, José R. Mora, Sebastian A. Cuesta, José Luis Paz, Braulio Insuasty, Rodrigo Abonia, Jairo Quiroga, Alberto Insuasty, Andres Coneo, Oscar Vidal, Edgar Márquez, Daniel Insuasty
المصدر: Antibiotics, Vol 12, Iss 1, p 61 (2022)
مصطلحات موضوعية: Mycobacterium tuberculosis, QSAR, docking, quinolinone, thiosemicarbazone, molecular dynamics and cytotoxicity, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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8دورية أكاديمية
المصدر: Pharmaceutics, Vol 14, Iss 12, p 2571 (2022)
مصطلحات موضوعية: cancer, MDR, olaparib, quinolinone, PARP1, selenium, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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9دورية أكاديمية
المؤلفون: Yu Zheng (2950), Zhi-Wei Wang (687399), Wen-Shuo Cheng (10331532), Zhen-Zhen Xie (6504290), Xian-Chen He (52255), Yan-Shan Chen (10331529), Kai Chen (129938), Hao-Yue Xiang (3328260), Xiao-Qing Chen (426077), Hua Yang (120668)
مصطلحات موضوعية: Biochemistry, Microbiology, Molecular Biology, Space Science, Environmental Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, 3 ‑( benzopyrrole, wittig cascade, successfully performing, situ reduction, significantly expanding, rationally combining, rapid assembly, quinolinone framework, privileged skeleton, pot process, first time, facilely synthesized, chemical space, catalytic manner, benzaldehyde derivatives, amino group, >- hydroxy
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10دورية أكاديمية
المؤلفون: Jie Fu, Fengqi Bao, Min Gu, Jing Liu, Zhipeng Zhang, Jiaoli Ding, Sai-Sai Xie, Jinsong Ding
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 118-128 (2020)
مصطلحات موضوعية: dithiocarbamate, quinolinone, cholinesterase, alzheimer’s disease, multifunctional inhibitors, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource