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1دورية أكاديمية
المؤلفون: James K. Morelli, Paul J. Ciaccio
المصدر: Journal of Toxicology, Vol 2013 (2013)
مصطلحات موضوعية: Toxicology. Poisons, RA1190-1270
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Linda R. Barone, Scott Boyer, James R. Damewood, James Fikes, Paul J. Ciaccio
المصدر: Journal of Toxicology, Vol 2012 (2012)
مصطلحات موضوعية: Toxicology. Poisons, RA1190-1270
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Mitchell H. Keylor (8615976), Anmol Gulati (1314951), Solomon D. Kattar (11888244), Rebecca E. Johnson (1361724), Ryan W. Chau (11888247), Kaila A. Margrey (1849126), Michael J. Ardolino (2154361), Cayetana Zarate (1516576), Kelsey E. Poremba (3903853), Vladimir Simov (2534833), Gregori J. Morriello (2645770), John J. Acton (11888250), Barbara Pio (1601539), Xin Yan (17064), Rachel L. Palte (8299626), Spencer E. McMinn (9931798), Lisa Nogle (2160265), Charles A. Lesburg (1834624), Donovon Adpressa (8448369), Shishi Lin (752964), Santhosh Neelamkavil (2679916), Ping Liu (156158), Jing Su (23377), Laxminarayan G. Hegde (2480896), Janice D. Woodhouse (8299629), Robert Faltus (11888253), Tina Xiong (6095357), Paul J. Ciaccio (11888256), Jennifer Piesvaux (5987792), Karin M. Otte (2459014), Harold B. Wood (1665394), Matthew E. Kennedy (2026285), David Jonathan Bennett (7456754), Erin F. DiMauro (797168), Matthew J. Fell (3839692), Peter H. Fuller (2400580)
مصطلحات موضوعية: Biochemistry, Medicine, Genetics, Neuroscience, Pharmacology, Biotechnology, Evolutionary Biology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, Information Systems not elsewhere classified, stereochemical design elements, hydrogen bond donor, friendly profile typified, central nervous system, selective lrrk2 inhibitors, encouraging brain penetration, 22 b, structural enablement, rigorous hit, quality molecules, preclinical models, pd ), parkinson ’, mediated efflux, low levels, functionally linked, enhancing increase
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4Early-Onset albuminuria and Associated Renal Pathology in Leucine-Rich Repeat Kinase 2 Knockout Rats
المؤلفون: Yi-Zhong Gu, Katerina Vlasakova, Glen Miller, Nicholas T. Gatto, Paul J. Ciaccio, Sabu Kuruvilla, Elizabeth G. Besteman, Roger Smith, Spencer J. Reynolds, Rupesh P. Amin, Warren E. Glaab, Gordon Wollenberg, Jose Lebron, Frank D. Sistare
المصدر: Toxicologic Pathology. :019262332311628
مصطلحات موضوعية: Cell Biology, Toxicology, Molecular Biology, Pathology and Forensic Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::ca81b65118f034c663e621457909c3ffTest
https://doi.org/10.1177/01926233231162809Test -
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المؤلفون: Frederique M. Poulet, J. Michael Ellis, Matthew E. Kennedy, Carrie G. Markgraf, Lauren M Timmins, Dianne K. Bryce, Sabu Kuruvilla, Janice D Woodhouse, Matthew J. Fell, Karin M. Otte, Christopher Ware, Laxminarayan G Hegde, Matthew L. Maddess, Paul J Ciaccio
المصدر: Journal of Pharmacology and Experimental Therapeutics. 377:11-19
مصطلحات موضوعية: Male, 0301 basic medicine, Indazoles, Parkinson's disease, Morpholines, Pharmacology, Leucine-Rich Repeat Serine-Threonine Protein Kinase-2, Mice, 03 medical and health sciences, 0302 clinical medicine, In vivo, medicine, Animals, Kinase activity, Protein Kinase Inhibitors, Lung, Kinase, business.industry, medicine.disease, Pulmonary Surfactant-Associated Protein C, LRRK2, nervous system diseases, Mice, Inbred C57BL, Pyrimidines, 030104 developmental biology, medicine.anatomical_structure, Alveolar Epithelial Cells, Molecular Medicine, Immunohistochemistry, business, 030217 neurology & neurosurgery, Protein C, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::50f51a63a6fe69d40bfa5ed39544e2ddTest
https://doi.org/10.1124/jpet.120.000217Test -
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المؤلفون: Mitchell H. Keylor, Anmol Gulati, Solomon D. Kattar, Rebecca E. Johnson, Ryan W. Chau, Kaila A. Margrey, Michael J. Ardolino, Cayetana Zarate, Kelsey E. Poremba, Vladimir Simov, Gregori J. Morriello, John J. Acton, Barbara Pio, Xin Yan, Rachel L. Palte, Spencer E. McMinn, Lisa Nogle, Charles A. Lesburg, Donovon Adpressa, Shishi Lin, Santhosh Neelamkavil, Ping Liu, Jing Su, Laxminarayan G. Hegde, Janice D. Woodhouse, Robert Faltus, Tina Xiong, Paul J. Ciaccio, Jennifer Piesvaux, Karin M. Otte, Harold B. Wood, Matthew E. Kennedy, David Jonathan Bennett, Erin F. DiMauro, Matthew J. Fell, Peter H. Fuller
المصدر: Journal of medicinal chemistry. 65(1)
مصطلحات موضوعية: Antiparkinson Agents, Models, Molecular, Structure-Activity Relationship, Drug Design, Drug Discovery, Quinazolines, Molecular Medicine, Biological Availability, Brain, Humans, Leucine-Rich Repeat Serine-Threonine Protein Kinase-2, Protein Kinase Inhibitors
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6720c280fccf3e18653a864a196348adTest
https://pubmed.ncbi.nlm.nih.gov/34967623Test -
7Optimization of brain-penetrant picolinamide derived leucine-rich repeat kinase 2 (LRRK2) inhibitors
المؤلفون: Blair T. Lapointe, Jack D. Scott, Xin Cindy Yan, Haiqun Tang, Janice D Woodhouse, Kaleen Konrad Childers, Robert Faltus, Erin F. DiMauro, Solomon Kattar, Charles S. Yeung, Ravi Kurukulasuriya, Vladimir Simov, Hakan Gunaydin, Anmol Gulati, Joey L. Methot, Rachel L. Palte, Ellen C. Minnihan, Greg Morriello, J. Michael Ellis, Harold B. Wood, Santhosh Neelamkavil, Karin M. Otte, Michael J. Ardolino, Barbara Pio, Ping Liu, Laxminarayan G Hegde, Matthew J. Fell, Vanessa L. Rada, Peter Fuller, Paul J Ciaccio
المصدر: RSC Med Chem
مصطلحات موضوعية: Pharmacology, 0303 health sciences, Trifluoromethyl, Chemistry, Metabolite, Organic Chemistry, Pharmaceutical Science, Pyrazole, Leucine-rich repeat, Biochemistry, LRRK2, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, 030220 oncology & carcinogenesis, Drug Discovery, Molecular Medicine, Kinome, Penetrant (biochemical), Linker, 030304 developmental biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6c8d45ea7dd7adda70471298a4476afaTest
https://europepmc.org/articles/PMC8292993Test/ -
8دورية أكاديمية
المؤلفون: Joseph Milano, Jenny Mckay, Claude Dagenais, Linda Foster-brown, Reto Gadient, Robert T. Jacobs, Anna Zacco, Barry Greenberg, Paul J, Paul J. Ciaccio, Astrazeneca Pharmaceuticals
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
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9دورية أكاديمية
المؤلفون: Paul J Ciaccio, Hongxie Shen, Anil K Jaiswal, Matthew H Lyttle, Kenneth D Tew, P J C, H S, A K J, K D T ), Terrapin
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
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المؤلفون: Marie Blais, Douglas Ferguson, Mark Pietras, Jim Fikes, Abhishek G. Sathe, Sally A. Price, Anshul Gupta, Melanie Galvin, Michael R. Hale, Robert L. Walsky, Yvonne P. Dragan, Frank McGrath, Crystal Brown, Paul J. Ciaccio, Gunther Kern, Matthew Wagoner, Letitia Cheatham, Nakpangi Johnson, Patricia Bentley, Natalie Keirstead, Debra Snow, Wenli Luo, Jennifer C. Sasaki
المصدر: Toxicological Sciences. 137:278-291
مصطلحات موضوعية: Male, medicine.medical_specialty, Cell Survival, medicine.drug_class, Polymyxin, Pharmacology, Toxicology, Cell Line, Nephrotoxicity, medicine, Animals, Rats, Wistar, Intensive care medicine, Blood urea nitrogen, Polymyxin B, Kidney, Dose-Response Relationship, Drug, Colistin, business.industry, Acute kidney injury, Prognosis, medicine.disease, Anti-Bacterial Agents, Rats, Early Diagnosis, medicine.anatomical_structure, Data Interpretation, Statistical, Biomarker (medicine), Kidney Diseases, business, Biomarkers, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::44e7ce12b5cc757b27009c075c2c9b9dTest
https://doi.org/10.1093/toxsci/kft247Test