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المؤلفون: Bogren, Mats, Soltesz, Monica, Hjorth, Stephan
المصدر: Frontiers in Psychiatry. 13
مصطلحات موضوعية: Antipsychotic polypharmacy, cognitive symptoms of schizophrenia, DA D2/D3 partial agonism, negative symptoms (schizophrenia), psychosocial symptoms, quality-of-life, reward system, Medicin och hälsovetenskap, Klinisk medicin, Psykiatri, Medical and Health Sciences, Clinical Medicine, Psychiatry
الوصول الحر: https://lup.lub.lu.se/record/6122ddb7-b386-4df7-a274-94032ab292b9Test
http://dx.doi.org/10.3389/fpsyt.2022.887547Test -
2دورية أكاديمية
المؤلفون: Stuart H. Isaacson, Robert A. Hauser, Rajesh Pahwa, David Gray, Sridhar Duvvuri
المصدر: Clinical Parkinsonism & Related Disorders, Vol 9, Iss , Pp 100212- (2023)
مصطلحات موضوعية: Parkinson’s disease, Dopamine agonists, D1 receptors, D2 receptors, Partial agonism, Dopamine receptor selectivity, Neurology. Diseases of the nervous system, RC346-429
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2590112523000300Test; https://doaj.org/toc/2590-1125Test
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3دورية أكاديمية
المؤلفون: Chan, John D, Cupit, Pauline M, Gunaratne, Gihan S, McCorvy, John D, Yang, Yang, Stoltz, Kristen, Webb, Thomas R, Dosa, Peter I, Roth, Bryan L, Abagyan, Ruben, Cunningham, Charles, Marchant, Jonathan S
المصدر: Nature communications. 8(1)
مصطلحات موضوعية: Mesenteric Arteries, Mesenteric Veins, Cell Line, Animals, Humans, Mice, Schistosoma mansoni, Schistosomiasis mansoni, Praziquantel, Receptor, Serotonin, 5-HT2B, Anthelmintics, Myography, Vasoconstriction, Computer Simulation, Female, Drug Partial Agonism, Serotonin 5-HT2 Receptor Agonists
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/1jh768mvTest
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4دورية أكاديمية
المصدر: Pharmaceuticals (Basel) ; ISSN:1424-8247 ; Volume:17 ; Issue:6
مصطلحات موضوعية: 5-HT1A receptors, 8-OH-DAPT, buspirone, depression, development, isolation rearing, partial agonism
العلاقة: https://doi.org/10.3390/ph17060717Test; https://pubmed.ncbi.nlm.nih.gov/38931384Test; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC11206366Test/
الإتاحة: https://doi.org/10.3390/ph17060717Test
https://pubmed.ncbi.nlm.nih.gov/38931384Test
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC11206366Test/ -
5دورية أكاديمية
المؤلفون: Leijten-van de Gevel, Iris A., van Herk, Kim H.N., de Vries, Rens M.J.M., Ottenheym, Nicolaas J., Ottmann, Christian, Brunsveld, Luc
المصدر: Leijten-van de Gevel , I A , van Herk , K H N , de Vries , R M J M , Ottenheym , N J , Ottmann , C & Brunsveld , L 2022 , ' Indazole MRL-871 interacts with PPARγ via a binding mode that induces partial agonism ' , Bioorganic and Medicinal Chemistry , vol. 68 , 116877 . https://doi.org/10.1016/j.bmc.2022.116877Test
مصطلحات موضوعية: Co-crystal structure, Nuclear Receptors, Partial Agonism, PPARγ, RORγt, Nuclear Receptor Subfamily 1, Group F, Member 3/metabolism, Protein Structure, Secondary, PPAR gamma/agonists, Indazoles/pharmacology, Ligands
وصف الملف: application/pdf
الإتاحة: https://doi.org/10.1016/j.bmc.2022.116877Test
https://research.tue.nl/en/publications/a3a998b0-c575-433d-a230-7f4bc2b62470Test
https://pure.tue.nl/ws/files/211567189/1_s2.0_S0968089622002693_main.pdfTest
http://www.scopus.com/inward/record.url?scp=85131964889&partnerID=8YFLogxKTest -
6دورية أكاديمية
المؤلفون: Staus, Dean P, Strachan, Ryan T, Manglik, Aashish, Pani, Biswaranjan, Kahsai, Alem W, Kim, Tae Hun, Wingler, Laura M, Ahn, Seungkirl, Chatterjee, Arnab, Masoudi, Ali, Kruse, Andrew C, Pardon, Els, Steyaert, Jan, Weis, William I, Prosser, R Scott, Kobilka, Brian K, Costa, Tommaso, Lefkowitz, Robert J
المصدر: Nature. 535(7612)
مصطلحات موضوعية: Humans, Isoproterenol, Receptors, Adrenergic, beta-2, Ligands, Crystallography, X-Ray, Nuclear Magnetic Resonance, Biomolecular, Allosteric Regulation, Allosteric Site, Protein Conformation, Models, Molecular, Drug Partial Agonism, Protein Stability, Adrenergic beta-2 Receptor Agonists, Single-Domain Antibodies, Crystallography, X-Ray, Models, Molecular, Nuclear Magnetic Resonance, Biomolecular, Receptors, Adrenergic, beta-2, General Science & Technology
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/4sf4012jTest
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7دورية أكاديمية
المؤلفون: Vafabakhsh, Reza, Levitz, Joshua, Isacoff, Ehud Y
المصدر: Nature. 524(7566)
مصطلحات موضوعية: Animals, Humans, Rats, Receptors, Metabotropic Glutamate, Ligands, Fluorescence Resonance Energy Transfer, Binding Sites, Protein Conformation, Protein Binding, Models, Biological, Models, Molecular, Drug Partial Agonism, General Science & Technology
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/8q29z78hTest
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8دورية أكاديمية
المؤلفون: Phil Pickford, Maria Lucey, Roxana-Maria Rujan, Emma Rose McGlone, Stavroula Bitsi, Fiona B. Ashford, Ivan R. Corrêa, David J. Hodson, Alejandra Tomas, Giuseppe Deganutti, Christopher A. Reynolds, Bryn M. Owen, Tricia M. Tan, James Minnion, Ben Jones, Stephen R. Bloom
المصدر: Molecular Metabolism, Vol 51, Iss , Pp 101242- (2021)
مصطلحات موضوعية: GLP-1, Glucagon, Oxyntomodulin, Biased agonism, Partial agonism, β-arrestin, Internal medicine, RC31-1245
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S2212877821000879Test; https://doaj.org/toc/2212-8778Test
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9دورية أكاديمية
المؤلفون: Taylor, Colin, Riley, Andrew M, Dupont, Genevieve, Rahman, Taufiq, Potter, Barry VL, Rossi, Ana M
مصطلحات موضوعية: Ca(2+) signaling, IP(3) receptor, IP(3) receptor antagonist, endoplasmic reticulum, intracellular Ca(2+) stores, partial agonist, quantal Ca(2+) release, receptor inactivation, Animals, Calcium, Calcium Signaling, Chickens, Drug Partial Agonism, HEK293 Cells, Humans, Inositol 1,4,5-Trisphosphate, Inositol 1,4,5-Trisphosphate Receptors, Inositol Phosphates, Time Factors
وصف الملف: application/pdf
الإتاحة: https://doi.org/10.17863/CAM.83531Test
https://www.repository.cam.ac.uk/handle/1810/336106Test -
10دورية أكاديمية
المؤلفون: Alessandro Bonifazi (1322385), Amy H. Newman (6191750), Thomas M. Keck (1322388), Silvia Gervasoni (6169202), Giulio Vistoli (1408930), Fabio Del Bello (7399721), Gianfabio Giorgioni (2519272), Pegi Pavletić (9400428), Wilma Quaglia (1484305), Alessandro Piergentili (1484281)
مصطلحات موضوعية: Biochemistry, Cell Biology, Genetics, Neuroscience, Pharmacology, Biotechnology, Evolutionary Biology, Immunology, Cancer, Mental Health, Infectious Diseases, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, substituted butyl chain, promising starting point, novel antipsychotic agents, interesting multitarget behavior, 2c sub, 2a sub, 1a sub, f -/ 3, r partial agonists, 3 sub, 3 b, r partial agonism, 4 sub, 2 sub, 6 b, n <, r agonism