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1دورية أكاديمية
المؤلفون: Rasco, Drew W, Medina, Theresa, Corrie, Pippa, Pavlick, Anna C, Middleton, Mark R, Lorigan, Paul, Hebert, Chris, Plummer, Ruth, Larkin, James, Agarwala, Sanjiv S, Daud, Adil I, Qiu, Jiaheng, Bozon, Viviana, Kneissl, Michelle, Barry, Elly, Olszanski, Anthony J
المصدر: Cancer chemotherapy and pharmacology. 92(1)
مصطلحات موضوعية: Humans, Neoplasms, Melanoma, Skin Neoplasms, Neoplasms, Second Primary, Proto-Oncogene Proteins B-raf, Mitogen-Activated Protein Kinase Kinases, Protein Kinase Inhibitors, Maximum Tolerated Dose, Adult, BRAF, Pan-RAF inhibitor, Phase 1, Tovorafenib, Clinical Trials and Supportive Activities, Clinical Research, Cancer, 6.1 Pharmaceuticals, Evaluation of treatments and therapeutic interventions, Pharmacology and Pharmaceutical Sciences, Oncology & Carcinogenesis
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/6jq463hgTest
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2دورية أكاديمية
المؤلفون: Yu Gao, Eva-Maria Packeiser, Sophia Wendt, Anett Sekora, Jessika-Maximiliane V. Cavalleri, Barbara Pratscher, Moosheer Alammar, Maja Hühns, Bertram Brenig, Christian Junghanss, Ingo Nolte, Hugo Murua Escobar
المصدر: Genes, Vol 15, Iss 2, p 202 (2024)
مصطلحات موضوعية: equine malignant melanoma, canine malignant melanoma, Pan-RAF inhibitor, LY3009120, DNA sequencing, genetic evaluation, Genetics, QH426-470
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Rasco, DW, Medina, T, Corrie, P, Pavlick, AC, Middleton, MR, Lorigan, P, Hebert, C, Plummer, R, Larkin, J, Agarwala, SS, Daud, AI, Qiu, J, Bozon, V, Kneissl, M, Barry, E, Olszanski, AJ
المساهمون: Larkin, James
مصطلحات موضوعية: BRAF, Melanoma, Pan-RAF inhibitor, Phase 1, Tovorafenib, Adult, Humans, Proto-Oncogene Proteins B-raf, Neoplasms, Skin Neoplasms, Protein Kinase Inhibitors, Second Primary, Mitogen-Activated Protein Kinase Kinases, Maximum Tolerated Dose
جغرافية الموضوع: Germany
وصف الملف: Print-Electronic; 28; application/pdf
العلاقة: Cancer Chemotherapy and Pharmacology, 2023, 92 (1), pp. 15 - 28; https://repository.icr.ac.uk/handle/internal/5936Test
الإتاحة: https://doi.org/10.1007/s00280-023-04544-5Test
https://repository.icr.ac.uk/handle/internal/5936Test -
4دورية أكاديمية
المؤلفون: Gao, Yu, Packeiser, Eva-Maria, Wendt, Sophia, Sekora, Anett, Cavalleri, Jessika-Maximiliane V, Pratscher, Barbara, Alammar, Moosheer, Hühns, Maja, Brenig, Bertram, Junghanss, Christian, Nolte, Ingo, Murua Escobar, Hugo
المصدر: Genes (Basel) ; ISSN:2073-4425 ; Volume:15 ; Issue:2
مصطلحات موضوعية: DNA sequencing, LY3009120, Pan-RAF inhibitor, canine malignant melanoma, cellular response, equine malignant melanoma, genetic evaluation
العلاقة: https://doi.org/10.3390/genes15020202Test; https://pubmed.ncbi.nlm.nih.gov/38397192Test; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10887541Test/
الإتاحة: https://doi.org/10.3390/genes15020202Test
https://pubmed.ncbi.nlm.nih.gov/38397192Test
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10887541Test/ -
5دورية أكاديمية
المؤلفون: Atefi, Mohammad, Titz, Bjoern, Avramis, Earl, Ng, Charles, Wong, Deborah JL, Lassen, Amanda, Cerniglia, Michael, Escuin-Ordinas, Helena, Foulad, David, Comin-Anduix, Begonya, Graeber, Thomas G, Ribas, Antoni
المصدر: Molecular Cancer. 14(1)
مصطلحات موضوعية: Biochemistry and Cell Biology, Biomedical and Clinical Sciences, Oncology and Carcinogenesis, Biological Sciences, Cancer, Development of treatments and therapeutic interventions, 5.1 Pharmaceuticals, Apoptosis, Cell Cycle, Cell Line, Tumor, Cell Proliferation, Cyclin D1, Cyclin D3, GTP Phosphohydrolases, Glycogen Synthase Kinase 3, Glycogen Synthase Kinase 3 beta, Humans, MAP Kinase Signaling System, Melanoma, Membrane Proteins, Mutation, Signal Transduction, Transcription, Genetic, raf Kinases, NRAS, MAPK, MEK inhibitor, pan-RAF inhibitor, Oncology & Carcinogenesis, Biochemistry and cell biology, Oncology and carcinogenesis
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/15p746hrTest
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6دورية أكاديمية
المؤلفون: Malcolm P. Huestis (10493092), Darlene Dela Cruz (10493095), Antonio G. DiPasquale (1274730), Matthew R. Durk (7052600), Charles Eigenbrot (1346406), Paul Gibbons (114343), Alberto Gobbi (1508113), Thomas L. Hunsaker (3160575), Hank La (438084), Dennis H. Leung (2106256), Wendy Liu (2057074), Shiva Malek (1346394), Mark Merchant (282025), John G. Moffat (413533), Christine S. Muli (10493098), Christine J. Orr (10493101), Brendan T. Parr (2342548), Frances Shanahan (655624), Christopher J. Sneeringer (10493104), Weiru Wang (640332), Ivana Yen (1346373), Jianping Yin (557395), Michael Siu (1503160), Joachim Rudolph (1464982)
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Cell Biology, Molecular Biology, Pharmacology, Cancer, Hematology, Infectious Diseases, Virology, Space Science, Chemical Sciences not elsewhere classified, Physical Sciences not elsewhere classified, kinase selectivity, vivo evaluation, solubility, Combination Treatment, MEK inhibitor cobimetinib, tumor growth inhibition, NH functionality, pathway inhibition, Strategic substitution, fluoroquinazolinone hinge-binding motif, xenograft mouse model, C 5 position, RAF-specific residue interactions, aryl urea RAF inhibitors, type II pan-RAF inhibitor GNE -0749, Targeting KRAS Mutant Cancers
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7
المؤلفون: Drew W. Rasco, Theresa Medina, Pippa Corrie, Anna C. Pavlick, Mark R. Middleton, Paul Lorigan, Chris Hebert, Ruth Plummer, James Larkin, Sanjiv S. Agarwala, Adil I. Daud, Jiaheng Qiu, Viviana Bozon, Michelle Kneissl, Elly Barry, Anthony J. Olszanski
المساهمون: Barry, Elly [0000-0002-6890-2444], Apollo - University of Cambridge Repository
المصدر: Cancer chemotherapy and pharmacology, vol 92, iss 1
مصطلحات موضوعية: Adult, Proto-Oncogene Proteins B-raf, Cancer Research, Skin Neoplasms, Maximum Tolerated Dose, Clinical Trials and Supportive Activities, Phase 1, Toxicology, BRAF, Clinical Research, Neoplasms, Humans, Pharmacology (medical), Oncology & Carcinogenesis, Melanoma, Protein Kinase Inhibitors, Pan-RAF inhibitor, Cancer, Pharmacology, Mitogen-Activated Protein Kinase Kinases, Evaluation of treatments and therapeutic interventions, Neoplasms, Second Primary, Pharmacology and Pharmaceutical Sciences, Second Primary, Oncology, 6.1 Pharmaceuticals, Tovorafenib
وصف الملف: application/pdf; application/zip; text/xml
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6be879ecf897194f5e93f0a32cbcfa4dTest
https://www.repository.cam.ac.uk/handle/1810/350906Test -
8دورية أكاديمية
المؤلفون: Park, Siyeon, Kim, Tae Min, Cho, Sung-Yup, Kim, Soyeon, Oh, Yumi, Kim, Miso, Keam, Bhumsuk, Kim, Dong-Wan, Heo, Dae Seog
المساهمون: 조성엽, 김동완, 허대석, Cho, Sung-Yup, Kim, Dong-Wan, Heo, Dae Seog
مصطلحات موضوعية: INHIBITION, GENOME, BRAF, PATIENT, PLK1, MEK, NRAS-mutant lung cancer, High-throughput screening, Pan-RAF inhibitor, PLK1 inhibitor
العلاقة: Cancer Letters, Vol.495, pp.135-144; 118788; https://hdl.handle.net/10371/171807Test; 000590212800003; 2-s2.0-85091652639
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9دورية أكاديمية
المؤلفون: Rasco, Drew W., Medina, Theresa, Corrie, Pippa, Pavlick, Anna C., Middleton, Mark R., Lorigan, Paul, Hebert, Chris, Plummer, Ruth, Larkin, James, Agarwala, Sanjiv S., Daud, Adil I., Qiu, Jiaheng, Bozon, Viviana, Kneissl, Michelle, Barry, Elly, Olszanski, Anthony J.
مصطلحات موضوعية: Phase 1, Pan-RAF inhibitor, Melanoma, BRAF, Tovorafenib
وصف الملف: application/pdf; application/zip; text/xml
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10دورية أكاديمية
المؤلفون: Yu Fu, Yuanyuan Wang, Shanhe Wan, Zhonghuang Li, Guangfa Wang, Jiajie Zhang, Xiaoyun Wu
المصدر: Molecules; Volume 22; Issue 4; Pages: 542
مصطلحات موضوعية: DFG-out, pan-RAF inhibitor, 1 H -pyrazolo[3,4- d ]pyrimidine derivatives, biological activities, molecular docking, molecular dynamics simulation
جغرافية الموضوع: agris
وصف الملف: application/pdf
العلاقة: Medicinal Chemistry; https://dx.doi.org/10.3390/molecules22040542Test