-
1دورية أكاديمية
المؤلفون: Nancy H.C. Loos, Irene A. Retmana, Jamie Rijmers, Yaogeng Wang, Changpei Gan, Maria C. Lebre, Rolf W. Sparidans, Jos H. Beijnen, Alfred H. Schinkel
المصدر: Biomedicine & Pharmacotherapy, Vol 166, Iss , Pp 115304- (2023)
مصطلحات موضوعية: Adagrasib, KRASG12C inhibitor, ABCB1/P-glycoprotein, ABCG2/Breast cancer resistance protein, Cytochrome P450 3A, Carboxylesterase 1, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S0753332223010958Test; https://doaj.org/toc/0753-3322Test
-
2دورية أكاديمية
المؤلفون: Nancy H.C. Loos, Jos H. Beijnen, Alfred H. Schinkel
المصدر: Biomedicine & Pharmacotherapy, Vol 162, Iss , Pp 114636- (2023)
مصطلحات موضوعية: Ritonavir, CYP3A, P-glycoprotein, Inhibition, Induction, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S0753332223004249Test; https://doaj.org/toc/0753-3322Test
-
3
المؤلفون: Nancy H.C. Loos, Hilde Rosing, Margarida L. F. Martins, Maria C. Lebre, Danielle de Jong, Alfred H. Schinkel, Jos H. Beijnen, Matthijs M. Tibben, Sümeyra Mucuk
المصدر: Molecular pharmaceutics. 18(12)
مصطلحات موضوعية: Genetically modified mouse, Indazoles, Abcg2, CYP3A, Metabolite, Pharmaceutical Science, Pharmacology, Poly(ADP-ribose) Polymerase Inhibitors, Madin Darby Canine Kidney Cells, chemistry.chemical_compound, Mice, Dogs, Pharmacokinetics, Piperidines, Tetrahydroisoquinolines, Drug Discovery, Distribution (pharmacology), Animals, Cytochrome P-450 CYP3A, Tissue Distribution, ATP Binding Cassette Transporter, Subfamily B, Member 1, CYP3A4, biology, Chemistry, Brain, Biological Transport, In vitro, Intestines, biology.protein, Molecular Medicine, Acridines
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c061d7a3983347bd5f4f1d4ccf059ff2Test
https://pubmed.ncbi.nlm.nih.gov/34730366Test -
4
المؤلفون: Nancy H.C. Loos, Alejandra Martínez-Chávez, Hilde Rosing, Alfred H. Schinkel, Jos H. Beijnen, Matthijs M. Tibben, Maria C. Lebre
المصدر: Pharmacological Research. 178:105954
مصطلحات موضوعية: CYP3A, Cmax, Aminopyridines, Pharmacology, Madin Darby Canine Kidney Cells, Mice, Dogs, Pharmacokinetics, Cyclin-dependent kinase, Oral administration, medicine, ATP Binding Cassette Transporter, Subfamily G, Member 2, Animals, Cytochrome P-450 CYP3A, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Active metabolite, Mice, Knockout, biology, Chemistry, Brain, Small intestine, Neoplasm Proteins, medicine.anatomical_structure, Pharmaceutical Preparations, Toxicity, biology.protein, Benzimidazoles
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5698acb6dea4155fdac3f38a29524799Test
https://doi.org/10.1016/j.phrs.2021.105954Test -
5دورية أكاديمية
المؤلفون: Nancy H.C. Loos, Margarida L. Ferreira Martins, Jamie Rijmers, Daniëlle de Jong, Maria C. Lebre, Matthijs Tibben, Jos H. Beijnen, Alfred H. Schinkel
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Cell Biology, Genetics, Physiology, Pharmacology, Biotechnology, Mental Health, Infectious Diseases, Computational Biology, Chemical Sciences not elsewhere classified, therefore study determinants, pharmacodynamic mouse studies, parameters showed rescue, oral formulation would, orally applied cabazitaxel, humanized mouse strains, >< sup ><, orally boosted cabazitaxel, boosted oral cabazitaxel, increased plasma auc, intestinal drug disposition, plasma auc, boosted setting, intestinal disposition, ablated strains, > sup, plasma ratio, plasma carboxylesterase
الإتاحة: https://doi.org/10.1021/acs.molpharmaceut.3c01205.s001Test
https://figshare.com/articles/journal_contribution/Interplay_of_Ritonavir-Boosted_Oral_Cabazitaxel_with_the_Organic_Anion-Transporting_Polypeptide_OATP_Uptake_Transporters_and_Carboxylesterase_1_in_Mice/25321868Test