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المؤلفون: Aaron T, Garrison, Douglas L, Orsi, Rory A, Capstick, David, Whomble, Jinming, Li, Trever R, Carter, Andrew S, Felts, Paige N, Vinson, Alice L, Rodriguez, Allie, Han, Krishma, Hajari, Hyekyung P, Cho, Laura B, Teal, Madeline G, Ragland, Masoud, Ghamari-Langroudi, Michael, Bubser, Sichen, Chang, Nathalie C, Schnetz-Boutaud, Olivier, Boutaud, Anna L, Blobaum, Daniel J, Foster, Colleen M, Niswender, P Jeffrey, Conn, Craig W, Lindsley, Carrie K, Jones, Changho, Han
المصدر: Journal of medicinal chemistry. 65(8)
مصطلحات موضوعية: Male, Rats, Sprague-Dawley, Receptor, Muscarinic M5, Dopaminergic Neurons, Receptor, Muscarinic M1, Animals, Opioid-Related Disorders, Receptors, Muscarinic, Rats
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::9138eeec6fc81e9c109df2fed42c17adTest
https://pubmed.ncbi.nlm.nih.gov/35417155Test -
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المؤلفون: Wessel A.C. Burger, Arthur Christopoulos, Jonathan B. Baell, Emma T van der Westhuizen, Geoff Thompson, Christopher J. Langmead, Celine Valant, Patrick R. Gentry, Kunio Hirata, Ziva Vuckovic, Raphaël Rahmani, Swapna Varghese, Patrick M. Sexton, David M. Thal, Alice E. Berizzi, Craig W. Lindsley, Andrew B. Tobin
المصدر: Proceedings of the National Academy of Sciences of the United States of America
مصطلحات موضوعية: Models, Molecular, crystal structure, drug design, Protein Conformation, Allosteric regulation, Ligands, Receptor subtype, 03 medical and health sciences, muscarinic receptor, 0302 clinical medicine, Allosteric Regulation, X-Ray Diffraction, Muscarinic acetylcholine receptor, Extracellular, Inverse agonist, Humans, G protein-coupled receptor, Receptor, 030304 developmental biology, Pharmacology, 0303 health sciences, Multidisciplinary, Binding Sites, Receptor, Muscarinic M5, Ligand, Chemistry, Rational design, Biological Sciences, Receptors, Muscarinic, 3. Good health, Kinetics, Drug development, Crystallization, Neuroscience, 030217 neurology & neurosurgery, Allosteric Site
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d059975532a5f53800def4cf5650944Test
http://europepmc.org/articles/PMC6926013Test -
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المؤلفون: Amir Rafiq, Christian Illig, Wolfgang Kummer, Klaus Deckmann, Melanie Durschnabel, Christian Erdmann, Wolfgang Weidner, Thomas Bschleipfer, Jürgen Wess
المصدر: The FASEB Journal. 32:2903-2910
مصطلحات موضوعية: 0301 basic medicine, Cell, Stimulation, Muscarinic Antagonists, Biochemistry, Mice, 03 medical and health sciences, 0302 clinical medicine, Allosteric Regulation, Urethra, stomatognathic system, Negative feedback, Muscarinic acetylcholine receptor, Genetics, medicine, Animals, Molecular Biology, Mice, Knockout, Receptor, Muscarinic M2, Receptor, Muscarinic M5, medicine.diagnostic_test, Reverse Transcriptase Polymerase Chain Reaction, Urinary Bladder, Overactive, business.industry, Research, fungi, Cystometry, Epithelial Cells, Cell biology, Brush Cell, 030104 developmental biology, medicine.anatomical_structure, Reflex, Cholinergic, business, 030217 neurology & neurosurgery, Biotechnology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cce86ff4b92355f07f228a2e0eda2f6bTest
https://doi.org/10.1096/fj.201700582rTest -
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المؤلفون: Jennie Garcia-Olivares, Aurelio Galli, Gonzalo E. Torres, Susan G. Amara, T Baust, Peter J. Hamilton, S S Harris
المصدر: Molecular Psychiatry. 22:1673-1679
مصطلحات موضوعية: 0301 basic medicine, Dopamine, Dopamine Plasma Membrane Transport Proteins, Biology, Pharmacology, Binding, Competitive, Article, Membrane Potentials, Rats, Sprague-Dawley, 03 medical and health sciences, Cellular and Molecular Neuroscience, Cricetulus, 0302 clinical medicine, GTP-Binding Protein gamma Subunits, parasitic diseases, mental disorders, medicine, Animals, Humans, Receptor, Molecular Biology, Cells, Cultured, Cellular localization, Dopamine transporter, Receptor, Muscarinic M5, Dopaminergic Neurons, GTP-Binding Protein beta Subunits, Dopaminergic, Brain, Transporter, Psychiatry and Mental health, 030104 developmental biology, nervous system, biology.protein, Female, Efflux, 030217 neurology & neurosurgery, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::401cafe43242147a29634f5d480c53a0Test
https://doi.org/10.1038/mp.2017.176Test -
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المؤلفون: Kellie D. Nance, Alexander R. Geanes, P. Jeffrey Conn, Hykeyung P. Cho, Craig W. Lindsley, Carrie K. Jones, Kevin M. McGowan, Jens Meiler
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:4487-4491
مصطلحات موضوعية: 0301 basic medicine, Quantitative structure–activity relationship, Stereochemistry, Clinical Biochemistry, Quantitative Structure-Activity Relationship, Pharmaceutical Science, CHO Cells, Muscarinic Antagonists, Ligands, Biochemistry, Article, 03 medical and health sciences, Cricetulus, Drug Discovery, Virtual screen, Animals, Humans, Molecular Biology, Sulfonyl, chemistry.chemical_classification, Virtual screening, Receptor, Muscarinic M5, Drug discovery, Ligand, Organic Chemistry, Cooperative binding, Combinatorial chemistry, 030104 developmental biology, chemistry, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dff9a41213b4cdedc46065cafa95286bTest
https://doi.org/10.1016/j.bmcl.2016.07.071Test -
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المؤلفون: Robert W, Gould, Barak W, Gunter, Michael, Bubser, Robert T, Matthews, Laura B, Teal, Madeline G, Ragland, Thomas M, Bridges, Aaron T, Garrison, Danny G, Winder, Craig W, Lindsley, Carrie K, Jones
المصدر: ACS Chem Neurosci
مصطلحات موضوعية: Male, Narcotics, Nociception, Receptor, Muscarinic M5, Behavior, Animal, Self Administration, Article, Rats, Rats, Sprague-Dawley, Remifentanil, Allosteric Regulation, Reward, Conditioning, Psychological, Animals, Conditioning, Operant, Cues, Oxycodone
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::01c72225a4a93c4a57187fb0b61623fbTest
https://pubmed.ncbi.nlm.nih.gov/31268669Test -
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المؤلفون: Paulina, Cieślik, Helena, Domin, Agnieszka, Chocyk, Piotr, Gruca, Ewa, Litwa, Agata, Płoska, Adrianna, Radulska, Iwona, Pelikant-Małecka, Piotr, Brański, Leszek, Kalinowski, Joanna M, Wierońska
المصدر: Neuropharmacology. 174
مصطلحات موضوعية: Male, Sulfonamides, Receptor, Muscarinic M5, Dose-Response Relationship, Drug, Pyridines, Receptor, Muscarinic M1, Receptors, Metabotropic Glutamate, Rats, Mice, Animals, Cognitive Dysfunction, Dizocilpine Maleate, Rats, Wistar, Excitatory Amino Acid Antagonists
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::1e50fdb739b861b14a4519362e5ed94bTest
https://pubmed.ncbi.nlm.nih.gov/31785263Test -
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المؤلفون: Aaron M, Bender, Aaron T, Garrison, Craig W, Lindsley
المصدر: ACS chemical neuroscience. 10(3)
مصطلحات موضوعية: Receptor, Muscarinic M5, Allosteric Regulation, Substance-Related Disorders, Drug Discovery, Animals, Humans, Muscarinic Antagonists, Muscarinic Agonists, Nervous System Diseases
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::3e031d56888b0169a26747b4a1e0c249Test
https://pubmed.ncbi.nlm.nih.gov/30280567Test -
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المؤلفون: Guangrong Zheng, Na-Ra Lee, Mahesh Darna, Xuan Zhang, Linda P. Dwoskin
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:5032-5035
مصطلحات موضوعية: Meperidine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Pharmacology, Ligands, Biochemistry, Article, Structure-Activity Relationship, Cricetulus, Drug Discovery, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M5, Muscarinic acetylcholine receptor M4, Animals, Humans, Molecular Biology, Receptor, Muscarinic M3, Receptor, Muscarinic M5, Chemistry, Chinese hamster ovary cell, Receptor, Muscarinic M1, Organic Chemistry, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M1, Affinities, Molecular Medicine, Female
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::852db3d67a8350d441062f4a1151f0d4Test
https://doi.org/10.1016/j.bmcl.2015.10.029Test -
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المؤلفون: Stefan Hallgren, Henrik Viberg, Anders Fredriksson
المصدر: Environmental Toxicology and Pharmacology. 40:409-416
مصطلحات موضوعية: Male, medicine.medical_specialty, Aché, Health, Toxicology and Mutagenesis, Gene Expression, Receptors, Nicotinic, Biology, GPI-Linked Proteins, Toxicology, Mice, chemistry.chemical_compound, Transcription (biology), Internal medicine, Gene expression, Halogenated Diphenyl Ethers, medicine, Animals, Gene, Flame Retardants, Pharmacology, Fluorocarbons, Receptor, Muscarinic M5, Behavior, Animal, Neurotoxicity, Brain, Gene Expression Regulation, Developmental, General Medicine, medicine.disease, Acetylcholinesterase, language.human_language, Endocrinology, Alkanesulfonic Acids, Animals, Newborn, chemistry, Cholinergic system, language, Cholinergic
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3b0d605ca2d76b1eb80d720f035dfd35Test
https://doi.org/10.1016/j.etap.2015.06.014Test