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1دورية أكاديمية
المؤلفون: Baofeng Zhang, Michael P. D’Erasmo, Ryan P. Murelli, Emilio Gallicchio
المصدر: ACS Omega, Vol 1, Iss 3, Pp 435-447 (2016)
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2470-1343Test
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المؤلفون: Madhuri Dasari, Stephen C. Pelly, Jiafeng Geng, Hannah B. Gold, Nicole Pribut, Savita K. Sharma, Michael P. D’Erasmo, Perry W. Bartsch, Carrie Sun, Kiran Toti, Rebecca S. Arnold, John A. Petros, Lingjie Xu, Yi Jiang, Eric J. Miller, Dennis C. Liotta
المصدر: ACS Pharmacology & Translational Science. 6:702-709
مصطلحات موضوعية: Pharmacology, Pharmacology (medical)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::ae41ed73a3e6aa38dfae85c4e54699f4Test
https://doi.org/10.1021/acsptsci.2c00252Test -
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المؤلفون: Ryan P. Murelli, Michael P. D'Erasmo, Emilio Gallicchio, Baofeng Zhang
المصدر: ACS Omega, Vol 1, Iss 3, Pp 435-447 (2016)
ACS Omegaمصطلحات موضوعية: 0301 basic medicine, General Chemical Engineering, Human immunodeficiency virus (HIV), Nanotechnology, Computational biology, medicine.disease_cause, 01 natural sciences, Article, lcsh:Chemistry, 03 medical and health sciences, Molecular dynamics, 0103 physical sciences, medicine, RNase H, Conformational isomerism, Virtual screening, 010304 chemical physics, biology, Chemistry, Active site, General Chemistry, Reverse transcriptase, 3. Good health, 030104 developmental biology, lcsh:QD1-999, Docking (molecular), biology.protein
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f632338e9afba70c0e564f975a5b6169Test
https://doaj.org/article/82448fee59e944c19519aaaa5ff991e5Test -
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المؤلفون: Maria Korom, Tiffany C. Edwards, Michael P. D'Erasmo, John E. Tavis, Eileen A. Moran, Peter J. Ireland, Bindi S. Patel, Mark M. Cadiz, Lynda A. Morrison, Ankit K. Gupta, Danielle R. Hirsch, Ryan P. Murelli
المصدر: Antimicrobial Agents and Chemotherapy. 60:2140-2149
مصطلحات موضوعية: 0301 basic medicine, Herpesvirus 2, Human, viruses, Herpesvirus 1, Human, Biology, Virus Replication, medicine.disease_cause, Antiviral Agents, Tropolone, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, Chlorocebus aethiops, Drug Resistance, Viral, medicine, Animals, Humans, Structure–activity relationship, Cytotoxic T cell, Pharmacology (medical), Viral shedding, Cytotoxicity, Vero Cells, Pharmacology, Wild type, Virology, 030104 developmental biology, Infectious Diseases, Herpes simplex virus, Viral replication, Pharmacophore
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::70bb6a6576be600400474a7722ae1b28Test
https://doi.org/10.1128/aac.02675-15Test -
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المؤلفون: John A. Beutler, Takashi Masaoka, Baofeng Zhang, Rajat K. Pal, Michael P. D'Erasmo, Christine Meck, Jennifer A. Wilson, Danielle R. Hirsch, Stuart F.J. Le Grice, Emilio Gallicchio, Ryan P. Murelli
المصدر: MedChemComm. 7:1783-1788
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, chemistry.chemical_classification, Natural product, 030106 microbiology, Organic Chemistry, Human immunodeficiency virus (HIV), Pharmaceutical Science, Biology, medicine.disease_cause, Biochemistry, Molecular biology, Article, Reverse transcriptase, In vitro, 03 medical and health sciences, chemistry.chemical_compound, Enzyme, chemistry, Drug development, Drug Discovery, medicine, Molecular Medicine, Ribonuclease H activity
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5ea992066e20109c2362f02ab54c9f6eTest
https://doi.org/10.1039/c6md00238bTest -
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المؤلفون: John A. Beutler, Takashi Masaoka, Jennifer A. Wilson, Errol M. Hunte, Stuart F. J. Le Grice, Ryan P. Murelli, Michael P. D'Erasmo
المصدر: MedChemComm. 7:1789-1792
مصطلحات موضوعية: Drug, Stereochemistry, media_common.quotation_subject, Pharmaceutical Science, 010402 general chemistry, Cleavage (embryo), 01 natural sciences, Biochemistry, Article, Drug Discovery, Molecule, RNase H, media_common, Pharmacology, chemistry.chemical_classification, Aqueous solution, biology, 010405 organic chemistry, Drug discovery, Organic Chemistry, Combinatorial chemistry, Cycloaddition, 3. Good health, 0104 chemical sciences, Enzyme, chemistry, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::17b2b9865ea3ac3541d77efff5a5b33eTest
https://doi.org/10.1039/c6md00237dTest -
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المؤلفون: Ryan P. Murelli, Michael P. D'Erasmo
مصطلحات موضوعية: Molecular Structure, 010405 organic chemistry, Extramural, Organic Chemistry, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, Cycloaddition, Time efficient, Article, Tropolone, 0104 chemical sciences, chemistry.chemical_compound, Fluorides, chemistry, Yield (chemistry), Amide, Phase (matter), Molecule
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::00e5661e2a620ef457660b9df9f2bf06Test
https://europepmc.org/articles/PMC5859309Test/ -
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المؤلفون: Gerard D. Wright, Noushad Mohd, Michael P. D'Erasmo, Christine Meck, Danielle R. Hirsch, Georgina Cox, Tushar Shakya, Ryan P. Murelli
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:4943-4947
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Antibiotics, Pharmaceutical Science, medicine.disease_cause, 01 natural sciences, Biochemistry, Tropolone, Article, Microbiology, 03 medical and health sciences, Antibiotic resistance, Drug Resistance, Bacterial, Drug Discovery, Escherichia coli, medicine, Molecular Biology, chemistry.chemical_classification, 0303 health sciences, Molecular Structure, biology, 010405 organic chemistry, 030306 microbiology, Organic Chemistry, Aminoglycoside, biology.organism_classification, Nucleotidyltransferases, ANT, Anti-Bacterial Agents, 3. Good health, 0104 chemical sciences, Enzyme, Models, Chemical, chemistry, Molecular Medicine, Gentamicin, Gentamicins, Bacteria, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3c8ff965dad490bbf7b3ee2e92e07dd4Test
https://doi.org/10.1016/j.bmcl.2014.09.037Test -
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المؤلفون: Luis E. N. Quadri, Poornima Mohandas, Alberto Munoz, Jason J. Marineau, James E. Bradner, William B. Smith, Andrew S. Au, Michael P. D'Erasmo, Ryan P. Murelli
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:4035-4038
مصطلحات موضوعية: Stereochemistry, Mycobacterium smegmatis, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Antineoplastic Agents, Microbial Sensitivity Tests, Biochemistry, Article, Molecular conformation, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Escherichia coli, Humans, Structure–activity relationship, Spiro Compounds, Molecular Biology, Cell Proliferation, Dose-Response Relationship, Drug, Chemistry, Organic Chemistry, Diastereomer, Anti-Bacterial Agents, Molecular Medicine, Drug Screening Assays, Antitumor, Bacillus subtilis
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a3b85098f158d0ba5ca58064861ab17Test
https://doi.org/10.1016/j.bmcl.2014.05.102Test -
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المصدر: Med. Chem. Commun.. 5:842-852
مصطلحات موضوعية: Pharmacology, Resource (project management), Biological studies, High interest, Management science, Drug Discovery, Organic Chemistry, Pharmaceutical Science, Molecular Medicine, Treatment options, Biology, Biochemistry, Article
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::427caa84fea3740f0144f8dce81443a2Test
https://doi.org/10.1039/c4md00055bTest