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1دورية أكاديمية
المؤلفون: Carlo Matera, Michael Kauk, Davide Cirillo, Marco Maspero, Claudio Papotto, Daniela Volpato, Ulrike Holzgrabe, Marco De Amici, Carsten Hoffmann, Clelia Dallanoce
المصدر: Molecules, Vol 28, Iss 5, p 2407 (2023)
مصطلحات موضوعية: muscarinic acetylcholine receptors, Xanomeline, 77-LH-28-1, bitopic hybrid ligands, synthesis, fluorescence resonance energy transfer, Organic chemistry, QD241-441
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Daniela Volpato, Michael Kauk, Regina Messerer, Marcel Bermudez, Gerhard Wolber, Andreas Bock, Carsten Hoffmann, Ulrike Holzgrabe
المصدر: ACS Omega, Vol 5, Iss 49, Pp 31706-31715 (2020)
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2470-1343Test
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المؤلفون: Christine S. Heinz, Marcel Bermudez, Natasha Jaiswal, Carolin Große, Michael Kauk, Carsten Hoffmann, Ulrike Holzgrabe
المصدر: Journal of Natural Products. 86:869-881
مصطلحات موضوعية: Pharmacology, Complementary and alternative medicine, Organic Chemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Analytical Chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::32f71a33ed39284cdbd1953238a63b20Test
https://doi.org/10.1021/acs.jnatprod.2c01079Test -
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المؤلفون: Matthias Irmen, Janine Holze, Michael Kauk, Marcel Bermudez, Marco De Amici, Clelia Dallanoce, Klaus Mohr, Theresa Bödefeld, Gabriele M. König, Andreas Bock, Eva Marie Pfeil, Carsten Hoffmann, Gerhard Wolber, Carlo Matera, Ulrike Holzgrabe, Evi Kostenis, Ramona Schrage, Christian Tränkle
المصدر: ACS Pharmacol Transl Sci
مصطلحات موضوعية: Pharmacology, Coupling (electronics), Chemistry, Allosteric regulation, Biophysics, Extracellular, Pharmacology (medical), Muscarinic acetylcholine receptor M1, Receptor, Intracellular, G Protein-Coupled Receptor Signaling, G protein-coupled receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::71b5f203c7b3b178ef34fa4414d35cbaTest
https://doi.org/10.1021/acsptsci.0c00069Test -
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المؤلفون: Monika Kustermann, Svenja Laue, Yinghong Cui, Douglas G. Tilley, Laurel A. Grisanti, Melanie Rothe, Michael Kauk, Carsten Hoffmann, Melanie Philipp, WH Zimmermann, Teresa Casar Tena, Allessandra Moretti, Farah Raad, Michael Kühl, Martina S. Burczyk, Sabrina Matysik, Martin D. Burkhalter, Cornelia Donow, Jürgen Wess
المصدر: JCI Insight
مصطلحات موضوعية: 0301 basic medicine, Embryo, Nonmammalian, Tolterodine Tartrate, Organogenesis, Muscarinic Antagonists, Mice, Xenopus laevis, 03 medical and health sciences, 0302 clinical medicine, Heart Conduction System, Muscarinic acetylcholine receptor, Heart rate, medicine, Animals, Humans, Myocytes, Cardiac, Receptor, Zebrafish, Mice, Knockout, Receptor, Muscarinic M3, Sinoatrial node, business.industry, fungi, Muscarinic acetylcholine receptor M3, Arrhythmias, Cardiac, General Medicine, Embryo, Mammalian, medicine.disease, 3. Good health, Disease Models, Animal, HEK293 Cells, 030104 developmental biology, medicine.anatomical_structure, 030220 oncology & carcinogenesis, Heart failure, Atrioventricular canal, Electrical conduction system of the heart, business, Neuroscience, Research Article
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2d95a3d11c2efe67a92a1fc8c1ec423aTest
https://doi.org/10.1172/jci.insight.121971Test -
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المؤلفون: Michael Kauk, Sven Höfling, Monika Emmerling, Martin Kamp, Katrin G. Heinze, Hannah S. Heil, Benjamin Schreiber, Carsten Hoffmann, Ingrid Tessmer, Ulrike Holzgrabe
المصدر: ACS Photonics. 5:2225-2233
مصطلحات موضوعية: 0301 basic medicine, Chemistry, Energy transfer, 02 engineering and technology, 021001 nanoscience & nanotechnology, Atomic and Molecular Physics, and Optics, Fluorescence spectroscopy, Electronic, Optical and Magnetic Materials, 03 medical and health sciences, 030104 developmental biology, Membrane, Förster resonance energy transfer, Microscopy, Biophysics, Electrical and Electronic Engineering, 0210 nano-technology, Receptor, Membrane biophysics, Biotechnology, G protein-coupled receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::c23fea38af4bbdcd85724055202f8ee0Test
https://doi.org/10.1021/acsphotonics.8b00072Test -
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المؤلفون: Regina Messerer, Luca Agnetta, Carsten Hoffmann, Ulrike Holzgrabe, Maria Consuelo Alonso Canizal, Michael Decker, Michael Kauk
المصدر: Angewandte Chemie. 129:7388-7393
مصطلحات موضوعية: 0301 basic medicine, 03 medical and health sciences, 030104 developmental biology, General Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::19f194052521672abd354863ac22c57eTest
https://doi.org/10.1002/ange.201701524Test -
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المؤلفون: Ulrike Zabel, Carsten Hoffmann, Jessika Klöckner, Susanne Nuber, Michael Kauk, Regina Messerer, Maria Consuelo Alonso Canizal, Daniela Volpato, Ulrike Holzgrabe
المصدر: ACS Chemical Biology. 12:833-843
مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Allosteric modulator, Stereochemistry, Carboxylic acid, Allosteric regulation, General Medicine, Muscarinic acetylcholine receptor M1, Biochemistry, 03 medical and health sciences, 030104 developmental biology, Förster resonance energy transfer, chemistry, Muscarinic acetylcholine receptor, medicine, Molecular Medicine, Pharmacophore, Acetylcholine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::d4d2fb6fd669960d0cf18f1b3cbbc4a2Test
https://doi.org/10.1021/acschembio.6b00828Test -
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المؤلفون: Michael Kauk, Carsten Hoffmann
المصدر: Trends in pharmacological sciences. 39(2)
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Chemistry, Protein Conformation, Energy transfer, Intermolecular force, Molecular Dynamics Simulation, Toxicology, Single Molecule Imaging, Receptors, G-Protein-Coupled, 03 medical and health sciences, 030104 developmental biology, Protein structure, Förster resonance energy transfer, Structural biology, Intramolecular force, Biophysics, Fluorescence Resonance Energy Transfer, Animals, Humans, G protein-coupled receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4b79208bf4ee88565d3f9df6d930d766Test
https://pubmed.ncbi.nlm.nih.gov/29180026Test -
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المؤلفون: Michael Decker, Michael Kauk, Luca Agnetta, Maria Consuelo Alonso Canizal, Ulrike Holzgrabe, Carsten Hoffmann, Regina Messerer
المصدر: Angewandte Chemie (International ed. in English). 56(25)
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Photochemistry, Allosteric regulation, 010402 general chemistry, Ligands, 01 natural sciences, Catalysis, Receptors, G-Protein-Coupled, 03 medical and health sciences, Muscarinic acetylcholine receptor, Fluorescence Resonance Energy Transfer, Humans, Binding site, Receptor, G protein-coupled receptor, Neurotransmitter Agents, Binding Sites, Chemistry, General Chemistry, Muscarinic acetylcholine receptor M1, Ligand (biochemistry), Receptors, Muscarinic, 0104 chemical sciences, 030104 developmental biology, Förster resonance energy transfer, Biophysics
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::222c47c73ee2f19333b0df1150eb2930Test
https://pubmed.ncbi.nlm.nih.gov/28510314Test