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المؤلفون: Paul Kirschmeier, Daniel J. Hicklin, M. Arshad Siddiqui, Payal R. Sheth, Huadong Tang, Elizabeth Smith, Bohdan Yaremko, Abdul Ponery, Lianzhu Liang, Suining Lee, Seema Tevar, Lissette Nale, Kimberly Gray, Chaoyang Dai, Ming Liu, Andrea D. Basso
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::323e1342aa3b907de9717e370e74f9efTest
https://doi.org/10.1158/1535-7163.22484694.v1Test -
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المؤلفون: Paul Kirschmeier, Daniel J. Hicklin, M. Arshad Siddiqui, Payal R. Sheth, Huadong Tang, Elizabeth Smith, Bohdan Yaremko, Abdul Ponery, Lianzhu Liang, Suining Lee, Seema Tevar, Lissette Nale, Kimberly Gray, Chaoyang Dai, Ming Liu, Andrea D. Basso
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6041f2cd41a43e8a9ab2086483f35521Test
https://doi.org/10.1158/1535-7163.c.6531537Test -
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المؤلفون: Guowei Zhou, Liping Yang, Neng-Yang Shih, M. Arshad Siddiqui, Vinay Girijavallabhan, Shiying Chen, Lei Chen, Dansu Li, Peter Orth, Zhuyan Guo, Bandarpalle B. Shankar, Kristin E. Rosner, Wensheng Yu, Ling Tong, Chaoyang Dai, Joseph A. Kozlowski, Aneta Kosinski, Xiaoda Niu, Seong Heon Kim, Daniel Lundell, Shelby Umland, Janeta Popovici-Muller
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:3037-3042
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Hydantoin, ADAM17 Protein, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Dogs, 0302 clinical medicine, Drug Discovery, Animals, Humans, Potency, Protease Inhibitors, Molecular Biology, Whole blood, chemistry.chemical_classification, Chemistry, Hydantoins, Organic Chemistry, Haplorhini, Rats, Enzyme Activation, 030104 developmental biology, Enzyme, ROC Curve, Area Under Curve, Molecular Medicine, Tumor necrosis factor alpha, Half-Life, 030215 immunology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5e9ae78bb60384e5c554a062fa84b16eTest
https://doi.org/10.1016/j.bmcl.2017.05.062Test -
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المصدر: Tetrahedron Letters. 54:6373-6377
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Drug Discovery, Biochemistry, Medicinal chemistry, Enol
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::0720e553ad1530d87c8d73deca76c78dTest
https://doi.org/10.1016/j.tetlet.2013.09.059Test -
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المؤلفون: Jeffrey P. Ciavarri, Thierry O. Fischmann, M. Arshad Siddiqui, Lianyun Zhao, Xingmin Zhang, Zhaoyang Meng, Panduranga Adulla P. Reddy, Charles E. Whitehurst, Andrew Mcriner, Yinyan Zhao
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2863-2867
مصطلحات موضوعية: Models, Molecular, Cell cycle checkpoint, Pyrimidine, Pyrazine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Protein Serine-Threonine Kinases, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Potency, Protein Kinase Inhibitors, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Organic Chemistry, Imidazoles, Intracellular Signaling Peptides and Proteins, Pyrimidines, chemistry, Pyrazines, Checkpoint Kinase 1, Molecular Medicine, biological phenomena, cell phenomena, and immunity, Protein Kinases
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3184c0b06ac4673d0478ae586fd6cc5aTest
https://doi.org/10.1016/j.bmcl.2013.03.100Test -
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المؤلفون: Cliff C. Cheng, Jose S. Duca, Wolfgang Seghezzi, Thierry O. Fischmann, David A. Parry, M. Arshad Siddiqui, Matthew Richards, Lianyun Zhao, Panduranga Adulla P. Reddy, Praveen K. Tadikonda, Xiaohua Huang, Nicole Davis, Gerald W. Shipps, Derek Wiswell
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2590-2594
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, Drug Discovery, medicine, Molecule, Protein Kinase Inhibitors, Molecular Biology, Topology (chemistry), Binding Sites, Chemistry, Cyclin-Dependent Kinase 2, Organic Chemistry, 2-aminothiazole, Amides, Molecular Docking Simulation, Thiazoles, Drug Design, Checkpoint Kinase 1, Molecular Medicine, Structure based, Surface protein, Selectivity, Protein Kinases, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f4dd9958354f4a0c663d0f92411fbb3aTest
https://doi.org/10.1016/j.bmcl.2013.02.108Test -
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المؤلفون: Mike Fleming, David B. Belanger, Kimberly Gray, Matthew P. Rainka, Andrea D. Basso, M. Arshad Siddiqui, Matthew Ernst Voss, Johannes H. Voigt, Alan Hruza, Lisa H. Peterson
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:3544-3549
مصطلحات موضوعية: Models, Molecular, Pyrazine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Protein Serine-Threonine Kinases, Pyrazole, Crystallography, X-Ray, Biochemistry, Cell activity, Structure-Activity Relationship, chemistry.chemical_compound, Acetic acid, Aurora kinase, Aurora Kinases, Drug Discovery, Protein Kinase Inhibitors, Molecular Biology, Kinase, Organic Chemistry, Imidazoles, Enzyme inhibition, chemistry, Pyrazines, Molecular Medicine, Selectivity
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8de034d96517afc96aac15977909ba4eTest
https://doi.org/10.1016/j.bmcl.2012.03.051Test -
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المؤلفون: Yan Wang, Patrick J. Curran, Jack B. Bracken, Gerald W. Shipps, M. Arshad Siddiqui, Hua Miao, David B. Belanger, Hongbo Zeng, Michael Malkowski
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5870-5875
مصطلحات موضوعية: Clinical Biochemistry, High selectivity, Dasatinib, Pharmaceutical Science, Breast Neoplasms, Protein Serine-Threonine Kinases, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Aurora Kinases, Proto-Oncogenes, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Computer Simulation, Molecular Targeted Therapy, Protein Kinase Inhibitors, Molecular Biology, Adaptor Proteins, Signal Transducing, Dose-Response Relationship, Drug, Chemistry, Kinase, Drug discovery, Organic Chemistry, Imidazoles, RNA-Binding Proteins, Signal transducing adaptor protein, Oncogenes, Protein-Tyrosine Kinases, Neoplasm Proteins, DNA-Binding Proteins, Thiazoles, Phenotype, Pyrimidines, Drug Design, Pyrazines, Melanocytes, Molecular Medicine, Female, PTK6, Drug Screening Assays, Antitumor, Tyrosine kinase, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c602c45bbeb7b8ec30580b6a5d7bc119Test
https://doi.org/10.1016/j.bmcl.2011.07.101Test -
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المؤلفون: Peter Orth, Bandarpalle B. Shankar, Daniel Lundell, Corey O. Strickland, Vinay Girijavallabhan, Chaoyang Dai, Joseph A. Kozlowski, Janeta Popovici-Muller, Brian J. Lavey, Jing Sun, Shiying Chen, Dansu Li, John J. Piwinski, Razia Rizvi, M. Arshad Siddiqui, Kristin E. Rosner, Lianyun Zhao, Zhuyan Guo, Wong Michael K C, Neng-Yang Shih, Xiaoda Niu
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3172-3176
مصطلحات موضوعية: Pyrrolidines, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Carboxamide, ADAM17 Protein, Tartrate, Biochemistry, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Oral administration, Amide, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Tartrates, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Organic Chemistry, Amides, Rats, Enzyme Activation, ADAM Proteins, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b5ffe3fdf02a5dba0580b311b55f7fe2Test
https://doi.org/10.1016/j.bmcl.2011.01.002Test -
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المؤلفون: Todd A. Black, U. Faruk Mansoor, Dilrukshi Vitharana, Dayna L. Daubaras, Paul M. McNicholas, Peter Orth, Panduranga Adulla P. Reddy, M. Arshad Siddiqui
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:1155-1161
مصطلحات موضوعية: Gram-negative bacteria, Clinical Biochemistry, Pharmaceutical Science, Microbial Sensitivity Tests, Crystallography, X-Ray, Hydroxamic Acids, Biochemistry, Catalysis, Amidohydrolases, Lipid A, Structure-Activity Relationship, chemistry.chemical_compound, Catalytic Domain, Gram-Negative Bacteria, Drug Discovery, Structure–activity relationship, Molecular Biology, Antibacterial agent, Benzodiazepinones, Binding Sites, Hydroxamic acid, biology, Chemistry, Organic Chemistry, biology.organism_classification, Anti-Bacterial Agents, Zinc, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Antibacterial activity, Bacterial outer membrane
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4e24e1aa00734c6354523e16694b6690Test
https://doi.org/10.1016/j.bmcl.2010.12.111Test