-
1
المؤلفون: Martin L. Stockley, Amanda Ferdinand, Giovanni Benedetti, Peter Blencowe, Susan M. Boyd, Mat Calder, Mark D. Charles, Lucy V. Edwardes, Tennyson Ekwuru, Harry Finch, Alessandro Galbiati, Lerin Geo, Diego Grande, Vera Grinkevich, Nicholas D. Holliday, Wojciech W. Krajewski, Ellen MacDonald, Jayesh B. Majithiya, Hollie McCarron, Claire L. McWhirter, Viral Patel, Chris Pedder, Eeson Rajendra, Marco Ranzani, Laurent J. M. Rigoreau, Helen M. R. Robinson, Theresia Schaedler, Julija Sirina, Graeme C. M. Smith, Martin E. Swarbrick, Andrew P. Turnbull, Simon Willis, Robert A. Heald
المصدر: Journal of Medicinal Chemistry. 65:13879-13891
مصطلحات موضوعية: DNA End-Joining Repair, Drug Discovery, Humans, Molecular Medicine, DNA, Poly(ADP-ribose) Polymerase Inhibitors, Ligands
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a3234589eaa7f5350d23a2af196b12eTest
https://doi.org/10.1021/acs.jmedchem.2c01142Test -
2
المؤلفون: Lucy V. Edwardes, Sarah J. Caswell, Mariacarmela Giurrandino, Xiang Zhai, Andrea Gohlke, Demetrios H. Kostomiris, Hannah K. Pollard, Alexander Pflug, Gregory R. Hamm, Kate V. Jervis, Paul N. Clarkson, Karl Syson
المصدر: Biochemistry. 61:1974-1987
مصطلحات موضوعية: Histones, Kinetics, Lysine, Intracellular Signaling Peptides and Proteins, Humans, Histone-Lysine N-Methyltransferase, Methylation, Biochemistry, Myeloid-Lymphoid Leukemia Protein
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4381a5f29cee7d23fa10c29cca9377deTest
https://doi.org/10.1021/acs.biochem.2c00385Test -
3
المؤلفون: Alice R Eddershaw, Karl Syson, Paul R. J. Davey, Gregory Hamm, Christopher D. Stubbs, Paul Clarkson, Elizabeth Underwood, Lucy V Edwardes
المصدر: Biochemistry. 59:4775-4786
مصطلحات موضوعية: Models, Molecular, Protein-Arginine N-Methyltransferases, Methyltransferase, Arginine, In Vitro Techniques, Biochemistry, Mass Spectrometry, Substrate Specificity, 03 medical and health sciences, Protein structure, Catalytic Domain, Humans, Protein Interaction Domains and Motifs, Amino Acid Sequence, Enzyme Inhibitors, Protein Structure, Quaternary, Ternary complex, Adaptor Proteins, Signal Transducing, 0303 health sciences, Chemistry, Protein arginine methyltransferase 5, 030302 biochemistry & molecular biology, Deuterium Exchange Measurement, Recombinant Proteins, Kinetics, Biophysics, Hydrogen–deuterium exchange, Steady state (chemistry)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e0c63875119c271f482688a035fe6bfcTest
https://doi.org/10.1021/acs.biochem.0c00554Test