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1
المؤلفون: Frederic J. de Sauvage, Robert L. Yauch, Stephen E. Gould, Suzie J. Scales, Dan Sutherlin, Kirk Robarge, Richard Goldsmith, Dan Burdick, Zora Modrusan, Kristina West, Thomas Januario, Lasse Weinmann, Bruno Alicke, Gerrit J. P. Dijkgraaf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bd80db1f9d1b999661f6a494b03c5e21Test
https://doi.org/10.1158/0008-5472.c.6502772Test -
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المؤلفون: Frederic J. de Sauvage, Robert L. Yauch, Stephen E. Gould, Suzie J. Scales, Dan Sutherlin, Kirk Robarge, Richard Goldsmith, Dan Burdick, Zora Modrusan, Kristina West, Thomas Januario, Lasse Weinmann, Bruno Alicke, Gerrit J. P. Dijkgraaf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::756df7575425785d5cd447ebe4a28bd7Test
https://doi.org/10.1158/0008-5472.22389962Test -
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المؤلفون: Frederic J. de Sauvage, Robert L. Yauch, Stephen E. Gould, Suzie J. Scales, Dan Sutherlin, Kirk Robarge, Richard Goldsmith, Dan Burdick, Zora Modrusan, Kristina West, Thomas Januario, Lasse Weinmann, Bruno Alicke, Gerrit J. P. Dijkgraaf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b05f5d20f7e4dd28d59546d16be17fefTest
https://doi.org/10.1158/0008-5472.22389968.v1Test -
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المؤلفون: Frederic J. de Sauvage, Robert L. Yauch, Stephen E. Gould, Suzie J. Scales, Dan Sutherlin, Kirk Robarge, Richard Goldsmith, Dan Burdick, Zora Modrusan, Kristina West, Thomas Januario, Lasse Weinmann, Bruno Alicke, Gerrit J. P. Dijkgraaf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::088e879ff92888701d72858a98dc149dTest
https://doi.org/10.1158/0008-5472.22389965Test -
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المؤلفون: BinQing Wei, Kirk Robarge, Sharada S. Labadie, Jinhua Chen, Laura B. Corson, Antonio DiPasquale, Peter S. Dragovich, Charles Eigenbrot, Marie Evangelista, Benjamin P. Fauber, Anna Hitz, Rebecca Hong, Kwong Wah Lai, Wenfeng Liu, Shuguang Ma, Shiva Malek, Thomas O'Brien, Jodie Pang, David Peterson, Laurent Salphati, Deepak Sampath, Steven Sideris, Mark Ultsch, Zijin Xu, Ivana Yen, Dong Yu, Qin Yue, Aihe Zhou, Hans E. Purkey
المصدر: Bioorganicmedicinal chemistry letters. 59
مصطلحات موضوعية: Dose-Response Relationship, Drug, L-Lactate Dehydrogenase, Lactams, Molecular Structure, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Cell Line, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, Microsomes, Liver, Molecular Medicine, Animals, Humans, Enzyme Inhibitors, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0770db4a66cefb70bb9bee4bcf37ca52Test
https://pubmed.ncbi.nlm.nih.gov/35065235Test -
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المؤلفون: Charles Z. Ding, Laurent Salphati, Hans E. Purkey, HongXiu Ge, Qin Yue, Antonio G. DiPasquale, Charles Eigenbrot, Qunh Ho, Kwong Wah Lai, Thomas O'Brien, Sharada Labadie, Zhongguo Chen, David A. Peterson, Shiva Malek, Laura Corson, Wenfeng Liu, Mark Ultsch, Jinhua Chen, Anna Hitz, Yajing Liu, Kirk Robarge, Jodie Pang, Chiho Li, Peter S. Dragovich, Binqing Wei, Shuguang Ma, Huihui Zhang, Steve Sideris, Zhenting Gao, Marie Evangelista, Ivana Yen, Aihe Zhou, Benjamin Fauber
المصدر: ACS Medicinal Chemistry Letters. 7:896-901
مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Organic Chemistry, Cell, Biology, Pharmacology, Biochemistry, Bioavailability, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, medicine.anatomical_structure, Enzyme, chemistry, Cell culture, 030220 oncology & carcinogenesis, Lactate dehydrogenase, Drug Discovery, medicine, Glycolysis, IC50
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5f0532bd0e9287d033f18781fd7cf755Test
https://doi.org/10.1021/acsmedchemlett.6b00190Test -
7
المؤلفون: Gary Salmon, Harvey Wong, Maxine Norman, Adrian Barnard, Aihe Zhou, Julie Hawkins, Benjamin Fauber, Adam R. Johnson, Arunima Ganguli, Yuzhong Deng, Susan Summerhill, Kirk Robarge, Celine Eidenschenk, Wenjun Ouyang, Christine Everett, Jianhua Cao, Wei Tang, Hank La, Alberto Gobbi
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:2907-2912
مصطلحات موضوعية: Pyrimidine, Pyridines, medicine.medical_treatment, Clinical Biochemistry, Retinoic acid, Chemical biology, Pharmaceutical Science, Biochemistry, Autoimmune Diseases, Cell Line, Structure-Activity Relationship, chemistry.chemical_compound, RAR-related orphan receptor gamma, Drug Discovery, medicine, Animals, Humans, Inverse agonist, Molecular Biology, Cells, Cultured, Orphan receptor, Interleukin-17, Organic Chemistry, Imidazoles, Nuclear Receptor Subfamily 1, Group F, Member 3, Rats, HEK293 Cells, Pyrimidines, Cytokine, Liver, chemistry, Nuclear receptor, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa9c3898f9ddd336ebaff802da33874cTest
https://doi.org/10.1016/j.bmcl.2015.05.055Test -
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المؤلفون: Binqing Wei, Erica VanderPorten, Mark Ultsch, Jason Boggs, Peter S. Dragovich, S. Sideris, Jinhua Chen, Huihui Zhang, Sharada Labadie, Qin Yue, Charles Z. Ding, Kirk Robarge, David Peterson, Shuguang Ma, Hans E. Purkey, Benjamin Fauber, HongXiu Ge, Aihe Zhou, Kwong Wah Lai, Qunh Ho, Shiva Malek, Xuying Zhang, Ivana Yen, Laura Corson, Charles Eigenbrot, Qing Xu, Laurent Salphati
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:75-82
مصطلحات موضوعية: Gene isoform, Stereochemistry, Lactate dehydrogenase A, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Madin Darby Canine Kidney Cells, chemistry.chemical_compound, Dogs, Oxidoreductase, Lactate dehydrogenase, Drug Discovery, Animals, Humans, Potency, Glycolysis, Enzyme Inhibitors, education, Molecular Biology, chemistry.chemical_classification, education.field_of_study, L-Lactate Dehydrogenase, Organic Chemistry, Madin Darby canine kidney cell, chemistry, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::921f2e384863aba9482741802d507295Test
https://doi.org/10.1016/j.bmcl.2014.11.008Test -
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المؤلفون: Philip Stephen Jackson, Pascal Savy, Jodie Pang, Wendy Lee, April Yang, Mark Ultsch, Robert Heald, Jason Boggs, Edna F. Choo, Charles Eigenbrot, Xioaye Yang, Kirk Robarge, Matthew Baumgardner, Joanne Hewitt, Steve Price, Brenda Burton, Christian Wiesmann
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:4714-4723
مصطلحات موضوعية: Models, Molecular, Pyrazine, Stereochemistry, Clinical Biochemistry, Diol, Pharmaceutical Science, Mitogen-activated protein kinase kinase, Ring (chemistry), Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Heterocyclic Compounds, Cell Line, Tumor, Drug Discovery, Pyridine, Humans, Structure–activity relationship, Protein Kinase Inhibitors, Molecular Biology, Cell Proliferation, Mitogen-Activated Protein Kinase Kinases, Dose-Response Relationship, Drug, Molecular Structure, Drug discovery, Organic Chemistry, Imidazoles, HCT116 Cells, chemistry, Ras Signaling Pathway, Pyrazines, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5a1ebaa13120fa34ee18794315152d4dTest
https://doi.org/10.1016/j.bmcl.2014.08.008Test -
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المؤلفون: Peter S. Dragovich, Benjamin P. Fauber, Jason Boggs, Jinhua Chen, Laura B. Corson, Charles Z. Ding, Charles Eigenbrot, HongXiu Ge, Anthony M. Giannetti, Thomas Hunsaker, Sharada Labadie, Chiho Li, Yichin Liu, Yingchun Liu, Shuguang Ma, Shiva Malek, David Peterson, Keith E. Pitts, Hans E. Purkey, Kirk Robarge, Laurent Salphati, Steve Sideris, Mark Ultsch, Erica VanderPorten, Jing Wang, BinQing Wei, Qing Xu, Ivana Yen, Qin Yue, Huihui Zhang, Xuying Zhang, Aihe Zhou
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:3764-3771
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, Oral administration, Lactate dehydrogenase, Drug Discovery, Animals, Humans, Glycolysis, Sulfhydryl Compounds, Enzyme Inhibitors, Surface plasmon resonance, Molecular Biology, Dose-Response Relationship, Drug, L-Lactate Dehydrogenase, Molecular Structure, Cyclohexanones, Chemistry, Organic Chemistry, High-Throughput Screening Assays, Rats, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4ed0191d5c5ad01b10f95a841198637Test
https://doi.org/10.1016/j.bmcl.2014.06.076Test