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1دورية أكاديمية
المؤلفون: Pirow Bekker, Karen Ebsworth, Matthew J. Walters, Robert D. Berahovich, Linda S. Ertl, Trevor T. Charvat, Sreenivas Punna, Jay P. Powers, James J. Campbell, Timothy J. Sullivan, Juan C. Jaen, Thomas J. Schall
المصدر: Mediators of Inflammation, Vol 2015 (2015)
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Guillaume Mata (1685596), Dillon H. Miles (8962160), Samuel L. Drew (8682102), Jeremy Fournier (3594275), Kenneth V. Lawson (2391673), Artur K. Mailyan (1588903), Ehesan U. Sharif (6847676), Xuelei Yan (1698157), Joel W. Beatty (1328199), Jesus Banuelos (4036886), Jie Chen (5892), Elaine Ginn (2124058), Ada Chen (1698127), Kimberline Y. Gerrick (6061382), Amber T. Pham (8682105), Kent Wong (2160739), Divyank Soni (9383865), Puja Dhanota (6506090), Stefan G. Shaqfeh (9383868), Cesar Meleza (6899225), Nell Narasappa (11592941), Hema Singh (11592944), Xiaoning Zhao (184301), Lixia Jin (1570120), Ulrike Schindler (9383871), Matthew J. Walters (296691), Stephen W. Young (7022015), Nigel P. Walker (8682108), Manmohan Reddy Leleti (8682111), Jay P. Powers (1721107), Jenna L. Jeffrey (2029015)
مصطلحات موضوعية: Biochemistry, Medicine, Pharmacology, Immunology, Developmental Biology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, early lead series, tumor immune microenvironment, significant immune response, molecular docking studies, selective pi3kγ inhibitors, pyrazolopyrimidine amide inhibitors, 56 b, immune cells, vitro <, studies indicate, pyrazolopyrimidine isoindolinones, optimal amide, metabolic stability, m1 macrophages, like properties, kinase γ, isoindolinone substituents, inflammatory phenotype, inflammatory mediators, increasing pro, highly potent, highly expressed, favorable drug
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المؤلفون: Matthew J. Walters, Kelsey E. Sivick, Uli Schindler, Jay P. Powers, Stephen W. Young, Jaroslaw Kalisiak, Nikki Kimura, Timothy W. Park, Bhamini Purandare, Susan L. Paprcka, Fangfang Yin, Akshata R. Udyavar, Elaine Ginn, Ada Chen, Kristen Zhang, Daniel DiRenzo, Nell Narasappa, Jesus Banuelos, Annette Becker, Joanne B.L. Tan, Dana Piovesan
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4eb5b5a4e6987b75f7ac46778faa4a20Test
https://doi.org/10.1158/1535-7163.22522347Test -
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المؤلفون: Matthew J. Walters, Kelsey E. Sivick, Uli Schindler, Jay P. Powers, Stephen W. Young, Jaroslaw Kalisiak, Nikki Kimura, Timothy W. Park, Bhamini Purandare, Susan L. Paprcka, Fangfang Yin, Akshata R. Udyavar, Elaine Ginn, Ada Chen, Kristen Zhang, Daniel DiRenzo, Nell Narasappa, Jesus Banuelos, Annette Becker, Joanne B.L. Tan, Dana Piovesan
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::35adf1efc1bd618059ec8b92f7b406e6Test
https://doi.org/10.1158/1535-7163.22522341Test -
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المؤلفون: Matthew J. Walters, Kelsey E. Sivick, Uli Schindler, Jay P. Powers, Stephen W. Young, Jaroslaw Kalisiak, Nikki Kimura, Timothy W. Park, Bhamini Purandare, Susan L. Paprcka, Fangfang Yin, Akshata R. Udyavar, Elaine Ginn, Ada Chen, Kristen Zhang, Daniel DiRenzo, Nell Narasappa, Jesus Banuelos, Annette Becker, Joanne B.L. Tan, Dana Piovesan
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9db083be516cf4170981d0503a34a58bTest
https://doi.org/10.1158/1535-7163.c.6543339.v1Test -
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المؤلفون: Dana Piovesan, Joanne B.L. Tan, Annette Becker, Jesus Banuelos, Nell Narasappa, Daniel DiRenzo, Kristen Zhang, Ada Chen, Elaine Ginn, Akshata R. Udyavar, Fangfang Yin, Susan L. Paprcka, Bhamini Purandare, Timothy W. Park, Nikki Kimura, Jaroslaw Kalisiak, Stephen W. Young, Jay P. Powers, Uli Schindler, Kelsey E. Sivick, Matthew J. Walters
المصدر: Molecular Cancer Therapeutics. 21:948-959
مصطلحات موضوعية: Mice, Cancer Research, Adenosine, Oncology, Programmed Cell Death 1 Receptor, Tumor Microenvironment, Animals, Humans, Immune Checkpoint Inhibitors, Melanoma
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fada8c684c9b4eda6511188f28c46437Test
https://doi.org/10.1158/1535-7163.mct-21-0802Test -
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المؤلفون: Dillon H. Miles, Ada Chen, Manmohan Reddy Leleti, Divyank Soni, Stephen W Young, Artur K. Mailyan, Kenneth V. Lawson, Stefan G Shaqfeh, Ehesan U. Sharif, Jenna L. Jeffrey, Jesus Banuelos, Xuelei Yan, Samuel L Drew, Kimberline Gerrick, Nigel Walker, Puja Dhanota, Lixia Jin, Jay P. Powers, Elaine Ginn, Guillaume Mata, Kent Wong, Hema Singh, Jeremy Fournier, Joel W. Beatty, Ulrike Schindler, Amber Pham, Matthew J. Walters, Jie Chen, Cesar Meleza, Xiaoning Zhao, Nell Narasappa
المصدر: Journal of Medicinal Chemistry. 65:1418-1444
مصطلحات موضوعية: Male, Pyrazolopyrimidine, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Immune system, Amide, Drug Discovery, Animals, Class Ib Phosphatidylinositol 3-Kinase, Humans, Structure–activity relationship, Potency, Phosphoinositide-3 Kinase Inhibitors, Phosphoinositide 3-kinase, biology, Amides, Phenotype, In vitro, Rats, Molecular Docking Simulation, Pyrimidines, chemistry, Biochemistry, Drug Design, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b37aec4464f4375ff8b99d31a40b9e89Test
https://doi.org/10.1021/acs.jmedchem.1c01153Test -
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المؤلفون: Dillon H. Miles, Nigel Walker, Manmohan Reddy Leleti, Xiaoning Zhao, Eric T. Newcomb, Kenneth V. Lawson, Jaroslaw Kalisiak, Erick Allen Lindsey, Lixia Jin, Ada Chen, Laurent Debien, Guifen Xu, Ehesan U. Sharif, Norbert Sträter, Brandon Reid Rosen, Stephen W Young, Emma Scaletti, Jay P. Powers
المصدر: Journal of Medicinal Chemistry. 64:845-860
مصطلحات موضوعية: Adenosine, Phosphorous Acids, Drug Evaluation, Preclinical, Molecular Dynamics Simulation, Crystallography, X-Ray, GPI-Linked Proteins, 01 natural sciences, Structure-Activity Relationship, 03 medical and health sciences, Immune system, ATP hydrolysis, Drug Discovery, medicine, Extracellular, Humans, Ectonucleotidase, 5'-Nucleotidase, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, Tumor microenvironment, Binding Sites, Adenosine receptor, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Enzyme, chemistry, Biochemistry, Drug Design, Molecular Medicine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0d84eb5999417f66c4c65efddd2d03a7Test
https://doi.org/10.1021/acs.jmedchem.0c01835Test -
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المؤلفون: Manmohan Reddy Leleti, Jeremy Fournier, Steven D. Jacob, Eric F. Connor, Grange Rebecca Louise, Kenneth V. Lawson, Anh Tran, Jaroslaw Kalisiak, Jay P. Powers, Xuelei Yan
المصدر: Organic Process Research & Development. 25:157-162
مصطلحات موضوعية: Computer science, Pancreatic cancer, Organic Chemistry, Core (graph theory), medicine, Computational biology, Physical and Theoretical Chemistry, medicine.disease, Small molecule
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::d580f50a6db851b07be5e001c64ef367Test
https://doi.org/10.1021/acs.oprd.0c00469Test -
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المؤلفون: Dillon H. Miles, Ada Chen, Manmohan Reddy Leleti, Divyank Soni, Stephen W Young, Artur K. Mailyan, Kenneth V. Lawson, Stefan G Shaqfeh, Ehesan U. Sharif, Pei-Yu Chen, Jenna L. Jeffrey, Jesus Banuelos, Xuelei Yan, Samuel L Drew, Nigel Walker, Puja Dhanota, Lixia Jin, Jay P. Powers, Elaine Ginn, Guillaume Mata, Kent Wong, Jeremy Fournier, Joel W. Beatty, Rhiannon Thomas-Tran, Ulrike Schindler, Amber Pham, Matthew J. Walters, Jie Chen, Cesar Meleza, Xiaoning Zhao
المصدر: Journal of Medicinal Chemistry. 63:11235-11257
مصطلحات موضوعية: Gene isoform, Stereochemistry, Crystallography, X-Ray, 01 natural sciences, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, Animals, Class Ib Phosphatidylinositol 3-Kinase, Humans, Binding site, Phosphoinositide-3 Kinase Inhibitors, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, Trifluoromethyl, Bicyclic molecule, Lipid signaling, Rats, 0104 chemical sciences, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Enzyme, chemistry, Drug Design, Molecular Medicine, Selectivity, Adenosine triphosphate
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::237c477c3969b94ce636dfc76aca3e4fTest
https://doi.org/10.1021/acs.jmedchem.0c01203Test