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1دورية أكاديمية
المؤلفون: Zhengyu Yuan, Dinesh V. Patel, Beat Weidmann, Richard J. White, Shi-hao Pan, Wilma L. Porter, Jeff Jacobs, Joaquim Trias, George Withers Iii, Helen Gu, Elina Dunn, R. Kulathila, Margolis Wen Wang Jim Koehn, James B. Mangold, Jeffrey A. Cramer, Peter S, Corinne J. Hackbarth, Dawn Z. Chen, Jason G. Lewis
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
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المؤلفون: James B. Mangold, Fan Wu, Sam Rebello
المصدر: Clinical Pharmacology in Drug Development. 5:245-249
مصطلحات موضوعية: CYP3A, business.industry, Pharmaceutical Science, Pharmacology, Bioinformatics, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, 030220 oncology & carcinogenesis, medicine, Biomarker (medicine), Midazolam, Pharmacology (medical), 4β hydroxycholesterol, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::63feb9238fc242aa4ad4d72f20eacc4eTest
https://doi.org/10.1002/cpdd.265Test -
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المؤلفون: Diego Albrecht, Priya Chandra, Su-Er W Huskey, Timothy Bedman, Helen Gu, Yancy Du, Lai Wang, Heidi J. Einolf, Jimmy Flarakos, Qusai Al-Share, Pierre Jordaan, James B. Mangold
المصدر: Xenobiotica. 46:986-1000
مصطلحات موضوعية: Adult, medicine.medical_specialty, Health, Toxicology and Mutagenesis, Tetrazoles, 030204 cardiovascular system & hematology, Pharmacology, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Sacubitril, Excretion, 03 medical and health sciences, 0302 clinical medicine, Internal medicine, medicine, Humans, Neprilysin, Active metabolite, Angiotensin II receptor type 1, Chemistry, Aminobutyrates, Biphenyl Compounds, General Medicine, Angiotensin II, Drug Combinations, Endocrinology, Valsartan, Angiotensin II Type 1 Receptor Blockers, Sacubitril, Valsartan, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5dd5ac3bc55fe71658e7ca18f5dc22d8Test
https://doi.org/10.3109/00498254.2015.1014944Test -
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المؤلفون: Alexandra Vargas, Oliver Simon, Matthias Kittelmann, Melissa M. Lin, Chun-qi Zhu, Hongmei Li, Su-Er W. Huskey, Helen Gu, Sarah Favara, Handan He, Jin Zhang, Ry R. Forseth, Lai Wang, Alexandre Luneau, Heidi J. Einolf, Fabian K. Eggimann, James B. Mangold
المصدر: Drug Metabolism and Disposition. 44:653-664
مصطلحات موضوعية: Male, 0301 basic medicine, Indoles, Stereochemistry, Metabolite, 030106 microbiology, Pharmaceutical Science, Hydroxylation, Feces, 03 medical and health sciences, chemistry.chemical_compound, Dogs, Cytochrome P-450 Enzyme System, Biotransformation, Spiroindolone, Animals, Bile, Humans, Spiro Compounds, Rats, Wistar, Pharmacology, CYP3A4, biology, CYP1A2, Cytochrome P450, Metabolism, Malaria, Rats, 030104 developmental biology, Biochemistry, chemistry, Hepatocytes, biology.protein
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::902b00e7c77e9089acdaff2832b721fbTest
https://doi.org/10.1124/dmd.115.069112Test -
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المؤلفون: Gangadhar Sunkara, Helen Gu, Tycho Heimbach, James B. Mangold, Handan He, Avantika Barve, Imad Hanna, Binfeng Xia, June Ke, Tao Zhang, Heidi J. Einolf, Natalya Alexander, Lai Wang
المصدر: European Journal of Pharmaceutical Sciences. 63:103-112
مصطلحات موضوعية: Physiologically based pharmacokinetic modelling, Alisporivir, Dose-Response Relationship, Drug, CYP3A4, Chemistry, Cmax, Administration, Oral, Pharmaceutical Science, Pharmacology, Models, Biological, Ketoconazole, Pharmacokinetics, In vivo, Cyclosporine, medicine, Cytochrome P-450 CYP3A, Humans, Distribution (pharmacology), Drug Interactions, Caco-2 Cells, Rifampin, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ebe29338a603ab86c1d2f89a19b88662Test
https://doi.org/10.1016/j.ejps.2014.06.021Test -
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المؤلفون: Handan He, Heidi J. Einolf, Christina S. Won, Lai Wang, Helen Gu, Wen Lin, Dung Yu Chun, James B. Mangold
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 45(12)
مصطلحات موضوعية: Physiologically based pharmacokinetic modelling, Indoles, medicine.drug_class, Midazolam, Pharmaceutical Science, Pharmacology, Hydroxamic Acids, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, In vivo, Panobinostat, medicine, Cytochrome P-450 CYP3A, Cytochrome P-450 Enzyme Inhibitors, Humans, Drug Interactions, Chemistry, Histone deacetylase inhibitor, Area under the curve, Gastric Acidity Determination, Drug interaction, Cytochrome P-450 CYP2C19, Histone Deacetylase Inhibitors, 030220 oncology & carcinogenesis, Enzyme Induction, Microsomes, Liver, Ketoconazole, Rifampin, Oxidation-Reduction, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::38cd9dac1e23d8ca3898d85896f59acaTest
https://pubmed.ncbi.nlm.nih.gov/28912253Test -
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المؤلفون: S. Ken Tanaka, Jimmy Flarakos, James B. Mangold, Yancy Du, Wenyu Hu, Wen Lin, Handan He, Stephen Villano
المصدر: Antimicrobial Agents and Chemotherapy
مصطلحات موضوعية: Male, 0301 basic medicine, medicine.medical_specialty, 030106 microbiology, Thyroid Gland, Administration, Oral, Bone and Bones, Drug Administration Schedule, Excretion, 03 medical and health sciences, Harderian gland, Pharmacokinetics, Internal medicine, Intestinal Elimination, medicine, Animals, Rats, Long-Evans, Tissue Distribution, Pharmacology (medical), aminomethylcycline, ADME, Melanins, Pharmacology, Volume of distribution, Bone mineral, Salivary gland, Harderian Gland, Chemistry, Thyroid, omadacycline, animal models, Anti-Bacterial Agents, Rats, Hepatobiliary Elimination, Infectious Diseases, medicine.anatomical_structure, Endocrinology, Tetracyclines, Administration, Intravenous, Half-Life
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fce5d50abef848379331c0a3cc492355Test
https://doi.org/10.1128/aac.01784-16Test -
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المؤلفون: Wenkui Li, Su-Er W Huskey, Jimmy Flarakos, James B. Mangold
المصدر: Bioanalysis. 6:617-628
مصطلحات موضوعية: Drug Industry, Computer science, Metabolite, Drug metabolite, Clinical Biochemistry, Drug Evaluation, Preclinical, Nanotechnology, General Medicine, Tiered approach, Biomarkers, Pharmacological, Analytical Chemistry, In vitro analysis, Medical Laboratory Technology, Identification (information), chemistry.chemical_compound, Pharmaceutical Preparations, Drug development, chemistry, Risk analysis (engineering), Drug Discovery, Plasma concentration, Humans, General Pharmacology, Toxicology and Pharmaceutics
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dfa27c767ad94acccaf31ee40a26b5caTest
https://doi.org/10.4155/bio.14.25Test -
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المؤلفون: S. Ken Tanaka, Daniel S. Stein, Yancy Du, Lillian Ting, Lai Wang, Heidi J. Einolf, James B. Mangold, Haiying Sun, Wei Zhou, Helen Gu, Adrienne Natrillo, Jimmy Flarakos, Stephen Villano, Imad Hanna, Bing Zhu, Natalia Alexander, Steven J. Kovacs, Kiran Dole, Dung Y Chun
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 47(8)
مصطلحات موضوعية: 0301 basic medicine, Adult, Male, medicine.medical_specialty, ATP Binding Cassette Transporter, Subfamily B, Metabolic Clearance Rate, Health, Toxicology and Mutagenesis, 030106 microbiology, Administration, Oral, Urine, Absorption (skin), Pharmacology, Biology, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Internal medicine, medicine, Distribution (pharmacology), Humans, Drug Interactions, Volume of distribution, Half-life, Cytochrome P450, General Medicine, Metabolism, Anti-Bacterial Agents, Endocrinology, Tetracyclines, Area Under Curve, Microsome, biology.protein, Microsomes, Liver, Half-Life
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::08bbb285a89d1f100a75a224e6ffc591Test
https://pubmed.ncbi.nlm.nih.gov/27499331Test -
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المؤلفون: Tsu-han Lin, Yanfeng Wang, Ke Hu, James B. Mangold, Jimmy Flarakos, Handan He, M. Sharr-McMahon
المصدر: Cancer Chemotherapy and Pharmacology. 72:181-188
مصطلحات موضوعية: Pharmacology, Cancer Research, medicine.medical_specialty, Somatostatin receptor binding, Metabolite, Half-life, Urine, Toxicology, Pasireotide, Intestinal absorption, Excretion, chemistry.chemical_compound, Endocrinology, Oncology, chemistry, Pharmacokinetics, Internal medicine, medicine, Pharmacology (medical)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::1b4703f1c0e48a344551f4acede3a36eTest
https://doi.org/10.1007/s00280-013-2183-0Test