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1دورية أكاديمية
المؤلفون: Shi Liu, Eileen J. Daley, Lauren My-Linh Tran, Zhen Yu, Monica Reyes, Thomas Dean, Ashok Khatri, Paul M. Levine, Aaron T. Balana, Matthew R. Pratt, Harald Jüppner, Samuel H. Gellman, Thomas J. Gardella
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Molecular Biology, Physiology, Pharmacology, Biotechnology, Immunology, Cancer, Science Policy, Biological Sciences not elsewhere classified, mediating calcium homeostasis, displays prolonged activity, peptidic pth1r inhibitor, peptidic pth1r antagonists, ameliorate pth1r malfunction, acting inverse agonist, backbone modification provides, inverse agonist, modification strategy, type pth1r, inverse agonists, therapeutic potential, therapeutic agents, poor pharmacokinetics, pharmacodynamics undermine, peptide may, key role, future development, bone development
الإتاحة: https://doi.org/10.1021/jacs.3c09694.s001Test
https://figshare.com/articles/journal_contribution/Backbone_Modification_Provides_a_Long-Acting_Inverse_Agonist_of_Pathogenic_Constitutively_Active_PTH1R_Variants/25308374Test -
2دورية أكاديمية
المؤلفون: István Ledneczki, Pál Tapolcsányi, Eszter Gábor, János Éles, Júlia Barabás, Zoltán Béni, Balázs Varga, Ottilia Balázs, Viktor Román, László Fodor, Judit Szikra, Mónika Vastag, György Lévay, Éva Schmidt, Balázs Lendvai, István Greiner, Béla Kiss, Zsolt Némethy, Sándor Mahó
مصطلحات موضوعية: Biochemistry, Molecular Biology, Neuroscience, Pharmacology, Cancer, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, vitro functional tests, r activity together, predict binding modes, molecular docking studies, inverse agonist property, inverse agonist features, based sar considerations, inverse agonists steroid, vivo dipsogenia test, rat liver microsomes, hts hit molecules, based histamine h, 3 sub, novel steroid, vivo potency, vivo h, special emphasis, receptor antagonists, place recognition, considerably stable
الإتاحة: https://doi.org/10.1021/acs.jmedchem.3c02117.s002Test
https://figshare.com/articles/journal_contribution/Discovery_of_Novel_Steroid-Based_Histamine_H_sub_3_sub_Receptor_Antagonists_Inverse_Agonists/25276448Test -
3دورية أكاديمية
المصدر: Exploration of Neuroprotective Therapy, Vol 3, Iss 5, Pp 258-267 (2023)
مصطلحات موضوعية: cannabinoid 2 receptor, jwh133, cannabinoid 2 receptor overexpression, constitutive cannabinoid 2 receptor activity, cannabinoid 2 inverse agonist/antagonist am630, mek-erk phosphorylation/activation, mouse brain cortex, Neurology. Diseases of the nervous system, RC346-429
وصف الملف: electronic resource
العلاقة: https://www.explorationpub.com/Journals/ent/Article/100450Test; https://doaj.org/toc/2769-6510Test
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4دورية أكاديمية
المؤلفون: Mariusz Geremek, Bogna Drozdzowska, Dorota Łażewska, Katarzyna Kieć-Kononowicz, Jerzy Jochem
المصدر: Pharmaceuticals, Vol 17, Iss 6, p 792 (2024)
مصطلحات موضوعية: periodontitis, H3 receptor antagonist/inverse agonist, RANKL/RANK/OPG, Medicine, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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5دورية أكاديمية
المؤلفون: Jacqueline C. Calderón, Passainte Ibrahim, Dorothea Gobbo, Francesco Luigi Gervasio, Timothy Clark
مصطلحات موضوعية: Biophysics, Biochemistry, Cell Biology, Molecular Biology, Neuroscience, Pharmacology, Immunology, Cancer, Hematology, Chemical Sciences not elsewhere classified, inverse agonists carazolol, inverse agonist ligands, agonist activity, inverse agonism, tempered multiple, seem also, receptor activity, neutral antagonists, neutral antagonist, neutral antagonism, metadynamics simulations, known microswitches, energy profiles, conformational states
الإتاحة: https://doi.org/10.1021/acs.jcim.3c01763.s001Test
https://figshare.com/articles/journal_contribution/Determinants_of_Neutral_Antagonism_and_Inverse_Agonism_in_the_sub_2_sub_Adrenergic_Receptor/25356196Test -
6دورية أكاديمية
المؤلفون: Miroslav Kosar, Roman C. Sarott, David A. Sykes, Alexander E. G. Viray, Rosa Maria Vitale, Nataša Tomašević, Xiaoting Li, Rudolf L. Z. Ganzoni, Bilal Kicin, Lisa Reichert, Kacper J. Patej, Uxía Gómez-Bouzó, Wolfgang Guba, Peter J. McCormick, Tian Hua, Christian W. Gruber, Dmitry B. Veprintsev, James A. Frank, Uwe Grether, Erick M. Carreira
مصطلحات موضوعية: Biophysics, Biochemistry, Molecular Biology, Neuroscience, Pharmacology, Immunology, Cancer, Infectious Diseases, Chemical Sciences not elsewhere classified, tailored functional response, privileged agonist hu, present study discloses, live cell erk, initial docking data, toggle switch trp258, inverse agonist functionality, probes employing bv, fluorescent probes retain, 9 b, 7 b, thereby stabilize cb, exhibits high affinity, 48 sup, 2 sub, 1 b, high affinity, >)-< b, inverse agonists, k <, gem <
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7دورية أكاديمية
المؤلفون: Yutaro Ohno, Eri Okita, Mika Kawai-Uchida, Youji Shoukei, Kazuhiro Soshiroda, Tomoyuki Kanda, Shinichi Uchida
المصدر: Journal of Pharmacological Sciences, Vol 152, Iss 3, Pp 193-199 (2023)
مصطلحات موضوعية: Anti-parkinsonian, Adenosine A2A receptor Antagonist/inverse agonist, L-DOPA, Dyskinesia, MPTP, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
العلاقة: http://www.sciencedirect.com/science/article/pii/S1347861323000312Test; https://doaj.org/toc/1347-8613Test
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8دورية أكاديمية
المؤلفون: Herbert P. Jennissen
المصدر: Frontiers in Bioengineering and Biotechnology, Vol 11 (2023)
مصطلحات موضوعية: angioinduction, osteoinduction, pico-technology, constitutive receptor activity, allosteric inverse agonist, orthosteric agonist, Biotechnology, TP248.13-248.65
وصف الملف: electronic resource
العلاقة: https://www.frontiersin.org/articles/10.3389/fbioe.2023.1226649/fullTest; https://doaj.org/toc/2296-4185Test
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9دورية أكاديمية
المؤلفون: Marcia G. Honig, Nobel A. Del Mar, Bob M. Moore, Anton Reiner
المصدر: Neurotrauma Reports, Vol 3, Iss 1, Pp 534-544 (2022)
مصطلحات موضوعية: anxiety, CB2 inverse agonist therapy, depression, fear, raloxifene, traumatic brain injury, Medical emergencies. Critical care. Intensive care. First aid, RC86-88.9
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2689-288XTest
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10دورية أكاديمية
المؤلفون: Wolfgang Sadee
المصدر: Molecules, Vol 28, Iss 17, p 6375 (2023)
مصطلحات موضوعية: GPCRs, ligand-free receptor signaling, inverse agonist, neutral antagonist, μ opioid receptor, opioid dependence, Organic chemistry, QD241-441
وصف الملف: electronic resource