-
1دورية أكاديمية
المؤلفون: Franck Brebion (2439052), Romain Gosmini (1738168), Pierre Deprez (1705699), Marie Varin (2479900), Christophe Peixoto (2035117), Luke Alvey (2035129), Hélène Jary (2035114), Natacha Bienvenu (1705657), Nicolas Triballeau (1400671), Roland Blanque (3989681), Céline Cottereaux (9412031), Thierry Christophe (242276), Nele Vandervoort (3989705), Patrick Mollat (206614), Robert Touitou (4376779), Philip Leonard (1621432), Frédéric De Ceuninck (1417306), Iuliana Botez (1701322), Alain Monjardet (3989687), Ellen van der Aar (3989690), David Amantini (232220)
مصطلحات موضوعية: Biochemistry, Medicine, Cell Biology, Neuroscience, Physiology, Pharmacology, Biotechnology, Cancer, Science Policy, Infectious Diseases, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, phase 2, knee OA, 1.5 μ M, DMOAD, hydantoin series, Biochemical activity, cocrystal structure, anticatabolic activity, IC 50, glycosaminoglycan release, disease-modifying osteoarthritis, mouse cartilage explants, NCT, GLPG, aggrecanase ADAMTS, HTS, fluorescence-based assay, AGC ELISA
-
2
المؤلفون: Alain Monjardet, Thierry Christophe, Nicolas Triballeau, Helene Jary, Luke Jonathan Alvey, Romain Luc Marie Gosmini, Frédéric André De Ceuninck, Pierre Deprez, Robert Touitou, Roland Blanque, D. Amantini, Nele Vandervoort, Ellen van der Aar, Philip Leonard, F. Brebion, Patrick Mollat, Natacha Bienvenu, C. Cottereaux, I. Botez, Varin Marie Laurence Claire, Christophe Peixoto
المصدر: Journal of Medicinal Chemistry. 64:2937-2952
مصطلحات موضوعية: Cartilage, Articular, Models, Molecular, Osteoarthritis, Pharmacology, 01 natural sciences, law.invention, Glycosaminoglycan, Mice, 03 medical and health sciences, Dogs, law, Drug Discovery, medicine, Animals, Humans, IC50, Aggrecan, Glycosaminoglycans, 030304 developmental biology, Aggrecanase, 0303 health sciences, Chemistry, Cartilage, ADAMTS, medicine.disease, Rats, 0104 chemical sciences, Mice, Inbred C57BL, 010404 medicinal & biomolecular chemistry, medicine.anatomical_structure, Recombinant DNA, Molecular Medicine, ADAMTS5 Protein
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e63e1d09bcd2c3ffc719892459e89ab3Test
https://doi.org/10.1021/acs.jmedchem.0c02008Test -
3
المؤلفون: Helene Jary, Pierre Deprez, Denis Guédin, Taoues Temal, Marielle Auberval, Sarah E. Lively, Jean-Paul Vevert
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2455-2459
مصطلحات موضوعية: Stereochemistry, Calcimimetic, Organic Chemistry, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Pharmacology, Biochemistry, chemistry.chemical_compound, chemistry, Benzothiazole, Oral administration, In vivo, Drug Discovery, Urea, Molecular Medicine, Calcium, Luciferase, Benzothiazoles, Calcium-sensing receptor, Receptors, Calcium-Sensing, Molecular Biology
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0c8a21b6d1e701976deea8c53e3973feTest
https://doi.org/10.1016/j.bmcl.2013.01.077Test -
4
المؤلفون: Catherine Robin-Jagerschmidt, Helene Jary, Ellen van der Aar, Nicolas Triballeau, Luke Jonathan Alvey, Francois Nique, Denis Guédin, Kris Van Beeck, Dominque Minet, Florence Namour, Jean H.M. Feyen, Pierre Deprez, Hugo Klaassen, Jean-Michel Lefrancois, Roland Blanque, Christophe Peixoto, Murielle Manioc, Séverine Hebbe, Stephen Robert Fletcher, Christopher Gaëtan Housseman
المصدر: Journal of Medicinal Chemistry. 55:8236-8247
مصطلحات موضوعية: Male, Models, Molecular, Transcriptional Activation, Stereochemistry, Molecular Conformation, Biological Availability, Hydantoin, Pharmacology, Partial agonist, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Anabolic Agents, In vivo, Drug Discovery, Androgen Receptor Antagonists, Animals, Humans, Hydroxymethyl, Muscle, Skeletal, Trifluoromethyl, Hydantoins, Prostate, Stereoisomerism, Organ Size, Rats, Bioavailability, Drug Partial Agonism, Androgen receptor, chemistry, Selective androgen receptor modulator, Receptors, Androgen, Androgens, Molecular Medicine, Orchiectomy, HeLa Cells
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::841982488e4fec11bfd3145a00ecb1c9Test
https://doi.org/10.1021/jm300281xTest -
5
المؤلفون: Sarah E. Lively, Jean-Paul Vevert, Helene Jary, Denis Guédin, Pierre Deprez, Marielle Auberval, Taoues Temal
المصدر: Bioorganicmedicinal chemistry letters. 23(8)
مصطلحات موضوعية: Fendiline, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Allosteric regulation, Substituent, Pharmaceutical Science, medicine.disease, Biochemistry, In vitro, chemistry.chemical_compound, Structure-Activity Relationship, chemistry, In vivo, Biomimetic Materials, Drug Discovery, Urea, medicine, Molecular Medicine, Secondary hyperparathyroidism, Calcium, Calcium-sensing receptor, Molecular Biology, Receptors, Calcium-Sensing
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cdfadc7accf2ee4adc8f34ad5287a975Test
https://pubmed.ncbi.nlm.nih.gov/23465611Test