المؤلفون: Gouault, Nicolas, Cariou, Alexandre, Cupif, Jean-François, Amaral, Patrícia de Aguiar, David, Michèle

المصدر: Química Nova. August 2016 39(7)

مصطلحات موضوعية: pyrazolones, fluorous tag, Heck coupling, allylic alcohols

وصف الملف: text/html

الوصول الحر: http://old.scielo.br/scielo.php?script=sci_arttext&pid=S0100-40422016000700825Test

المؤلفون: Amaral, Patricia de A., Petrignet, Julien, Gouault, Nicolas, Agustini, Taciane, Lohézic-Ledévéhat, Françoise, Cariou, Alexandre, Grée, René, Eifler-Lima, Vera L., David, Michèle

المصدر: Journal of the Brazilian Chemical Society. January 2009 20(9)

مصطلحات موضوعية: δ-valerolactones, kavaïn analogues, Heck, Sonogashira-Hagihara, Suzuki-Miyaura, tandem isomerization-aldolization, cytotoxicity

وصف الملف: text/html

الوصول الحر: http://old.scielo.br/scielo.php?script=sci_arttext&pid=S0103-50532009000900018Test

المؤلفون: Gantasala, Naresh, Fournet, Corentin, Roch, Myriam, Le, Lalli, Claudia, Pabbaraja, Srihari, Gouault, Nicolas

المساهمون: CSIR Indian Institute of Chemical Technology Hyderabad (IICT), Institut des Sciences Chimiques de Rennes (ISCR), Université de Rennes (UR)-Institut National des Sciences Appliquées - Rennes (INSA Rennes), Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Ecole Nationale Supérieure de Chimie de Rennes (ENSCR)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)

المصدر: ISSN: 1477-0520.

مصطلحات موضوعية: [CHIM.ORGA]Chemical Sciences/Organic chemistry

العلاقة: hal-04159035; https://hal.science/hal-04159035Test; https://hal.science/hal-04159035/documentTest; https://hal.science/hal-04159035/file/Revised-Article-2.pdfTest

الإتاحة: https://doi.org/10.1039/D3OB00545CTest
https://hal.science/hal-04159035Test
https://hal.science/hal-04159035/documentTest
https://hal.science/hal-04159035/file/Revised-Article-2.pdfTest

المؤلفون: Bergounioux, Alexandre, Lhotellier, Romane, Roisnel, Thierry, Gouault, Nicolas, Argouarch, Gilles, Lalli, Claudia

المساهمون: Institut des Sciences Chimiques de Rennes (ISCR), Université de Rennes (UR)-Institut National des Sciences Appliquées - Rennes (INSA Rennes), Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Ecole Nationale Supérieure de Chimie de Rennes (ENSCR)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)

المصدر: ISSN: 1615-4150.

مصطلحات موضوعية: Aza-Prins, Ketones, 2-Spiropiperidines, tetrasubstituted stereocenter, Titanium, [CHIM.ORGA]Chemical Sciences/Organic chemistry

العلاقة: hal-04357455; https://hal.science/hal-04357455Test; https://hal.science/hal-04357455/documentTest; https://hal.science/hal-04357455/file/revised%20draft.pdfTest

الإتاحة: https://doi.org/10.1002/adsc.202301116Test
https://hal.science/hal-04357455Test
https://hal.science/hal-04357455/documentTest
https://hal.science/hal-04357455/file/revised%20draft.pdfTest

المؤلفون: Le Roch, Myriam, Renault, Jacques, Argouarch, Gilles, Lenci, Elena, Trabocchi, Andrea, Roisnel, Thierry, Gouault, Nicolas, Lalli, Claudia

المساهمون: Institut des Sciences Chimiques de Rennes (ISCR), Université de Rennes (UR)-Institut National des Sciences Appliquées - Rennes (INSA Rennes), Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Ecole Nationale Supérieure de Chimie de Rennes (ENSCR)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS), Dipartimento di Chimica 'Ugo Schiff' Sesto Fiorentino (DICUS UniFI), Università degli Studi di Firenze = University of Florence = Université de Florence (UniFI), The authors thank Université de Rennes and CNRS for the financial support. The program “International Emerging Actions” of the CNRS is warmly acknowledged for founding this collaborative project. The CRMPO of the Institut des Sciences Chimiques de Rennes for mass measurement, the Centre de Diffractométrie X for X-ray analyses, and FEDER funds for acquisition of single-crystal equipment are gratefully acknowledged. Part of this work has been performed using the PRISM core facility (Biogenouest, UMS Biosit, Université de Rennes, 35000 Rennes, France). A.T. and E.L. acknowledge financial support provided by the MUR─Dipartimenti di Eccellenza 2023-2027 (DICUS 2.0) to the Department of Chemistry “Ugo Schiff”. Finally, Solenn Ferron is acknowledged for running 19F NMR experiments and Pr. Ph. Uriac for enriching discussions.

المصدر: ISSN: 0022-3263.

مصطلحات موضوعية: [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [CHIM.CHEM]Chemical Sciences/Cheminformatics

العلاقة: hal-04506336; https://hal.science/hal-04506336Test; https://hal.science/hal-04506336/documentTest; https://hal.science/hal-04506336/file/revised%20draft.pdfTest

الإتاحة: https://doi.org/10.1021/acs.joc.4c00143Test
https://hal.science/hal-04506336Test
https://hal.science/hal-04506336/documentTest
https://hal.science/hal-04506336/file/revised%20draft.pdfTest

المؤلفون: Brahmaiah, Dabbugoddu, Bhavani, Anagani Kanaka Durga, Aparna, Pasula, Kumar, Nangunoori Sampath, Solhi, Hélène, Le Guével, Rémy, Baratte, Blandine, Robert, Thomas, Ruchaud, Sandrine, Bach, Stéphane, Singh Jadav, Surender, Reddy, Chada Raji, Mosset, Paul, Gouault, Nicolas, Levoin, Nicolas, Grée, René

المساهمون: Jawaharlal Nehru Technological University, Hyderabad 500085, India (JNTU), Chemveda Life Sciences India, Osmania University, Plate-forme ImPACcell (ImPACcell), Structure Fédérative de Recherche en Biologie et Santé de Rennes ( Biosit : Biologie - Santé - Innovation Technologique ), ABiMS - Informatique et bioinformatique = Analysis and Bioinformatics for Marine Science (ABIMS), Fédération de recherche de Roscoff (FR2424), Station biologique de Roscoff = Roscoff Marine Station (SBR), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Station biologique de Roscoff = Roscoff Marine Station (SBR), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS), Laboratoire de Biologie Intégrative des Modèles Marins (LBI2M), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Station biologique de Roscoff = Roscoff Marine Station (SBR), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Centre National de la Recherche Scientifique (CNRS), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS), North-West University South Aftrica (NWU), Council of Scientific and Industrial Research India (CSIR), Institut des Sciences Chimiques de Rennes (ISCR), Université de Rennes (UR)-Institut National des Sciences Appliquées - Rennes (INSA Rennes), Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Ecole Nationale Supérieure de Chimie de Rennes (ENSCR)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS), Bioprojet-Biotech, Ligue contre le Cancer, Conseil Interregional Grand Ouest, Osmania University C-DST-PURSE-II/15/2019

المصدر: ISSN: 1420-3049 ; Molecules ; https://hal.science/hal-03828358Test ; Molecules, 2022, 27 (19), pp.6149. ⟨10.3390/molecules27196149⟩.

مصطلحات موضوعية: kinases, CLK-kinases, DYRK1A kinase, quinazoline, cytotoxicity, molecular modelling, [CHIM]Chemical Sciences

العلاقة: info:eu-repo/semantics/altIdentifier/pmid/36234686; hal-03828358; https://hal.science/hal-03828358Test; https://hal.science/hal-03828358/documentTest; https://hal.science/hal-03828358/file/molecules-27-06149-v2.pdfTest; PUBMED: 36234686

الإتاحة: https://doi.org/10.3390/molecules27196149Test
https://hal.science/hal-03828358Test
https://hal.science/hal-03828358/documentTest
https://hal.science/hal-03828358/file/molecules-27-06149-v2.pdfTest

المؤلفون: Dias de Melo, Guilherme, Coatnoan, Nicolas, Gouault, Nicolas, Cupif, Jean-François, Renault, Jacques, Cosson, Alain, Uriac, Philippe, Blondel, Arnaud, Minoprio, Paola

المساهمون: Processus infectieux à Trypanosomatidés - Trypanosomatids Infectious Processes, Institut Pasteur Paris (IP)-Université Paris Cité (UPCité), Institut des Sciences Chimiques de Rennes (ISCR), Université de Rennes (UR)-Institut National des Sciences Appliquées - Rennes (INSA Rennes), Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Ecole Nationale Supérieure de Chimie de Rennes (ENSCR)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS), Bioinformatique structurale - Structural Bioinformatics, Institut Pasteur Paris (IP)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité), This research project received financial support from the Agence Nationale pour la Recherche ANR-14-CE16-0001-01 and the recurring budget of the Institut Pasteur to the Laboratoire des Processus Infectieux à Trypanosomatidés. GDM was supported by ANR and Institut Carnot–Pasteur Microbes et Santé (Pasteur M&S) fellowships. Part of this work was performed at the UtechS Photonic BioImaging (PBI) platform, a member of the France Life Imaging network grant ANR-11-INBS-0006 ., ANR-14-CE16-0001,CHAGAS,Validation et optimisation de nouveaux composés thérapeutiques contre la Maladie de Chagas(2014), ANR-11-INBS-0006,FLI,France Life Imaging(2011)

المصدر: ISSN: 2213-7165.

مصطلحات موضوعية: Chagas disease, antiparasitic agents, drug development, enzyme inhibitor, medicinal chemistry, [SDV.MP]Life Sciences [q-bio]/Microbiology and Parasitology, [CHIM]Chemical Sciences

العلاقة: info:eu-repo/semantics/altIdentifier/pmid/34929377; hal-03504248; https://hal.science/hal-03504248Test; https://hal.science/hal-03504248/documentTest; https://hal.science/hal-03504248/file/Dias%20de%20Melo_1-s2.0-S2213716521002794-main.pdfTest; PUBMED: 34929377

الإتاحة: https://doi.org/10.1016/j.jgar.2021.10.030Test
https://hal.science/hal-03504248Test
https://hal.science/hal-03504248/documentTest
https://hal.science/hal-03504248/file/Dias%20de%20Melo_1-s2.0-S2213716521002794-main.pdfTest

المؤلفون: Gateau, Cécile, Dias de Melo, Guilherme, Uriac, Philippe, Tasseau, Olivier, Renault, Jacques, Blondel, Arnaud, Gouault, Nicolas, Barbut, Frédéric, Minoprio, Paola

المساهمون: Physiopathologie et Pharmacotoxicologie Placentaire Humaine (U1139), Université Paris Descartes - Paris 5 (UPD5)-Institut National de la Santé et de la Recherche Médicale (INSERM), CHU Saint-Antoine AP-HP, Assistance publique - Hôpitaux de Paris (AP-HP) (AP-HP)-Sorbonne Université (SU), Processus infectieux à Trypanosomatidés - Trypanosomatids Infectious Processes, Institut Pasteur Paris (IP)-Université Paris Cité (UPCité), Institut des Sciences Chimiques de Rennes (ISCR), Université de Rennes (UR)-Institut National des Sciences Appliquées - Rennes (INSA Rennes), Institut National des Sciences Appliquées (INSA)-Institut National des Sciences Appliquées (INSA)-Ecole Nationale Supérieure de Chimie de Rennes (ENSCR)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS), Bioinformatique structurale - Structural Bioinformatics, Institut Pasteur Paris (IP)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité), Institut Carnot Pasteur Microbes & Santé CARNOT/MS (ANR-16-CARN-0023-01 - non référencé dans AuréHAL), ANR-16-CARN-0025,PolyNat Carnot Institute,PolyNat Carnot Institute(2011)

المصدر: ISSN: 1747-0277.

مصطلحات موضوعية: Clostridioides difficile, antibacterial, enzyme inhibitors, proline racemase, structure-activity relationship, [SDV.MP]Life Sciences [q-bio]/Microbiology and Parasitology, [CHIM]Chemical Sciences

العلاقة: info:eu-repo/semantics/altIdentifier/pmid/34918458; hal-03504249; https://hal.science/hal-03504249Test; https://hal.science/hal-03504249/documentTest; https://hal.science/hal-03504249/file/Gateau%20et%20al.%20-%202022%20-%20Irreversible%20inhibitors%20of%20the%20proline%20racemase%20%28P.pdfTest; PUBMED: 34918458

الإتاحة: https://doi.org/10.1111/cbdd.14005Test
https://hal.science/hal-03504249Test
https://hal.science/hal-03504249/documentTest
https://hal.science/hal-03504249/file/Gateau%20et%20al.%20-%202022%20-%20Irreversible%20inhibitors%20of%20the%20proline%20racemase%20%28P.pdfTest

المؤلفون: de Melo, Guilherme Dias, Coatnoan, Nicolas, Gouault, Nicolas, Cupif, Jean-François, Renault, Jacques, Cosson, Alain, Uriac, Philippe, Blondel, Arnaud, Minoprio, Paola

المصدر: Journal of Global Antimicrobial Resistance ; volume 28, page 84-89 ; ISSN 2213-7165

مصطلحات موضوعية: Microbiology (medical), Immunology, Immunology and Allergy, Microbiology

الإتاحة: https://doi.org/10.1016/j.jgar.2021.10.030Test
https://api.elsevier.com/content/article/PII:S2213716521002794?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S2213716521002794?httpAccept=text/plainTest

المؤلفون: Bergounioux, Alexandre, Lhotellier, Romane, Roisnel, Thierry, Gouault, Nicolas, Argouarch, Gilles, Lalli, Claudia

المصدر: Advanced Synthesis & Catalysis; 1/9/2024, Vol. 366 Issue 1, p31-35, 5p

مصطلحات موضوعية: KETONES, CARBON, DIASTEREOISOMERS, ISOMERS, RING formation (Chemistry), AZA compounds, TITANIUM