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1
المؤلفون: William J. Greenlee, William Billard, Herbert Binch, Lian-Yong Chen, Ruth A. Duffy, Charles Liu, Gordon Crosby, Stuart W. McCombie, John W. Clader, Jennifer Ford, Shengjian Li, Joseph A. Kozlowski, Gowei Zhou, Vice Susan F, Jean E. Lachowicz
المصدر: Bioorganic & Medicinal Chemistry. 12:319-326
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Biological Availability, Pharmaceutical Science, Carboxamide, CHO Cells, Muscarinic Antagonists, Pharmacology, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Piperidines, In vivo, Cricetinae, Drug Discovery, Muscarinic acetylcholine receptor, Avoidance Learning, medicine, Animals, Structure–activity relationship, ortho-Aminobenzoates, Molecular Biology, Receptor, Muscarinic M2, Dose-Response Relationship, Drug, Chemistry, Organic Chemistry, Antagonist, In vitro, Rats, Bioavailability, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e7fb6725ef949509463e302ecb37ec1fTest
https://doi.org/10.1016/j.bmc.2003.11.005Test -
2
المؤلفون: Dennis V. Nazareno, Guowei Zhou, Herbert Binch, William J. Greenlee, Mary Cohen-Williams, Jayaram R. Tagat, Diane E. Grotz, Jean E. Lachowicz, James J. Kaminski, Joseph A. Kozlowski, Gordon Crosby, Stuart W. McCombie, Vicki L. Coffin, Kathleen Cox, Vilma Ruperto, Craig D. Boyle, Samuel Chackalamannil, Ruth A. Duffy, Hubert B. Josien, Yuguang Wang, John W. Clader, William Billard
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2311-2314
مصطلحات موضوعية: Stereochemistry, Microdialysis, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Dioxoles, Muscarinic Antagonists, Benzylidene Compounds, Biochemistry, Structure-Activity Relationship, Cytochrome P-450 Enzyme System, Drug Stability, Pharmacokinetics, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Humans, Moiety, Sulfones, Molecular Biology, Receptor, Muscarinic M2, Oxidative metabolism, Chemistry, Organic Chemistry, Muscarinic antagonist, Receptors, Muscarinic, Acetylcholine, Rats, Bioavailability, Macaca fascicularis, Area Under Curve, Drug Design, Microsomes, Liver, Microsome, Molecular Medicine, Selectivity, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4596ee0f6758218aaf4305ca38b8523fTest
https://doi.org/10.1016/s0960-894xTest(01)00435-8 -
3
المؤلفون: Ruth A. Duffy, Sundeep Dugar, Gordon Crosby, Vilma Ruperto, Herbert Binch, Robert D. McQuade, Lian-Yong Chen, Kristen Bratzler, John W. Clader, Lisa A. Taylor, Pradeep B. Pushpavanam, Jean E. Lachowicz, William Billard
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2209-2212
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Muscarinic Antagonists, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Potency, Molecular Biology, Acetylcholine receptor, Receptor, Muscarinic M2, Molecular Structure, Chemistry, Organic Chemistry, Receptors, Muscarinic, Acetylcholine, Corpus Striatum, Rats, Piperazine, Molecular Medicine, Piperidine, Lead compound, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6a0f16531fa2122abbc029d35dfcd592Test
https://doi.org/10.1016/s0960-894xTest(00)00437-6 -
4
المؤلفون: Samuel Chackalamannil, Ruth A. Duffy, William J. Greenlee, Gordon Crosby, Zhiyong Hu, Robert D. McQuade, Herbert Binch, Vilma Ruperto, William Billard, Yuguang Wang, John W. Clader, Jean E. Lachowicz
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2247-2250
مصطلحات موضوعية: Microdialysis, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Muscarinic Antagonists, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Piperidines, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Molecular Biology, Acetylcholine receptor, Receptor, Muscarinic M2, Chemistry, Receptor, Muscarinic M1, Organic Chemistry, Antagonist, Brain, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Receptors, Muscarinic, Acetylcholine, Rats, Drug Design, Molecular Medicine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::db62408e0f1c04cc91498acbe2956e04Test
https://doi.org/10.1016/s0960-894xTest(00)00457-1 -
5
المؤلفون: Guowei Zhou, Ruth A. Duffy, Herbert Binch, Jean E. Lachowicz, Lisa A. Taylor, William Billard, Derek B. Lowe, Joseph A. Kozlowski, Robert D. McQuade, Gordon Crosby, Vilma Ruperto, Henry Guzik
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2255-2257
مصطلحات موضوعية: Pyridines, Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Muscarinic Antagonists, Naphthalenes, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Alkaloids, Piperidines, Dibenzazepines, Drug Discovery, Muscarinic acetylcholine receptor, Benzene Derivatives, medicine, Animals, Humans, Structure–activity relationship, Furans, Receptor, Molecular Biology, Receptor, Muscarinic M2, Organic Chemistry, Antagonist, Muscarinic antagonist, Muscarinic acetylcholine receptor M2, Sulfoxide, Receptors, Muscarinic, Acetylcholine, Corpus Striatum, Recombinant Proteins, Rats, chemistry, Drug Design, Molecular Medicine, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4687a6dfde6b8966420c582c2ce3bbebTest
https://doi.org/10.1016/s0960-894xTest(00)00438-8 -
6
المؤلفون: Gordon Crosby, Ruth A. Duffy, Allen Barnett, Cheryl C. Anderson, Robert D. McQuade, Richard E. Chipkin, Vicki L. Coffin
المصدر: Journal of Neurochemistry. 57:2001-2010
مصطلحات موضوعية: Male, Time Factors, Stereochemistry, Pharmacology, Ligands, Tritium, Binding, Competitive, Biochemistry, Receptors, Dopamine, Cellular and Molecular Neuroscience, chemistry.chemical_compound, Dopamine receptor D1, In vivo, polycyclic compounds, medicine, Radioligand, Animals, heterocyclic compounds, Receptor, SCH-23390, Behavior, Animal, Chemistry, Receptors, Dopamine D1, organic chemicals, Antagonist, Dopamine antagonist, Rats, Inbred Strains, Benzazepines, Corpus Striatum, In vitro, Rats, carbohydrates (lipids), nervous system, Dopamine Antagonists, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c38d7e56a20ffb019766b75477fda742Test
https://doi.org/10.1111/j.1471-4159.1991.tb06415.xTest -
7
المؤلفون: Samuel Chackalamannil, Ruth A. Duffy, Yuguang Wang, Herbert Binch, Zhiyong Hu, William Billard, Mary Cohen-Williams, Kathleen Cox, William J. Greenlee, Diane E. Grotz, Vilma Ruperto, Gordon Crosby, Craig D. Boyle, Vicki L. Coffin, John W. Clader, James J. Kaminski, Jean E. Lachowicz
المصدر: Journal of medicinal chemistry. 45(25)
مصطلحات موضوعية: Drug, media_common.quotation_subject, Microdialysis, Molecular Conformation, Administration, Oral, Muscarinic Antagonists, Pharmacology, In Vitro Techniques, chemistry.chemical_compound, Structure-Activity Relationship, Pharmacokinetics, Piperidines, In vivo, Oral administration, Drug Discovery, Muscarinic acetylcholine receptor, Avoidance Learning, Animals, Humans, media_common, Acetylcholine receptor, Autoreceptors, Receptor, Muscarinic M2, Chemistry, Antagonist, Receptors, Muscarinic, Acetylcholine, Corpus Striatum, Rats, Molecular Medicine, Piperidine, Central Nervous System Agents
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b8f01b5159480e9fea3765195aa02e5dTest
https://pubmed.ncbi.nlm.nih.gov/12459007Test -
8
المؤلفون: Kathleen Cox, Vilma Ruperto, Stuart W. McCombie, Claire M. Lankin, Gordon Crosby, Vice Susan F, Vicki L. Coffin, Diane E. Grotz, Mary-Cohen Williams, Craig D. Boyle, Jean E. Lachowicz, Herbert Binch, Samuel Chackalamannil, Ruth A. Duffy, Jennifer Campion, William Billard
المصدر: Bioorganicmedicinal chemistry letters. 12(23)
مصطلحات موضوعية: Stereochemistry, Microdialysis, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Muscarinic Antagonists, Biochemistry, Chemical synthesis, Benzylidene Compounds, Sulfone, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, Animals, Humans, Benzamide, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, Receptors, Muscarinic, Acetylcholine, Bioavailability, Rats, Area Under Curve, Drug Design, Benzamides, Microsomes, Liver, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::14a5968458929f694f38fca5c0351bd4Test
https://pubmed.ncbi.nlm.nih.gov/12419388Test -
9
المؤلفون: Robert A McQuade, Herbert Binch, Vilma Ruperto, Jean E. Lachowicz, Guowei Zhou, Stuart W. McCombie, William Billard, Sue Ing Lin, Ruth A. Duffy, Gordon Crosby, Lisa A. Taylor, Jayaram R. Tagat, Joseph A. Kozlowski
المصدر: Bioorganicmedicinal chemistry letters. 12(5)
مصطلحات موضوعية: Microdialysis, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Ligands, Biochemistry, Chemical synthesis, Piperazines, Sulfone, chemistry.chemical_compound, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Molecular Biology, Acetylcholine receptor, Receptor, Muscarinic M2, Binding Sites, Bicyclic molecule, Molecular Structure, Chemistry, Organic Chemistry, Receptor, Muscarinic M1, Receptors, Muscarinic, Acetylcholine, Rats, Molecular Medicine, Selectivity, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::483484643f1278578603267627de339aTest
https://pubmed.ncbi.nlm.nih.gov/11859004Test -
10
المؤلفون: Michael Grzelak, William Billard, Henry Guzik, Herbert Binch, Derek B. Lowe, Pond Annamarie, Galen J Carey, Joseph A. Kozlowski, Mary Cohen-Williams, Gordon Crosby, Vicki L. Coffin, Robert W. Watkins, Richard P. Tedesco
المصدر: European journal of pharmacology. 431(2)
مصطلحات موضوعية: Male, Microdialysis, Time Factors, Scopolamine, Blood Pressure, Striatum, CHO Cells, Muscarinic Antagonists, Pharmacology, Piperazines, Rats, Sprague-Dawley, Mice, Cognition, Heart Rate, Cricetinae, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M4, medicine, Animals, Saimiri, Cholinesterase, Receptor, Muscarinic M2, biology, Molecular Structure, Chemistry, Antagonist, Brain, Muscarinic acetylcholine receptor M2, Receptors, Muscarinic, Acetylcholine, Rats, biology.protein, Neuroscience, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::388b7b6c66eb795f1e93a028ba5aee5fTest
https://pubmed.ncbi.nlm.nih.gov/11728425Test