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1دورية أكاديمية
المؤلفون: Mori, Matteo, Cocorullo, Mario, Tresoldi, Andrea, Cazzaniga, Giulia, Gelain, Arianna, Stelitano, Giovanni, Chiarelli, Laurent R, Tomaiuolo, Martina, Delre, Pietro, Mangiatordi, Giuseppe F, Garofalo, Mariangela, Cassetta, Alberto, Covaceuszach, Sonia, Villa, Stefania, Meneghetti, Fiorella
المساهمون: M. Mori, M. Cocorullo, A. Tresoldi, G. Cazzaniga, A. Gelain, G. Stelitano, L.R. Chiarelli, M. Tomaiuolo, P. Delre, G.F. Mangiatordi, M. Garofalo, A. Cassetta, S. Covaceuszach, S. Villa, F. Meneghetti
مصطلحات موضوعية: Chorismate, Crystal structure, Cystic fibrosi, Inhibition, Mycobacterium abscessu, Non-tuberculous mycobacteria, Salicylate synthase, Siderophore, Settore CHIM/08 - Chimica Farmaceutica
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/38169270; volume:265; firstpage:1; lastpage:13; numberofpages:13; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/2434/1023181Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85181702111
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2دورية أكاديمية
المؤلفون: Cazzaniga, Giulia, Tresoldi, Andrea, Gelain, Arianna, Meneghetti, Fiorella, Mori, Matteo, Villa, Stefania
المصدر: Chemistry & Biodiversity ; volume 21, issue 2 ; ISSN 1612-1872 1612-1880
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3دورية أكاديمية
المؤلفون: Mori, Matteo, Stelitano, Giovanni, Griego, Anna, Chiarelli, Laurent R, Cazzaniga, Giulia, Gelain, Arianna, Pini, Elena, Camera, Marina, Canzano, Paola, Fumagalli, Andrea, Scarpa, Edoardo, Cordiglieri, Chiara, Rizzello, Loris, Villa, Stefania, Meneghetti, Fiorella
المساهمون: M. Mori, G. Stelitano, A. Griego, L.R. Chiarelli, G. Cazzaniga, A. Gelain, E. Pini, M. Camera, P. Canzano, A. Fumagalli, E. Scarpa, C. Cordiglieri, L. Rizzello, S. Villa, F. Meneghetti
مصطلحات موضوعية: drug development, drug resistance, furan, murine alveolar-like macrophage, mycobactin, siderophore, tuberculosi, Settore CHIM/08 - Chimica Farmaceutica
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/36015139; info:eu-repo/semantics/altIdentifier/wos/WOS:000846563600001; volume:15; issue:8; firstpage:1; lastpage:22; numberofpages:22; journal:PHARMACEUTICALS; http://hdl.handle.net/2434/936726Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85137364957
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4دورية أكاديمية
المساهمون: M. Mori, G. Cazzaniga, F. Meneghetti, S. Villa, A. Gelain
مصطلحات موضوعية: Sirtuin 5, HDAC, activator, inhibitor, natural compound, small molecule, Settore CHIM/08 - Chimica Farmaceutica
العلاقة: info:eu-repo/semantics/altIdentifier/wos/WOS:000833379300001; volume:27; issue:14; firstpage:4449; lastpage:1; numberofpages:17; journal:MOLECULES; http://hdl.handle.net/2434/934006Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85135111597
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5دورية أكاديمية
المؤلفون: Mori, Matteo, Stelitano, Giovanni, Gelain, Arianna, Pini, Elena, Chiarelli, Laurent, Sammartino, José, Poli, Giulio, Tuccinardi, Tiziano, Beretta, Giangiacomo, Porta, Alessio, Bellinzoni, Marco, Villa, Stefania, Meneghetti, Fiorella
المساهمون: Università degli Studi di Milano = University of Milan (UNIMI), Università degli Studi di Pavia = University of Pavia (UNIPV), University of Pisa - Università di Pisa, Temple University Philadelphia, Pennsylvania Commonwealth System of Higher Education (PCSHE), Microbiologie structurale - Structural Microbiology (Microb. Struc. (UMR_3528 / U-Pasteur_5)), Institut Pasteur Paris (IP)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité), This work was funded by University of Milan (Linea B) and the Italian Ministry of Education, University and Research (MIUR): Dipartimenti di Eccellenza Program (2018–2022) - Dept. of Biology and Biotechnology “L. Spallanzani”, University of Pavia. Partial support was also provided by institutional grants from Institut Pasteur and CNRS.
المصدر: ISSN: 0022-2623.
مصطلحات موضوعية: MESH: Crystallography, X-Ray, MESH: Drug Design, MESH: Lyases, MESH: Magnesium, MESH: Models, Molecular, MESH: Mycobacterium tuberculosis, MESH: Protein Conformation, MESH: Structure-Activity Relationship, [CHIM.CRIS]Chemical Sciences/Cristallography, [SDV.BBM.BS]Life Sciences [q-bio]/Biochemistry, Molecular Biology/Structural Biology [q-bio.BM], [SDV.BBM]Life Sciences [q-bio]/Biochemistry, Molecular Biology, [INFO.INFO-BI]Computer Science [cs]/Bioinformatics [q-bio.QM], [PHYS.PHYS.PHYS-BIO-PH]Physics [physics]/Physics [physics]/Biological Physics [physics.bio-ph], [SDV.BC]Life Sciences [q-bio]/Cellular Biology
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/32530281; pasteur-03257004; https://pasteur.hal.science/pasteur-03257004Test; https://pasteur.hal.science/pasteur-03257004/documentTest; https://pasteur.hal.science/pasteur-03257004/file/acs.jmedchem.0c00373.pdfTest; PUBMED: 32530281; PUBMEDCENTRAL: PMC8008425
الإتاحة: https://doi.org/10.1021/acs.jmedchem.0c00373Test
https://pasteur.hal.science/pasteur-03257004Test
https://pasteur.hal.science/pasteur-03257004/documentTest
https://pasteur.hal.science/pasteur-03257004/file/acs.jmedchem.0c00373.pdfTest -
6دورية أكاديمية
المؤلفون: Chiarelli, Laurent R, Mori, Matteo, Barlocco, Daniela, Beretta, Giangiacomo, Gelain, Arianna, Pini, Elena, Porcino, Marianna, Mori, Giorgia, Stelitano, Giovanni, Costantino, Luca, Lapillo, Margherita, Bonanni, Davide, Poli, Giulio, Tuccinardi, Tiziano, Villa, Stefania, Meneghetti, Fiorella
المساهمون: Chiarelli, Laurent R, Mori, Matteo, Barlocco, Daniela, Beretta, Giangiacomo, Gelain, Arianna, Pini, Elena, Porcino, Marianna, Mori, Giorgia, Stelitano, Giovanni, Costantino, Luca, Lapillo, Margherita, Bonanni, Davide, Poli, Giulio, Tuccinardi, Tiziano, Villa, Stefania, Meneghetti, Fiorella
مصطلحات موضوعية: Antimycobacterial drug, Drug design, Iron, Siderophore, Tuberculosi, Virtual screening, Antitubercular Agent, Dose-Response Relationship, Drug, Enzyme Inhibitor, Lyase, Microbial Sensitivity Test, Models, Molecular, Molecular Structure, Mycobacterium tuberculosi, Structure-Activity Relationship, Drug Discovery
وصف الملف: ELETTRONICO
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/29940465; info:eu-repo/semantics/altIdentifier/wos/WOS:000441856300060; volume:155; firstpage:754; lastpage:763; numberofpages:10; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/11568/944058Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85048885433; https://www.sciencedirect.com/science/article/pii/S0223523418305245Test
الإتاحة: https://doi.org/10.1016/j.ejmech.2018.06.033Test
http://hdl.handle.net/11568/944058Test
https://www.sciencedirect.com/science/article/pii/S0223523418305245Test -
7دورية أكاديمية
المؤلفون: Pini, Elena, Poli, Giulio, Tuccinardi, Tiziano, Chiarelli, Laurent Roberto, Mori, Matteo, Gelain, Arianna, Costantino, Luca, Villa, Stefania, Meneghetti, Fiorella, Barlocco, Daniela
المساهمون: Pini, Elena, Poli, Giulio, Tuccinardi, Tiziano, Chiarelli, Laurent Roberto, Mori, Matteo, Gelain, Arianna, Costantino, Luca, Villa, Stefania, Meneghetti, Fiorella, Barlocco, Daniela
مصطلحات موضوعية: MD simulation, antimycobacterial agent, chorismate, consensus docking, iron, mycobactin, siderophore, Amino Acid Motif, Antitubercular Agent, Bacterial Protein, Catalytic Domain, Chorismic Acid, Chroman, Enzyme Inhibitor, Gene Expression, Kinetic, Lyase, Molecular Docking Simulation, Mycobacterium tuberculosi, Protein Binding, Protein Interaction Domains and Motif, Protein Structure, Secondary, Recombinant Protein, Structure-Activity Relationship, Substrate Specificity, Thermodynamics
وصف الملف: ELETTRONICO
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/29933627; info:eu-repo/semantics/altIdentifier/wos/WOS:000445301800009; volume:23; issue:7; journal:MOLECULES; http://hdl.handle.net/11568/944112Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85049414949; https://www.mdpi.com/1420-3049/23/7/1506Test
الإتاحة: https://doi.org/10.3390/molecules23071506Test
http://hdl.handle.net/11568/944112Test
https://www.mdpi.com/1420-3049/23/7/1506Test -
8دورية أكاديمية
المؤلفون: Mori, Matteo, Sammartino, José Camilla, Costantino, Luca, Gelain, Arianna, Meneghetti, Fiorella, Villa, Stefania, Chiarelli, Laurent Roberto
المساهمون: M. Mori, J.C. Sammartino, L. Costantino, A. Gelain, F. Meneghetti, S. Villa, L.R. Chiarelli
مصطلحات موضوعية: Serine/Threonine Protein Kinase, Tuberculosi, antitubercular drug, kinase inhibition, transmembrane signal transduction, virulence inhibition, Settore CHIM/08 - Chimica Farmaceutica, Settore BIO/10 - Biochimica
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/30827246; info:eu-repo/semantics/altIdentifier/wos/WOS:000472149500002; volume:19; issue:9; firstpage:646; lastpage:661; numberofpages:16; journal:CURRENT TOPICS IN MEDICINAL CHEMISTRY; http://hdl.handle.net/2434/632603Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85069274320
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9دورية أكاديمية
المؤلفون: Gelain, Arianna, Mori, Matteo, Meneghetti, Fiorella, Porta, Federica, Basile, Livia, Marverti, Gaetano, Asai, Akira, Hyeraci, Mariafrancesca, García-Argáez, Aída Nelly, Via, Lisa Dalla, Guccione, Salvatore, Villa, Stefania
المساهمون: A. Gelain, M. Mori, F. Meneghetti, F. Porta, L. Basile, G. Marverti, A. Asai, M. Hyeraci, A.N. García-Argáez, L.D. Via, S. Guccione, S. Villa
مصطلحات موضوعية: Cytotoxicity, Docking studie, HCT-116, HeLa, Oxadiazole, Topoisomerase I, Oncology, Cancer Research, Settore CHIM/08 - Chimica Farmaceutica
العلاقة: info:eu-repo/semantics/altIdentifier/wos/WOS:000454413400016; volume:39; issue:1; firstpage:135; lastpage:144; numberofpages:10; journal:ANTICANCER RESEARCH; http://hdl.handle.net/2434/632615Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85059228102
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10دورية أكاديمية
المؤلفون: Ehrsam, Daniel, Porta, Fabiola, Mori, Matteo, Schwabedissen, Henriette E Meyer Zu, Dalla Via, Lisa, Garcia-Argaez, Aìda Nelly, Basile, Livia, Meneghetti, Fiorella, Villa, Stefania, Gelain, Arianna
المساهمون: D. Ehrsam, F. Porta, M. Mori, H.E.M.Z. Schwabedissen, L. Dalla Via, A.N. Garcia-Argaez, L. Basile, F. Meneghetti, S. Villa, A. Gelain
مصطلحات موضوعية: Furazane, HCT-116, HeLa, MCF-7, MDA-MB 468, cytotoxicity, topoisomerase II, Settore CHIM/08 - Chimica Farmaceutica
العلاقة: info:eu-repo/semantics/altIdentifier/pmid/31262869; info:eu-repo/semantics/altIdentifier/wos/WOS:000482700300021; volume:39; issue:7; firstpage:3453; lastpage:3461; numberofpages:9; journal:ANTICANCER RESEARCH; http://hdl.handle.net/2434/653492Test; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85068252611