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1
المؤلفون: Edward C. Hulme
المصدر: Trends in Pharmacological Sciences. 34:67-84
مصطلحات موضوعية: Models, Molecular, Pharmacology, Agonist, Receptor, Muscarinic M2, Protein Conformation, G protein, Stereochemistry, medicine.drug_class, Receptor, Muscarinic M1, Adrenergic beta-Agonists, Biology, Crystallography, X-Ray, Toxicology, Receptors, G-Protein-Coupled, Cell biology, Structure-Activity Relationship, Protein structure, Receptors, Adrenergic, beta, Muscarinic acetylcholine receptor, medicine, Humans, Signal transduction, Receptor, Ternary complex, G protein-coupled receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0363fc1c9dc4a6bc6b0506a8b49d8906Test
https://doi.org/10.1016/j.tips.2012.11.002Test -
2
المؤلفون: Edward C. Hulme, José W. Saldanha, Robert G. Kaye, Zhi-Liang Lu
المصدر: Molecular Pharmacology. 79:701-709
مصطلحات موضوعية: G protein, Stereochemistry, Protein Structure, Secondary, GTP-binding protein regulators, GTP-Binding Proteins, Chlorocebus aethiops, Muscarinic acetylcholine receptor M5, Animals, 5-HT5A receptor, Binding site, Pharmacology, G protein-coupled receptor kinase, Alanine, Binding Sites, Dose-Response Relationship, Drug, biology, Receptor, Muscarinic M1, Articles, Transmembrane protein, Protein Structure, Tertiary, Rats, Mutagenesis, COS Cells, biology.protein, Biophysics, Molecular Medicine, Protein G
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4a79e654696299e47ed8599a733095f1Test
https://doi.org/10.1124/mol.110.070177Test -
3
المؤلفون: Edward C. Hulme, Mike Trevethick
المصدر: British Journal of Pharmacology. 161:1219-1237
مصطلحات موضوعية: Pharmacology, Dissociation constant, Computational chemistry, Chemistry, Stereochemistry, Drug discovery, Ligand binding assay, Allosteric regulation, Radioligand, Plasma protein binding, Ligand (biochemistry), Radioligand Assay
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::5da64be8f169d31d4ce43c17b4a201b7Test
https://doi.org/10.1111/j.1476-5381.2009.00604.xTest -
4
المؤلفون: Zhi-Liang Lu, M.S. Bee, José W. Saldanha, Edward C. Hulme
المصدر: Biochemical Society Transactions. 31:29-34
مصطلحات موضوعية: Models, Molecular, Agonist, Protein Conformation, medicine.drug_class, Stereochemistry, Scopolamine, Ligands, Biochemistry, Muscarinic acetylcholine receptor M5, Muscarinic acetylcholine receptor, medicine, Animals, Point Mutation, Homology modeling, Binding site, Receptor, Binding Sites, biology, Chemistry, Receptor, Muscarinic M1, Hydrogen Bonding, Receptors, Muscarinic, Acetylcholine, Protein Structure, Tertiary, Mutagenesis, Rhodopsin, biology.protein, Cattle, Protein Binding, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bacbc5f0164a1b9d253f257d1215638dTest
https://doi.org/10.1042/bst0310029Test -
5
المؤلفون: José W. Saldanha, Zhi-Liang Lu, Edward C. Hulme
المصدر: Trends in Pharmacological Sciences. 23:140-146
مصطلحات موضوعية: Rhodopsin, Protein Conformation, G protein, Stereochemistry, Receptors, Cell Surface, Plasma protein binding, Crystallography, X-Ray, Ligands, Toxicology, Receptors, G-Protein-Coupled, Protein structure, GTP-Binding Proteins, Muscarinic acetylcholine receptor, Humans, Receptor, G protein-coupled receptor, Pharmacology, Binding Sites, biology, Chemistry, Structural biology, Mutagenesis, Site-Directed, biology.protein, Biophysics, Protein Binding
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b3762fdb3cb7ff23aed2cebe27199337Test
https://doi.org/10.1016/s0165-6147Test(00)01973-8 -
6
المؤلفون: Carol A. M. Curtis, M. Bee, Edward C. Hulme, Z-L. Lu, José W. Saldanha
المصدر: Life Sciences. 68:2495-2500
مصطلحات موضوعية: Rhodopsin, Protein Conformation, Ligands, General Biochemistry, Genetics and Molecular Biology, GTP-Binding Proteins, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M5, medicine, Animals, General Pharmacology, Toxicology and Pharmaceutics, Acetylcholine receptor, Binding Sites, biology, Chemistry, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, General Medicine, Muscarinic acetylcholine receptor M1, Receptors, Muscarinic, COS Cells, Mutagenesis, Site-Directed, biology.protein, Biophysics, Acetylcholine, Protein Binding, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::23559586a4fc2221f14b8cfe193849a5Test
https://doi.org/10.1016/s0024-3205Test(01)01044-x -
7
المؤلفون: Edward C. Hulme, Zhi-Liang Lu
المصدر: Journal of Biological Chemistry. 275:5682-5686
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Stereochemistry, Receptors, Cell Surface, Muscarinic Antagonists, Ligands, Phosphatidylinositols, Transfection, Polymerase Chain Reaction, Biochemistry, Protein Structure, Secondary, Protein structure, Animals, Histidine, Binding site, Receptor, Molecular Biology, Alanine, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Chemistry, Membrane Proteins, Cell Biology, Receptors, Muscarinic, Acetylcholine, Transmembrane protein, Amino acid, Kinetics, Zinc, Transmembrane domain, COS Cells, Mutagenesis, Site-Directed
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a6103ca05742881feb99f41623836d03Test
https://doi.org/10.1074/jbc.275.8.5682Test -
8
المؤلفون: Stuart D. C. Ward, Carol A. M. Curtis, Edward C. Hulme
المصدر: Molecular Pharmacology. 56:1031-1041
مصطلحات موضوعية: Atropine, Stereochemistry, Receptor expression, Muscarinic Antagonists, Muscarinic Agonists, Ligands, Phosphatidylinositols, Binding, Competitive, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M5, Animals, Receptor, Acetylcholine receptor, Pharmacology, Alanine, Chemistry, Oxotremorine, Receptor, Muscarinic M1, Pilocarpine, N-Methylscopolamine, Alanine scanning, Immunohistochemistry, Receptors, Muscarinic, Acetylcholine, Protein Structure, Tertiary, Rats, Quinuclidinyl Benzilate, Transmembrane domain, COS Cells, Mutagenesis, Site-Directed, Tyrosine, Molecular Medicine, Binding domain
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa102ce82d80efac82af0f9d2162fbafTest
https://doi.org/10.1124/mol.56.5.1031Test -
9
المصدر: European Journal of Pharmacology. 375:247-260
مصطلحات موضوعية: Pharmacology, Binding Sites, Stereochemistry, Cell Membrane, Molecular Conformation, Biology, Receptors, Muscarinic, Transmembrane protein, Cell membrane, Transmembrane domain, medicine.anatomical_structure, GTP-binding protein regulators, GTP-Binding Proteins, Cell surface receptor, Mutagenesis, Site-Directed, medicine, Biophysics, Receptors, Cholinergic, Signal transduction, Receptor, Acetylcholine receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::98a394a7487c7419f4766bf62b986debTest
https://doi.org/10.1016/s0014-2999Test(99)00297-6 -
10
المؤلفون: Edward C. Hulme, Zhi-Liang Lu
المصدر: Journal of Biological Chemistry. 274:7309-7315
مصطلحات موضوعية: Stereochemistry, Chemistry, Mutagenesis, Pilocarpine, Cell Biology, Muscarinic Agonists, Tritium, Receptors, Muscarinic, Biochemistry, Acetylcholine, Protein Structure, Secondary, Transmembrane domain, COS Cells, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M5, Helix, Animals, Guanosine Triphosphate, Receptor, Molecular Biology, Protein secondary structure, Signal Transduction, Acetylcholine receptor
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::127866e0cd1b98638ddd8182ef62fc97Test
https://doi.org/10.1074/jbc.274.11.7309Test