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1دورية أكاديمية
المؤلفون: Xiaolei Ma, Barbara Leon, Elizabeth Ornelas, Dustin Dovala, Laura Tandeske, Catherine Luu, Gwynn Pardee, Stephania Widger, Jonathan M. Solomon, Rohan E. J. Beckwith, Heinz Moser, Matthew C. Clifton, Charles A. Wartchow
المصدر: Scientific Reports, Vol 13, Iss 1, Pp 1-8 (2023)
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2045-2322Test
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2دورية أكاديمية
المؤلفون: Ala M. Shaqra, Sarah N. Zvornicanin, Qiu Yu J. Huang, Gordon J. Lockbaum, Mark Knapp, Laura Tandeske, David T. Bakan, Julia Flynn, Daniel N. A. Bolon, Stephanie Moquin, Dustin Dovala, Nese Kurt Yilmaz, Celia A. Schiffer
المصدر: Nature Communications, Vol 13, Iss 1, Pp 1-11 (2022)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2041-1723Test
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3دورية أكاديمية
المؤلفون: Ethan S. Toriki, James W. Papatzimas, Kaila Nishikawa, Dustin Dovala, Andreas O. Frank, Matthew J. Hesse, Daniela Dankova, Jae-Geun Song, Megan Bruce-Smythe, Heidi Struble, Francisco J. Garcia, Scott M. Brittain, Andrew C. Kile, Lynn M. McGregor, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura
المصدر: ACS Central Science, Vol 9, Iss 8, Pp 1702-1702 (2023)
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2374-7951Test
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4دورية أكاديميةComprehensive fitness landscape of SARS-CoV-2 Mpro reveals insights into viral resistance mechanisms
المؤلفون: Julia M Flynn, Neha Samant, Gily Schneider-Nachum, David T Barkan, Nese Kurt Yilmaz, Celia A Schiffer, Stephanie A Moquin, Dustin Dovala, Daniel NA Bolon
المصدر: eLife, Vol 11 (2022)
مصطلحات موضوعية: Mpro, SARS-CoV-2, deep mutational scanning, main protease, Medicine, Science, Biology (General), QH301-705.5
وصف الملف: electronic resource
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5دورية أكاديمية
المؤلفون: Sarah N. Zvornicanin, Ala M. Shaqra, Qiuyu J. Huang, Elizabeth Ornelas, Mallika Moghe, Mark Knapp, Stephanie Moquin, Dustin Dovala, Celia A. Schiffer, Nese Kurt Yilmaz
المصدر: Viruses, Vol 15, Iss 3, p 781 (2023)
مصطلحات موضوعية: coronaviruses, main protease, GC376, crystal structure, lufotrelvir, HKU15, Microbiology, QR1-502
وصف الملف: electronic resource
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6دورية أكاديمية
المؤلفون: Julia M. Flynn, Sarah N. Zvornicanin, Tenzin Tsepal, Ala M. Shaqra, Nese Kurt Yilmaz, Weiping Jia, Stephanie Moquin, Dustin Dovala, Celia A. Schiffer, Daniel N. A. Bolon
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Microbiology, Genetics, Pharmacology, Evolutionary Biology, Cancer, Mental Health, Hematology, Infectious Diseases, Virology, Computational Biology, Chemical Sciences not elsewhere classified, rapidly evolving diseases, mutational scanning approach, grown viruses selected, future surveillance efforts, reduced apparent binding, observed 3 times, affect enzyme function, possible individual mutations, hyperactive mutations occurred, pro sup, dynamics impacting activity, cause drug resistance, nirmatrelvir binding mutations, hyperactive mutations contribute, cov ‑ 2, hyperactive mutations
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7دورية أكاديمية
المؤلفون: Angel Gonzalez-Valero (14241129), Audrey G. Reeves (14099493), Annika C. S. Page (5697644), Patrick J. Moon (1784497), Edward Miller (4268530), Katia Coulonval (416512), Steven W. M. Crossley (14241132), Xiao Xie (133080), Dan He (145755), Patricia Z. Musacchio (14241135), Alec H. Christian (1810894), Jeffrey M. McKenna (1311780), Richard A. Lewis (535635), Eric Fang (3909934), Dustin Dovala (5398325), Yipin Lu (1693645), Lynn M. McGregor (1273941), Markus Schirle (1433161), John A. Tallarico (308350), Pierre P. Roger (11845427), F. Dean Toste (1311783), Christopher J. Chang (151940)
مصطلحات موضوعية: Biophysics, Biochemistry, Medicine, Cell Biology, Genetics, Molecular Biology, Pharmacology, Cancer, Environmental Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, stereochemically rich substituents, breast cancer cells, bonding interactions stabilizing, activated chemical tagging, based protein profiling, based oxaziridine platform, dependent kinase 4, activating t172 site, selective methionine modification, allosteric m169 site, developing covalent ligands, m169 site, t172 phosphorylation, purified protein, generalizable platform, covalent modifier, m169 oxidation, dependent manner, dependent inhibition
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8
المؤلفون: Ethan S. Toriki, James W. Papatzimas, Kaila Nishikawa, Dustin Dovala, Andreas O. Frank, Matthew J. Hesse, Daniela Dankova, Jae-Geun Song, Megan Bruce-Smythe, Heidi Struble, Francisco J. Garcia, Scott M. Brittain, Andrew C. Kile, Lynn M. McGregor, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Daniel K. Nomura
المصدر: ACS Central Science. 9:915-926
مصطلحات موضوعية: General Chemical Engineering, General Chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::8c2b9836c00807bb6ad517e9fb4b667bTest
https://doi.org/10.1021/acscentsci.2c01317Test -
9دورية أكاديمية
المؤلفون: Scott B. Biering (10974637), Erik Van Dis (10090835), Eddie Wehri (10974640), Livia H. Yamashiro (10974643), Xammy Nguyenla (10974646), Claire Dugast-Darzacq (6294668), Thomas G. W. Graham (10090826), Julien R. Stroumza (10974649), Guillaume R. Golovkine (10974652), Allison W. Roberts (10974655), Daniel M. Fines (10974658), Jessica N. Spradlin (9029189), Carl C. Ward (1310889), Teena Bajaj (6828443), Dustin Dovala (5398325), Ursula Schulze-Gamen (10974661), Ruchika Bajaj (1431883), Douglas M. Fox (1289136), Melanie Ott (26926), Niren Murthy (1320648), Daniel K. Nomura (198023), Julia Schaletzky (4923427), Sarah A. Stanley (525257)
مصطلحات موضوعية: Biochemistry, Medicine, Pharmacology, Biotechnology, Immunology, Cancer, Infectious Diseases, Virology, Environmental Sciences not elsewhere classified, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, Information Systems not elsewhere classified, combination therapies, 13 compounds, epithelial cells, syndrome coronavirus 2, COVID -19 pandemic, SARS-CoV -2, FDA, B 02 exhibits synergy, SARS-CoV -2 replication, coronavirus disease 2019, anti-inflammatory activity, compound screening strategy, host pathways, Bioactive Compounds, drug repurposing screens, health threat, Antiviral Activity, combination therapy
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10
المؤلفون: Angel Gonzalez-Valero, Audrey G. Reeves, Annika C. S. Page, Patrick J. Moon, Edward Miller, Katia Coulonval, Steven W. M. Crossley, Xiao Xie, Dan He, Patricia Z. Musacchio, Alec H. Christian, Jeffrey M. McKenna, Richard A. Lewis, Eric Fang, Dustin Dovala, Yipin Lu, Lynn M. McGregor, Markus Schirle, John A. Tallarico, Pierre P. Roger, F. Dean Toste, Christopher J. Chang
المصدر: J Am Chem Soc
مصطلحات موضوعية: Colloid and Surface Chemistry, General Chemistry, Biochemistry, Article, Catalysis
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58682786d527195267ba39692a00c91bTest
https://doi.org/10.1021/jacs.2c04039Test