نتائج البحث - "Daniel da Costa Pereira"

المصدر: ACS Chemical Neuroscience, 14(4), 645-656. American Chemical Society
Rahman, S N, McNaught-Flores, D A, Huppelschoten, Y, da Costa Pereira, D, Christopoulos, A, Leurs, R & Langmead, C J 2023, ' Structural and Molecular Determinants for Isoform Bias at Human Histamine H 3 Receptor Isoforms ', ACS Chemical Neuroscience, vol. 14, no. 4, pp. 645-656 . https://doi.org/10.1021/acschemneuro.2c00425Test

مصطلحات موضوعية: Physiology, Cognitive Neuroscience, G protein-coupled receptor (GPCR), Cell Biology, General Medicine, Biochemistry, histamine H receptor (hHR), SDG 3 - Good Health and Well-being, neuromodulation, isoform bias, biased signaling, structure−activity relationship (SAR)

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::718f465c1b7d96c399b53e24acad288aTest
https://research.vu.nl/en/publications/c685e773-f7c9-4902-a64c-18c3df4fd827Test

6

SAR exploration of the non-imidazole histamine H

المؤلفون: Gábor, Wágner, Tamara A M, Mocking, Xiaoyuan, Ma, Inna, Slynko, Daniel, Da Costa Pereira, Robin, Breeuwer, Niek J N, Rood, Cas, van der Horst, Henry F, Vischer, Chris, de Graaf, Iwan J P, de Esch, Maikel, Wijtmans, Rob, Leurs

المصدر: Archiv der PharmazieREFERENCES. 356(1)

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::0393ef5c5a5fc9c67738bd435cb1c7c9Test
https://pubmed.ncbi.nlm.nih.gov/36310109Test

7

Fragment Screening Yields a Small-Molecule Stabilizer of 14-3-3 Dimers That Modulates Client Protein Interactions

المؤلفون: Hendrik J. Brink, Rick Riemens, Stephanie Thee, Berend Beishuizen, Daniel da Costa Pereira, Maikel Wijtmans, Iwan de Esch, Martine J. Smit, Albertus H. de Boer

المساهمون: Medicinal chemistry, Chemistry and Pharmaceutical Sciences, AIMMS, Molecular and Computational Toxicology

المصدر: ChemBioChem, 23(17):e202200178, 1-11. Wiley-VCH Verlag
Brink, H J, Riemens, R, Thee, S, Beishuizen, B, da Costa Pereira, D, Wijtmans, M, de Esch, I, Smit, M J & de Boer, A H 2022, ' Fragment Screening Yields a Small-Molecule Stabilizer of 14-3-3 Dimers That Modulates Client Protein Interactions ', ChemBioChem, vol. 23, no. 17, e202200178, pp. 1-11 . https://doi.org/10.1002/cbic.202200178Test

مصطلحات موضوعية: Organic Chemistry, Drug Evaluation, Preclinical, protein-protein interactions, Biochemistry, drug discovery, stabilizers, 14-3-3 Proteins, SDG 3 - Good Health and Well-being, estrogen receptor alpha, fragments, Molecular Medicine, Humans, Molecular Biology, Protein Binding

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::755cf103a39c32e583e10d0070ba7b34Test
https://research.vu.nl/en/publications/9cab963a-1956-4659-8b0e-c71ac894a98bTest

8

Capturing time-dependent activation of genes and stress-response pathways using transcriptomics in iPSC-derived renal proximal tubule cells

المؤلفون: Paul Jennings, Giada Carta, Pranika Singh, Daniel da Costa Pereira, Anita Feher, Andras Dinnyes, Thomas E. Exner, Anja Wilmes

المساهمون: Molecular and Computational Toxicology, AIMMS

المصدر: Jennings, P, Jennings, P, Singh, P, da Costa Pereira, D, Feher, A, Dinnyes, A, Exner, T E & Wilmes, A 2022, ' Capturing time-dependent activation of genes and stress-response pathways using transcriptomics in iPSC-derived renal proximal tubule cells ', Cell biology and toxicology . https://doi.org/10.1007/s10565-022-09783-5Test
Cell biology and toxicology. Springer Netherlands

مصطلحات موضوعية: Health, Toxicology and Mutagenesis, Cell Biology, Toxicology

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7626ff9d6b35df57d0acbec77d2cc02aTest
https://pubmed.ncbi.nlm.nih.gov/36586010Test

9

4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H3 Receptor Agonists with in Vivo Central Nervous System Activity

المؤلفون: Henry F. Vischer, Bruna Silva-Marques, Gniewomir Latacz, Gábor Wágner, Tamara A. M. Mocking, Daniel Da Costa Pereira, Maikel Wijtmans, Marta Arimont, Christina Karatzidou, Rob Leurs, Iwan J. P. de Esch, Katarzyna Kieć-Kononowicz, Barbara Rani, Gustavo Provensi

المساهمون: Theoretical Chemistry, AIMMS, Medicinal chemistry, Molecular and Computational Toxicology, Chemistry and Pharmaceutical Sciences

المصدر: Journal of Medicinal Chemistry, 62(23), 10848-10866. American Chemical Society
Wágner, G, Mocking, T A M, Arimont, M, Provensi, G, Rani, B, Silva-Marques, B, Latacz, G, Da Costa Pereira, D, Karatzidou, C, Vischer, H F, Wijtmans, M, Kieć-Kononowicz, K, De Esch, I J P & Leurs, R 2019, ' 4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H 3 Receptor Agonists with in Vivo Central Nervous System Activity ', Journal of Medicinal Chemistry, vol. 62, no. 23, pp. 10848-10866 . https://doi.org/10.1021/acs.jmedchem.9b01462Test

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::37d0b6fe13ca4e18f1a527fef8942b14Test
https://research.vu.nl/en/publications/f56090ec-0d06-41e2-bc72-bb43cd430fd1Test

10

4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H

المؤلفون: Gábor, Wágner, Tamara A M, Mocking, Marta, Arimont, Gustavo, Provensi, Barbara, Rani, Bruna, Silva-Marques, Gniewomir, Latacz, Daniel, Da Costa Pereira, Christina, Karatzidou, Henry F, Vischer, Maikel, Wijtmans, Katarzyna, Kieć-Kononowicz, Iwan J P, de Esch, Rob, Leurs

المصدر: Journal of Medicinal Chemistry

مصطلحات موضوعية: Behavior, Animal, Molecular Structure, Protein Conformation, Article, Histamine Agonists, Molecular Docking Simulation, Mice, HEK293 Cells, Memory, Animals, Humans, Amines, Social Behavior, Protein Binding

الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::3aac0e5e7c872e9df9b0086c3e3934b4Test
https://pubmed.ncbi.nlm.nih.gov/31675226Test

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