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المؤلفون: Karen Collins, Donald Wojciechowicz, Judy Lucas, Nancy Torres, Jeremy I. Levin, Yongbo Hu, Cilien Hanna, Dan M. Berger, Edward J. Salaski, Eileen Frommer, Minu Dutia, Wang Xiaolun, Dennis Powell
المصدر: Journal of Medicinal Chemistry. 53:7874-7878
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Indazoles, Transplantation, Heterologous, Mutant, Antineoplastic Agents, Pharmacology, Mice, Structure-Activity Relationship, Pyrimidine analogue, chemistry.chemical_compound, Pharmacokinetics, In vivo, Cell Line, Tumor, Drug Discovery, Animals, Humans, Chemistry, Kinase, Bridged Bicyclo Compounds, Heterocyclic, humanities, Pyrimidines, Biochemistry, Mutation, Pyrazoles, Molecular Medicine, Drug Screening Assays, Antitumor, Selectivity, Lead compound, Neoplasm Transplantation
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f5cfb7f80cde520202634116ccfc59adTest
https://doi.org/10.1021/jm1007566Test -
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المؤلفون: Cilien Hanna, Clark Eid, Erick Honores, Weiguo Zhang, Leif M. Laakso, Ayako Yamashita, Bernard Dean Johnson, Leonard A. McDonald, Zhong Li, Weidong Ding, Dennis Powell, Jeremy I. Levin, Girija Krishnamurthy, Keiko Tabei, Jaechul Shim, Edward J. Salaski, Shabana Insaf, Lourdes Toral-Barza, Ker Yu, Tarek S. Mansour
المصدر: Journal of Medicinal Chemistry. 52:2181-2184
مصطلحات موضوعية: Alkylation, Stereochemistry, Antineoplastic Agents, Lactones, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Humans, Structure–activity relationship, Cysteine, Protein kinase B, Cell Proliferation, Pyrans, chemistry.chemical_classification, biology, Kinase, Stereoisomerism, Oncogene Protein v-akt, Enzyme, chemistry, Mechanism of action, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, medicine.symptom, Signal transduction, Biomarkers, Naphthoquinones
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5485ad3ec1278f1fbce482a2a467aff3Test
https://doi.org/10.1021/jm900075gTest -
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المؤلفون: Ayako Yamashita, Cilien Hanna, Edward J. Salaski, Jaechul Shim, Dahui Zhou, Emily B. Norton, Tarek S. Mansour
المصدر: ChemInform. 37
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Organic Chemistry, Potassium tert-butoxide, Polymer chemistry, Organic chemistry, General Medicine, Ring (chemistry), Medicinal chemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::48cc1b2b66f0c2e39d5600be43033defTest
https://doi.org/10.1002/chin.200634136Test