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1دورية أكاديمية
المؤلفون: Siqueira-Neto, Jair, Wicht, Kathryn, Chibale, Kelly, Burrows, Jeremy, Fidock, David, Winzeler, Elizabeth
المصدر: Nature Reviews Drug Discovery. 22(10)
مصطلحات موضوعية: Animals, Female, Humans, Antimalarials, Plasmodium, Drug Resistance, Drug Discovery
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/21j7z4d2Test
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2دورية أكاديمية
المؤلفون: Arendse, Lauren, Murithi, James, Qahash, Tarrick, Pasaje, Charisse, Godoy, Luiz, Dey, Sumanta, Gibhard, Liezl, Ghidelli-Disse, Sonja, Drewes, Gerard, Bantscheff, Marcus, Lafuente-Monasterio, Maria, Fienberg, Stephen, Wambua, Lynn, Gachuhi, Samuel, Coertzen, Dina, van der Watt, Mariëtte, Reader, Janette, Aswat, Ayesha, Erlank, Erica, Venter, Nelius, Mittal, Nimisha, Luth, Madeline, Ottilie, Sabine, Koekemoer, Lizette, Birkholtz, Lyn-Marie, Niles, Jacquin, Llinás, Manuel, Fidock, David, Chibale, Kelly, Winzeler, Elizabeth
المصدر: Science Translational Medicine. 14(667)
مصطلحات موضوعية: Animals, Humans, Antimalarials, Plasmodium falciparum, MTOR Inhibitors, 1-Phosphatidylinositol 4-Kinase, Guanosine Monophosphate, Life Cycle Stages, TOR Serine-Threonine Kinases, Plasmodium, Sirolimus, Mammals
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/6kx4p874Test
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3دورية أكاديمية
المؤلفون: Murithi, James, Deni, Ioanna, Pasaje, Charisse, Okombo, John, Bridgford, Jessica, Gnädig, Nina, Edwards, Rachel, Yeo, Tomas, Mok, Sachel, Burkhard, Anna, Coburn-Flynn, Olivia, Istvan, Eva, Sakata-Kato, Tomoyo, Gomez-Lorenzo, Maria, Cowell, Annie, Wicht, Kathryn, Le Manach, Claire, Kalantarov, Gavreel, Dey, Sumanta, Duffey, Maëlle, Laleu, Benoît, Lukens, Amanda, Ottilie, Sabine, Vanaerschot, Manu, Trakht, Ilya, Gamo, Francisco-Javier, Wirth, Dyann, Goldberg, Daniel, Odom John, Audrey, Chibale, Kelly, Winzeler, Elizabeth, Niles, Jacquin, Fidock, David
المصدر: Cell Chemical Biology. 29(5)
مصطلحات موضوعية: ABCI3, CRISPR/Cas9, Plasmodium falciparum malaria, biphasic dose-response curves, cellular accumulation assays, conditional knockdowns, copy-number variations, heme fractionation, pfcrt, ATP-Binding Cassette Transporters, Animals, Antimalarials, Folic Acid Antagonists, Heme, Malaria, Falciparum, Membrane Transport Proteins, Parasites, Plasmodium falciparum, Protozoan Proteins, Quinolines
وصف الملف: application/pdf
الوصول الحر: https://escholarship.org/uc/item/4277b0xkTest
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4دورية أكاديمية
المؤلفون: Dziwornu, Godwin Akpeko, Seanego, Donald, Fienberg, Stephen, Clements, Monica, Ferreira, Jasmin, Sypu, Venkata S., Samanta, Sauvik, Bhana, Ashlyn D., Korkor, Constance M., Garnie, Larnelle F., Teixeira, Nicole, Wicht, Kathryn J., Taylor, Dale, Olckers, Ronald, Njoroge, Mathew, Gibhard, Liezl, Salomane, Nicolaas, Wittlin, Sergio, Mahato, Rohit, Chakraborty, Arnish, Sevilleno, Nicole, Coyle, Rachael, Lee, Marcus C. S., Godoy, Luiz C., Pasaje, Charisse Flerida, Niles, Jacquin C., Reader, Janette, van der Watt, Mariette, Birkholtz, Lyn-Marié, Bolscher, Judith M., de Bruijni, Marloes H. C., Coulson, Lauren B., Basarab, Gregory S., Ghorpade, Sandeep R., Chibale, Kelly
المصدر: Journal of Medicinal Chemistry ; ISSN 0022-2623 1520-4804
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5دورية أكاديمية
المؤلفون: Hlozek, Jason, Chibale, Kelly, Woodland, John G.
المصدر: ACS Medicinal Chemistry Letters ; ISSN 1948-5875 1948-5875
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6دورية أكاديمية
المؤلفون: Mambwe, Dickson, Coertzen, Dina, Leshabane, Meta, Mulubwa, Mwila, Njoroge, Mathew, Gibhard, Liezl, Girling, Gareth, Wicht, Kathryn J., Lee, Marcus C. S., Wittlin, Sergio, Moreira, Diogo Rodrigo Magalhães, Birkholtz, Lyn-Marie, Chibale, Kelly
المساهمون: Funda????o Oswaldo Cruz, Minist??rio da Ci??ncia, Tecnologia e Inova????o, University of Cape Town, National Research Foundation, South African Medical Research Council
المصدر: ACS Medicinal Chemistry Letters ; volume 15, issue 4, page 463-469 ; ISSN 1948-5875 1948-5875
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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7دورية أكاديمية
المؤلفون: Byl, Jo Ann W., Mueller, Rudolf, Bax, Ben, Basarab, Gregory S., Chibale, Kelly, Osheroff, Neil
وصف الملف: application/pdf
العلاقة: https://orca.cardiff.ac.uk/id/eprint/157504/1/acsinfecdis.3c00012.pdfTest; Byl, Jo Ann W., Mueller, Rudolf, Bax, Ben https://orca.cardiff.ac.uk/view/cardiffauthors/A2393082O.htmlTest orcid:0000-0003-1940-3785 orcid:0000-0003-1940-3785, Basarab, Gregory S., Chibale, Kelly and Osheroff, Neil 2023. A series of Spiropyrimidinetriones that enhances DNA cleavage mediated by Mycobacterium tuberculosis gyrase. ACS Infectious Diseases 9 (3) , pp. 706-715. 10.1021/acsinfecdis.3c00012 https://doi.org/10.1021/acsinfecdis.3c00012Test file https://orca.cardiff.ac.uk/id/eprint/157504/1/acsinfecdis.3c00012.pdfTest
الإتاحة: https://doi.org/10.1021/acsinfecdis.3c00012Test
https://orca.cardiff.ac.uk/id/eprint/157504Test/
https://orca.cardiff.ac.uk/id/eprint/157504/1/acsinfecdis.3c00012.pdfTest -
8دورية أكاديمية
المؤلفون: Turon, Gemma, Hlozek, Jason, Woodland, John G., Kumar, Ankur, Chibale, Kelly, Duran-Frigola, Miquel
المساهمون: Merck KGaA, Harry Crossley Foundation
المصدر: Nature Communications ; volume 14, issue 1 ; ISSN 2041-1723
مصطلحات موضوعية: General Physics and Astronomy, General Biochemistry, Genetics and Molecular Biology, General Chemistry, Multidisciplinary
الإتاحة: https://doi.org/10.1038/s41467-023-41512-2Test
https://www.nature.com/articles/s41467-023-41512-2.pdfTest
https://www.nature.com/articles/s41467-023-41512-2Test -
9دورية أكاديمية
المؤلفون: Cabrera, Diego González, Smith, Dennis A., Basarab, Gregory S., Duffy, James, Spangenberg, Thomas, Chibale, Kelly
المساهمون: Merck KGaA, Medicines for Malaria Venture
المصدر: ACS Medicinal Chemistry Letters ; volume 14, issue 7, page 875-878 ; ISSN 1948-5875 1948-5875
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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10دورية أكاديمية
المساهمون: University of Cape Town, National Research Foundation, South African Medical Research Council
المصدر: ACS Infectious Diseases ; volume 9, issue 4, page 928-942 ; ISSN 2373-8227 2373-8227
مصطلحات موضوعية: Infectious Diseases