التفاصيل البيبلوغرافية
العنوان: |
Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors |
المؤلفون: |
Calvo, Veronica, Surguladze, David, Li, An-Hu, Surman, Matthew D., Malibhatla, Srikanth, Bandaru, Madhavarao, Jonnalagadda, Suresh Krishna, Adarasandi, Ravi, Velmala, Madhusudhan, Singireddi, Durga Rama Prasad, Velpuri, Mahendar, Nareddy, Bhaskar Reddy, Sastry, Visweswara, Mandati, Chiranjeevi, Guguloth, Rambabu, Siddiqui, Shapi, Patil, Basanagoud S., Chad, Elena, Wolfley, Jennifer, Gasparek, Jennifer, Feldman, Kirsten, Betzenhauser, Matthew, Wiens, Brent, Koszelak-Rosenblum, Mary, Zhu, Guangyu, Du, Hongwen, Rigby, Alan C., Mulvihill, Mark J. |
المساهمون: |
National Cancer Institute, National Institute of General Medical Sciences, National Institutes of Health, Office of Science, Argonne National Laboratory, U.S. Department of Energy |
المصدر: |
Bioorganic & Medicinal Chemistry Letters ; volume 43, page 128058 ; ISSN 0960-894X |
بيانات النشر: |
Elsevier BV |
سنة النشر: |
2021 |
المجموعة: |
ScienceDirect (Elsevier - Open Access Articles via Crossref) |
مصطلحات موضوعية: |
Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Biology, Molecular Medicine, Biochemistry |
نوع الوثيقة: |
article in journal/newspaper |
اللغة: |
English |
DOI: |
10.1016/j.bmcl.2021.128058 |
الإتاحة: |
https://doi.org/10.1016/j.bmcl.2021.128058Test https://api.elsevier.com/content/article/PII:S0960894X21002845?httpAccept=text/xmlTest https://api.elsevier.com/content/article/PII:S0960894X21002845?httpAccept=text/plainTest |
حقوق: |
https://www.elsevier.com/tdm/userlicense/1.0Test/ ; http://creativecommons.org/licenses/by-nc-nd/4.0Test/ |
رقم الانضمام: |
edsbas.CBF46243 |
قاعدة البيانات: |
BASE |