دورية أكاديمية

Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors

التفاصيل البيبلوغرافية
العنوان: Discovery of 2-amino-3-amido-5-aryl-pyridines as highly potent, orally bioavailable, and efficacious PERK kinase inhibitors
المؤلفون: Calvo, Veronica, Surguladze, David, Li, An-Hu, Surman, Matthew D., Malibhatla, Srikanth, Bandaru, Madhavarao, Jonnalagadda, Suresh Krishna, Adarasandi, Ravi, Velmala, Madhusudhan, Singireddi, Durga Rama Prasad, Velpuri, Mahendar, Nareddy, Bhaskar Reddy, Sastry, Visweswara, Mandati, Chiranjeevi, Guguloth, Rambabu, Siddiqui, Shapi, Patil, Basanagoud S., Chad, Elena, Wolfley, Jennifer, Gasparek, Jennifer, Feldman, Kirsten, Betzenhauser, Matthew, Wiens, Brent, Koszelak-Rosenblum, Mary, Zhu, Guangyu, Du, Hongwen, Rigby, Alan C., Mulvihill, Mark J.
المساهمون: National Cancer Institute, National Institute of General Medical Sciences, National Institutes of Health, Office of Science, Argonne National Laboratory, U.S. Department of Energy
المصدر: Bioorganic & Medicinal Chemistry Letters ; volume 43, page 128058 ; ISSN 0960-894X
بيانات النشر: Elsevier BV
سنة النشر: 2021
المجموعة: ScienceDirect (Elsevier - Open Access Articles via Crossref)
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Biology, Molecular Medicine, Biochemistry
نوع الوثيقة: article in journal/newspaper
اللغة: English
DOI: 10.1016/j.bmcl.2021.128058
الإتاحة: https://doi.org/10.1016/j.bmcl.2021.128058Test
https://api.elsevier.com/content/article/PII:S0960894X21002845?httpAccept=text/xmlTest
https://api.elsevier.com/content/article/PII:S0960894X21002845?httpAccept=text/plainTest
حقوق: https://www.elsevier.com/tdm/userlicense/1.0Test/ ; http://creativecommons.org/licenses/by-nc-nd/4.0Test/
رقم الانضمام: edsbas.CBF46243
قاعدة البيانات: BASE