-
1
المؤلفون: Xiaolian Xu, Seong Heon Kim, Qingbei Zeng, Joseph A. Kozlowski, Carolyn DiIanni Carroll, Neng-Yang Shih, Baldwin John J, Wensheng Yu, Yueheng Jiang, Guizhen Dong, Yuefei Shao, Brian F. Mcguinness, Gopinadhan N. Anilkumar, Lisa Guise Zawacki, Doug W. Hobbs, Chung-Her Jenh, James W. Hall, Stuart B. Rosenblum, Bandarpalle B. Shankar, De-Yi Yang
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6982-6986
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, Receptors, CXCR3, Clinical Biochemistry, hERG, Pharmaceutical Science, C-C chemokine receptor type 7, C-C chemokine receptor type 6, CCR5 receptor antagonist, Pharmacology, Biochemistry, Piperazines, Inhibitory Concentration 50, Structure-Activity Relationship, Chemokine receptor, stomatognathic system, Drug Discovery, Animals, Structure–activity relationship, cardiovascular diseases, skin and connective tissue diseases, Molecular Biology, Molecular Structure, biology, Chemistry, Organic Chemistry, Rats, stomatognathic diseases, Pyrazines, biology.protein, Molecular Medicine, Receptor antagonist activity, Protein Binding, CCL21
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4c65b7371750c0100d6b469612e6fd2fTest
https://doi.org/10.1016/j.bmcl.2011.09.120Test -
2
المؤلفون: Cangming Yang, Biji Jacob-Samuel, Doug W. Hobbs, Joseph A. Kozlowski, Lisa Guise Zawacki, Gopinadhan N. Anilkumar, Guizhen Dong, Carolyn DiIanni Carroll, Brian F. Mcguinness, Stuart B. Rosenblum, Chung-Her Jenh, James W. Hall
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:5205-5208
مصطلحات موضوعية: Receptors, CXCR3, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Solid-phase synthesis, Piperidines, Drug Discovery, medicine, Combinatorial Chemistry Techniques, Humans, Molecule, Molecular Biology, Aryl, Organic Chemistry, In vitro, Piperazine, chemistry, Molecular Medicine, Piperidine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6f918421b8905c07f0d3f98fb7d7c2deTest
https://doi.org/10.1016/j.bmcl.2009.07.020Test -
3
المؤلفون: Babu Suresh D, R. Kuvelkar, Yuhua Huang, A.W. Stamford, Qi Zhang, Lili Zhang, P. Gaspari, J. Pan, Wang Lingyan, L. Ozgur, Ge Li, Yusheng Wu, Johannes H. Voigt, Xiao Chen, Kurt W. Saionz, J. Lowrie, Tao Guo, Ulrich Iserloh, N.A. McHugh, D. Tadesse, Le Thuy X H, Matthew E. Kennedy, Doug W. Hobbs, Leonard Favreau, Carolyn DiIanni Carroll, Corey Strickland, Jared N. Cumming, Eric M. Parker
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:3236-3241
مصطلحات موضوعية: Models, Molecular, Imidazolidinone, medicine.drug_class, Stereochemistry, Peptidomimetic, Memapsin-2, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Mice, Transgenic, Carboxamide, Crystallography, X-Ray, Imidazolidines, Biochemistry, Piperazines, Mice, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Aspartic Acid Endopeptidases, Humans, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, Rational design, Disease Models, Animal, Drug Design, β secretase, Molecular Medicine, Amyloid Precursor Protein Secretases, Aspartic Endopeptidases
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6ecdbdfa7bbf11174961bb58e02315b3Test
https://doi.org/10.1016/j.bmcl.2008.04.050Test -
4
المؤلفون: Wong Michael K C, Yueheng Jiang, Qingbei Zeng, Chung-Her Jenh, Stuart B. Rosenblum, De-Yi Yang, Yuefei Shao, Anilkumar G. Nair, Jingqi Duo, Doug W. Hobbs, Brian F. Mcguinness, Joseph A. Kozlowski, Lisa Guise Zawacki, Neng-Yang Shih, Carolyn DiIanni Carroll, Youheng Shu, Seong Heon Kim
المصدر: Bioorganicmedicinal chemistry letters. 24(4)
مصطلحات موضوعية: Receptors, CXCR3, Metabolite, Clinical Biochemistry, hERG, Pharmaceutical Science, CXCR3, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Heterocyclic Compounds, Amide, Drug Discovery, Animals, Humans, Molecular Biology, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Combinatorial chemistry, Amides, Ether-A-Go-Go Potassium Channels, Rats, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::126a3924ad6c61b713b4a73725849822Test
https://pubmed.ncbi.nlm.nih.gov/24486132Test -
5
المؤلفون: Roland E. Dolle, Linda O’Brien, Marc Orlowski, John C. Reader, Cullen L. Cavallaro, Ying Jin, William J. Egan, Wenni Li, Mark Piznik, Joan Guo, Biji Jacob-Samuel, Carolyn DiIanni Carroll, Andrew Laird Roughton, Kevin J. Bowman, Qian Zhao
المصدر: Journal of Combinatorial Chemistry. 2:716-731
مصطلحات موضوعية: Chemistry, media_common.quotation_subject, Sampling (statistics), Fidelity, General Chemistry, Bead, Combinatorial chemistry, Set (abstract data type), Sample size determination, Liquid chromatography–mass spectrometry, visual_art, visual_art.visual_art_medium, Algorithm, media_common
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa969037d0b245d9ac56f01fc0648d54Test
https://doi.org/10.1021/cc000052kTest -
6
المؤلفون: Anna Oksman, Daniel E. Goldberg, Roland E. Dolle, Theodore O. Johnson, Daniel Chelsky, Marc Orlowski, Joan Guo, Carolyn DiIanni Carroll, Ilya Y. Gluzman, Tao Guo, Zhen-Min He, Cullen L. Cavallaro, Hitesh K. Patel, James A. Connelly
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:2315-2320
مصطلحات موضوعية: Plasmodium falciparum, Clinical Biochemistry, Protozoan Proteins, Pharmaceutical Science, Biochemistry, Substrate Specificity, Apicomplexa, Antimalarials, Hemoglobins, Structure-Activity Relationship, chemistry.chemical_compound, Plasmepsin II, Peptide Library, parasitic diseases, Drug Discovery, Statine, Animals, Aspartic Acid Endopeptidases, Humans, Structure–activity relationship, Protease Inhibitors, Amino Acids, Cloning, Molecular, Peptide library, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Organic Chemistry, biology.organism_classification, Recombinant Proteins, Enzyme, Databases as Topic, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Oligopeptides
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd938f8a4ac0e0a6defa4e6293b3b48aTest
https://doi.org/10.1016/s0960-894xTest(98)00419-3 -
7
المؤلفون: Gopinadhan N. Anilkumar, Qingbei Zeng, Brian F. Mcguinness, Chung-Her Jenh, Guizhen Dong, Lisa Guise Zawacki, Inna Schulman, Yueheng Jiang, Seong Heon Kim, Yuefei Shao, Youheng Shu, Wong Michael K C, Doug W. Hobbs, Stuart B. Rosenblum, Neng-Yang Shih, James W. Hall, Carolyn DiIanni Carroll, Wensheng Yu, Joseph A. Kozlowski
المصدر: Bioorganicmedicinal chemistry letters. 21(5)
مصطلحات موضوعية: Receptors, CXCR3, Stereochemistry, medicine.drug_class, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CXCR3, Biochemistry, Piperazines, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, stomatognathic system, Piperidines, immune system diseases, Drug Discovery, medicine, Moiety, Humans, skin and connective tissue diseases, Receptor, Molecular Biology, IC50, Piperazine, Molecular Structure, Organic Chemistry, Antagonist, hemic and immune systems, In vitro, stomatognathic diseases, chemistry, Molecular Medicine, Piperidine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9894b320a60ce2053010ea1122688132Test
https://pubmed.ncbi.nlm.nih.gov/21277198Test -
8
المؤلفون: Carolyn Diianni Carroll, Jiuqiao Zhao, Maria L. Webb, Laura L. Rokosz, Kenneth C. Appell, Tsung Lin, James R Beasley
المصدر: Expert opinion on therapeutic targets. 12(7)
مصطلحات موضوعية: Clinical Biochemistry, Dasatinib, Piperazines, hemic and lymphatic diseases, Drug Discovery, medicine, Bruton's tyrosine kinase, Animals, Humans, Rho-associated protein kinase, Protein Kinase Inhibitors, Pharmacology, Inflammation, Clinical Trials as Topic, ABL, biology, business.industry, Protein-Tyrosine Kinases, Thiazoles, Imatinib mesylate, Pyrimidines, Immune System Diseases, Benzamides, Chronic Disease, biology.protein, Cancer research, Imatinib Mesylate, Molecular Medicine, Janus kinase, business, Tyrosine kinase, Platelet-derived growth factor receptor, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::734e08ffb505766b453b5a79e3a7b829Test
https://pubmed.ncbi.nlm.nih.gov/18554156Test -
9
المؤلفون: Roland E. Dolle, Marc Orlowski, Ilya Y. Gluzman, Giorgio Lauri, Carolyn DiIanni Carroll, Daniel E. Goldberg, Shewei Tao, Theodore O. Johnson
المصدر: Bioorganicmedicinal chemistry letters. 8(22)
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Protozoan Proteins, Pharmaceutical Science, Cathepsin D, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Plasmepsin II, Amide, Drug Discovery, Statine, Structure–activity relationship, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, Amino Acids, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Combinatorial chemistry, Amides, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a36d736b9d159d1b4c7ff0d0754a0cbaTest
https://pubmed.ncbi.nlm.nih.gov/9873703Test -
10
المؤلفون: Carolyn DiIanni Carroll, Marc Orlowski
المصدر: Aspartic Proteinases ISBN: 9781461374527
مصطلحات موضوعية: chemistry.chemical_classification, Cathepsin, Protease, Enzyme, Plasmepsin II, Aspartate protease, chemistry, Biochemistry, medicine.medical_treatment, medicine, High Throughput Assay, Cathepsin D, Peptide sequence
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::b137233f9cc253079654ffdfd6039c69Test
https://doi.org/10.1007/978-1-4615-5373-1_52Test