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المؤلفون: Alice R Eddershaw, Karl Syson, Paul R. J. Davey, Gregory Hamm, Christopher D. Stubbs, Paul Clarkson, Elizabeth Underwood, Lucy V Edwardes
المصدر: Biochemistry. 59:4775-4786
مصطلحات موضوعية: Models, Molecular, Protein-Arginine N-Methyltransferases, Methyltransferase, Arginine, In Vitro Techniques, Biochemistry, Mass Spectrometry, Substrate Specificity, 03 medical and health sciences, Protein structure, Catalytic Domain, Humans, Protein Interaction Domains and Motifs, Amino Acid Sequence, Enzyme Inhibitors, Protein Structure, Quaternary, Ternary complex, Adaptor Proteins, Signal Transducing, 0303 health sciences, Chemistry, Protein arginine methyltransferase 5, 030302 biochemistry & molecular biology, Deuterium Exchange Measurement, Recombinant Proteins, Kinetics, Biophysics, Hydrogen–deuterium exchange, Steady state (chemistry)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e0c63875119c271f482688a035fe6bfcTest
https://doi.org/10.1021/acs.biochem.0c00554Test -
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المؤلفون: Cheryl M. Koh, Christopher D. Stubbs, Puneet Khurana, Gavin W. Collie, Ian L. Dale, Alice R Eddershaw, Joseph Shaw, Fredrik Mauritzson, Tony Cheung, Arjan Snijder, Edward J. Hennessy, Christopher R. Phillips, Louise Barlind, Daniel O'Neill, Ana J. Narvaez
المصدر: ACS Medicinal Chemistry Letters
مصطلحات موضوعية: Letter, cMET, kinase, Mutant, medicine.disease_cause, 01 natural sciences, Biochemistry, Receptor tyrosine kinase, Drug Discovery, medicine, Transferase, X-ray crystallography, Mutation, drug resistance, biology, 010405 organic chemistry, Kinase, Chemistry, Organic Chemistry, small molecule inhibitor, Small molecule, First generation, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Savolitinib, Cancer research, biology.protein
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1db8fce6c00b422a455792c6c6c627faTest
http://europepmc.org/articles/PMC6746082Test