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1دورية أكاديمية
المؤلفون: Claire M. Patterson, Srividya B. Balachander, Iain Grant, Petar Pop-Damkov, Brian Kelly, William McCoull, Jeremy Parker, Michael Giannis, Kathryn J. Hill, Francis D. Gibbons, Edward J. Hennessy, Paul Kemmitt, Alexander R. Harmer, Sonya Gales, Stuart Purbrick, Sean Redmond, Matthew Skinner, Lorraine Graham, J. Paul Secrist, Alwin G. Schuller, Shenghua Wen, Ammar Adam, Corinne Reimer, Justin Cidado, Martin Wild, Eric Gangl, Stephen E. Fawell, Jamal Saeh, Barry R. Davies, David J. Owen, Marianne B. Ashford
المصدر: Communications Biology, Vol 4, Iss 1, Pp 1-14 (2021)
مصطلحات موضوعية: Biology (General), QH301-705.5
وصف الملف: electronic resource
العلاقة: https://doaj.org/toc/2399-3642Test
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المؤلفون: Frederick W, Goldberg, Attilla K T, Ting, David, Beattie, Gillian M, Lamont, Charlene, Fallan, M Raymond V, Finlay, Beth, Williamson, Marianne, Schimpl, Alexander R, Harmer, Oladipupo B, Adeyemi, Pär, Nordell, Anna S, Cronin, Mercedes, Vazquez-Chantada, Derek, Barratt, Antonio, Ramos-Montoya, Elaine B, Cadogan, Barry R, Davies
المصدر: ACS medicinal chemistry letters. 13(8)
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::2661b30d6b91249b7feab29e38d45bb4Test
https://pubmed.ncbi.nlm.nih.gov/35978693Test -
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المؤلفون: Frederick W. Goldberg, Attilla K. T. Ting, David Beattie, Gillian M. Lamont, Charlene Fallan, M. Raymond V. Finlay, Beth Williamson, Marianne Schimpl, Alexander R. Harmer, Oladipupo B. Adeyemi, Pär Nordell, Anna S. Cronin, Mercedes Vazquez-Chantada, Derek Barratt, Antonio Ramos-Montoya, Elaine B. Cadogan, Barry R. Davies
المصدر: ACS Medicinal Chemistry Letters. 13:1295-1301
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::cf9dfca39604357a47354a464d4b09f5Test
https://doi.org/10.1021/acsmedchemlett.2c00172Test -
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المؤلفون: Gregory Hamm, Gareth Maglennon, Beth Williamson, Ruth Macdonald, Ann Doherty, Stewart Jones, Jayne Harris, James Blades, Alexander R. Harmer, Peter Barton, Philip B. Rawlins, Paul Smith, Jon Winter-Holt, Lindsay McMurray, Julia Johansson, Paul Fitzpatrick, William McCoull, Muireann Coen
المصدر: Archives of Toxicology. 96:613-624
مصطلحات موضوعية: Male, Mice, Knockout, c-Mer Tyrosine Kinase, Health, Toxicology and Mutagenesis, Retinal Degeneration, Retinal Pigment Epithelium, General Medicine, Toxicology, Multimodal Imaging, Mass Spectrometry, Cell Line, Rats, Mice, Inbred C57BL, Mice, Phagocytosis, Animals, Humans, Female, Rats, Long-Evans, Tissue Distribution, sense organs, Rats, Wistar, Photoreceptor Cells, Vertebrate
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1c26625750e5c3c3d003dbd985eddb7aTest
https://doi.org/10.1007/s00204-021-03197-8Test -
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المؤلفون: Tarjinder Sahota, Stein Schalkwijk, Alexander R. Harmer, Remy B. Verheijen, Ghada F. Ahmed
المصدر: The AAPS Journal. 23
مصطلحات موضوعية: biology, business.industry, Metabolite, hERG, QTcF Prolongation, Prolongation, Cmax, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, QT interval, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, chemistry, 030220 oncology & carcinogenesis, biology.protein, Medicine, business, IC50, EC50
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::82371156f681427747712f98c2b5a10aTest
https://doi.org/10.1208/s12248-021-00573-1Test -
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المؤلفون: Ammar Adam, David J. Owen, Justin Cidado, Claire Patterson, Matthew Skinner, Stuart Purbrick, Lorraine Graham, Petar Pop-Damkov, Michael Giannis, Srividya B. Balachander, Francis D. Gibbons, William McCoull, Marianne Ashford, Hill Kathryn Jane, Martin Wild, Eric Gangl, Stephen Fawell, Corinne Reimer, Sean Redmond, Paul D. Kemmitt, Barry R. Davies, Jamal Carlos Saeh, Shenghua Wen, J. Paul Secrist, Alwin Schuller, Edward J. Hennessy, Sonya Gales, Iain Grant, Alexander R. Harmer, Jeremy S. Parker, Brian Kelly
المصدر: Communications Biology
Communications Biology, Vol 4, Iss 1, Pp 1-14 (2021)مصطلحات موضوعية: Male, 0301 basic medicine, Drug, Dendrimers, QH301-705.5, media_common.quotation_subject, bcl-X Protein, Medicine (miscellaneous), Drug development, Antineoplastic Agents, Mice, SCID, Pharmacology, Conjugated system, Article, General Biochemistry, Genetics and Molecular Biology, Mice, 03 medical and health sciences, Targeted therapies, Dogs, 0302 clinical medicine, Therapeutic index, Neoplasms, Dendrimer, Tumor Cells, Cultured, Animals, Humans, Medicine, Biology (General), Rats, Wistar, media_common, Haematological cancer, business.industry, Xenograft Model Antitumor Assays, Rats, Mice, Inbred C57BL, Therapeutic Index, 030104 developmental biology, Proto-Oncogene Proteins c-bcl-2, Tolerability, 030220 oncology & carcinogenesis, Drug delivery, Female, General Agricultural and Biological Sciences, business, Conjugate
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f928851dba9fe7a39b683d8c12e8a5dTest
https://doi.org/10.1038/s42003-020-01631-8Test -
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المؤلفون: Stein, Schalkwijk, Tarjinder, Sahota, Remy B, Verheijen, Alexander R, Harmer, Ghada F, Ahmed
المصدر: The AAPS journal. 23(3)
مصطلحات موضوعية: Male, Electrocardiography, Inhibitory Concentration 50, Long QT Syndrome, Double-Blind Method, Heart Rate, Triazines, Pyrazines, Humans, Middle Aged, Models, Biological, Protein Kinase Inhibitors, Healthy Volunteers
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::97390e21db5b7c455ab11ed3ddc84f44Test
https://pubmed.ncbi.nlm.nih.gov/33733338Test -
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المؤلفون: Ross Overman, Evan Barry, Sylvie Guichard, Crystal Brown, Oladipupo Adeyemi, Deborah Lawson, Rhys D.O. Jones, Venkatesh Pilla Reddy, Sabina Cosulich, Jerome T. Mettetal, Haiyun Wang, Teresa Collins, Martin J. Packer, Erica Banks, Stephen Fawell, Lisa Drew, Alexander R. Harmer, Deepa Bhavsar, David Wilson, Jason Grant Kettle, Wenlin Shao, Corinne Reimer, Michael Grondine, Rana Anjum
المصدر: Science translational medicine. 12(541)
مصطلحات موضوعية: Vascular Endothelial Growth Factor A, Receptor, Platelet-Derived Growth Factor alpha, Gastrointestinal Stromal Tumors, Antineoplastic Agents, medicine.disease_cause, chemistry.chemical_compound, Regorafenib, medicine, Animals, Humans, Urea, Pyrroles, Stromal tumor, Naphthyridines, neoplasms, Protein Kinase Inhibitors, Mutation, GiST, business.industry, Sunitinib, Triazines, Imatinib, General Medicine, medicine.disease, digestive system diseases, Rats, Vascular endothelial growth factor A, Proto-Oncogene Proteins c-kit, chemistry, Drug Resistance, Neoplasm, Cancer research, Pyrazoles, Sarcoma, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6fcdee9e22eb865b4d98090dd3ef4933Test
https://pubmed.ncbi.nlm.nih.gov/32350132Test -
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المؤلفون: Christopher Hardy, Matthew Skinner, Teresa Collins, Michal Bista, Kelly Gray, Jerome T. Mettetal, Haiyun Wang, Alexander R. Harmer
المصدر: British Journal of Pharmacology. 175:618-630
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Side effect, business.industry, Kinase, Axitinib, 03 medical and health sciences, Dose–response relationship, 030104 developmental biology, Pharmacokinetics, cardiovascular system, medicine, Potency, business, Tyrosine kinase, IC50, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::e029e19c600917d5467b5495041f099aTest
https://doi.org/10.1111/bph.14103Test -
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المؤلفون: Eric Gangl, Francis D. Gibbons, William McCoull, Martin Wild, Lorraine Graham, Hill Kathryn Jane, Brian Kelly, Srividya B. Balachander, David J. Owen, Sean Redmond, Marianne Ashford, Barry R. Davies, Alexander R. Harmer, Shenghua Wen, Iain Grant, Sonya Gales
المصدر: Cancer Research. 80:1718-1718
مصطلحات موضوعية: Cancer Research, Therapeutic index, Oncology, Tolerability, Chemistry, In vivo, Dendrimer, Pharmacology, Nanocarriers, Linker, Controlled release, Conjugate
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::8cc5b5a8344d601e4a673da8cfe48853Test
https://doi.org/10.1158/1538-7445.am2020-1718Test