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المؤلفون: Alessandro Schipani, Andrew Owen, Oluseye O. Bolaji, Saye Khoo, Adeniyi Olagunju
المصدر: J Antimicrob Chemother
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPYمصطلحات موضوعية: Adult, Cyclopropanes, Microbiology (medical), medicine.medical_specialty, Efavirenz, Adolescent, Anti-HIV Agents, Population, Black People, Nigeria, HIV Infections, Context (language use), Pharmacology, 030226 pharmacology & pharmacy, Article, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Pregnancy, Internal medicine, Genotype, medicine, Humans, Pharmacology (medical), 030212 general & internal medicine, Dosing, education, Cytochrome P-450 CYP2B6 Inducers, education.field_of_study, business.industry, medicine.disease, Infectious Disease Transmission, Vertical, Benzoxazines, Cytochrome P-450 CYP2B6, Infectious Diseases, chemistry, Alkynes, Toxicity, Female, business
وصف الملف: application/vnd.openxmlformats-officedocument.wordprocessingml.document
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ff5c04fceadf7e6b1e5dc96b36fff7b2Test
https://doi.org/10.1093/jac/dkx334Test -
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المؤلفون: Gerry Davies, Alessandro Schipani, Elizabeth Molyneux, Steve A. Ward, Rachel Mlota, Fraction K. Dzinjalamala, Saye Khoo, Henry Pertinez, Joep J. van Oosterhout, Nuria Lopez
المصدر: British Journal of Clinical Pharmacology. 81:679-687
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, education.field_of_study, Pediatrics, medicine.medical_specialty, Tuberculosis, business.industry, 030106 microbiology, Population, Fixed-dose combination, medicine.disease, 030226 pharmacology & pharmacy, Bioavailability, NONMEM, 03 medical and health sciences, 0302 clinical medicine, medicine, Pharmacology (medical), Dosing, Young adult, education, business, Rifampicin, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::04d56fce15bc3bcee396e326d20b6d38Test
https://doi.org/10.1111/bcp.12848Test -
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المؤلفون: Wouter H. J. Vaes, Kevin Park, Lindsay Byrne, Grzegorz Grynkiewicz, Alessandro Schipani, Jane Lass, Heili Varendi, Andrew M. Selby, Francis P. Crawley, Mark A. Turner, Sarah Siner, Esther van Duijn, Wioletta Maruszak, Rianne deLigt, Neil French, Colin R. Garner, Caroline Earnshaw
المصدر: British Journal of Clinical Pharmacology. 80:157-167
مصطلحات موضوعية: Pharmacology, Volume of distribution, Microdosing, business.industry, Area under the curve, Enteral administration, Therapeutic index, MicroDose, Pharmacokinetics, Medicine, Pharmacology (medical), Biological half-life, business
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::7234c220f9e560c9f5a2b9b5fc0a2ff5Test
https://doi.org/10.1111/bcp.12597Test -
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المؤلفون: David Back, Alessandro Schipani, Gerry Davies, Marco Siccardi, Saye Khoo, Andrew Owen
المصدر: Clinical Pharmacokinetics. 54:107-116
مصطلحات موضوعية: Adult, Cyclopropanes, Male, Drug, Efavirenz, Nevirapine, Adolescent, media_common.quotation_subject, Population, In Vitro Techniques, Pharmacology, Models, Biological, Maraviroc, Young Adult, chemistry.chemical_compound, Cyclohexanes, HIV Fusion Inhibitors, Humans, Medicine, Computer Simulation, Pharmacology (medical), Dosing, education, Aged, ADME, media_common, Clinical Trials as Topic, education.field_of_study, Dose-Response Relationship, Drug, business.industry, Middle Aged, Triazoles, Benzoxazines, Discontinuation, Anti-Retroviral Agents, chemistry, Alkynes, Reverse Transcriptase Inhibitors, Female, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0b6c3c7f80a500121c6ef5b40ccb66c3Test
https://doi.org/10.1007/s40262-014-0184-8Test -
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المؤلفون: David Back, Adeniyi Olagunju, Saye Khoo, Marco Siccardi, Alessandro Schipani, Andrew Owen, Deirdre Egan
المصدر: Pharmacogenetics and Genomics. 24:459-463
مصطلحات موضوعية: Adult, Male, Mrna expression, Population, Human immunodeficiency virus (HIV), Organic Anion Transporters, HIV Infections, Single-nucleotide polymorphism, Biology, Pharmacology, medicine.disease_cause, Polymorphism, Single Nucleotide, Lopinavir, Pharmacokinetics, Genetics, medicine, Cytochrome P-450 CYP3A, Humans, General Pharmacology, Toxicology and Pharmaceutics, education, Molecular Biology, Genetics (clinical), Aged, education.field_of_study, CYP3A4, Liver-Specific Organic Anion Transporter 1, Genetic Variation, HIV Protease Inhibitors, Middle Aged, Minor allele frequency, Molecular Medicine, Female, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::906eb0f8c973e2b9d84186ca0b0ef046Test
https://doi.org/10.1097/fpc.0000000000000073Test -
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المؤلفون: Andrew Owen, Alessandro Schipani, Marco Siccardi
المصدر: Pharmaceutical Nanotechnology: Innovation and Production ISBN: 9783527800681
Pharmaceutical Nanotechnology: Innovation and Productionمصطلحات موضوعية: medicine.medical_specialty, Chemistry, Blood circulation, Drug delivery, medicine, Nanomedicine, Intensive care medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::1f36511d22450046800106e8ad863598Test
https://doi.org/10.1002/9783527800681.ch15Test -
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المؤلفون: Saye Khoo, Alessandro Schipani, Giovanni Di Perri, Marco Simiele, Antonio D'Avolio, Howard L. McLeod, Gerry Davies, Charoen Chuchuttaworn, Sonia Rodríguez Novoa, Marco Siccardi, Janelle M. Hoskins, Vincent Soriano, Natpratou Saguenwong, Andrew Owen, David Back, Lorena Baietto, Anne M. Dvorak, Nitipatana Chierakul, Stefano Bonora, Lorena Cuenca
المصدر: Antimicrobial Agents and Chemotherapy. 54:5242-5250
مصطلحات موضوعية: Adult, Male, Receptors, Steroid, medicine.medical_specialty, ATP Binding Cassette Transporter, Subfamily B, Genotype, Pyridines, Atazanavir Sulfate, Population, Organic Anion Transporters, HIV Infections, Pharmacology, Polymorphism, Single Nucleotide, Young Adult, Gene Frequency, Pharmacokinetics, Internal medicine, medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, education, Aged, education.field_of_study, biology, CYP3A4, Liver-Specific Organic Anion Transporter 1, Pregnane X Receptor, Middle Aged, Circadian Rhythm, Bioavailability, Atazanavir, Infectious Diseases, Endocrinology, biology.protein, Female, Ritonavir, SLCO1B1, Oligopeptides, human activities, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ea0c40bb12e28f42007d3168cf036e6eTest
https://doi.org/10.1128/aac.00781-10Test -
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المؤلفون: Alex Musso Buendía, Alessandro Schipani, Dolores Gonzalez Pacanowska, Orla K. Mc Carthy, Luis M. Ruiz-Pérez, Reto Brun, Marcel Kaiser, Ian H. Gilbert
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:3809-3812
مصطلحات موضوعية: Stereochemistry, Trypanosoma cruzi, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Inhibitory Concentration 50, chemistry.chemical_compound, DUTP pyrophosphatase, Acetamides, parasitic diseases, Drug Discovery, Peptide synthesis, Animals, Chagas Disease, Amino Acids, Enzyme Inhibitors, Pyrophosphatases, Uracil, Molecular Biology, chemistry.chemical_classification, Dipeptide, biology, Organic Chemistry, biology.organism_classification, Trypanocidal Agents, Amino acid, Models, Chemical, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Acetamide
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::876734f3e2d26e47a398aed67fdca0d6Test
https://doi.org/10.1016/j.bmcl.2006.04.027Test -
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المؤلفون: Corinne Nguyen, Isabel Leal, Dolores González-Pacanowska, Britt-Louise Sahlberg, Alessandro Schipani, Luis M Ruiz-Pérez, Nils Gunnar Johansson, Ian H. Gilbert, Alexander Musso-Buendia, Marcel Kaiser, Ganasan Kasinathan, Gian Filippo Ruda, Reto Brun
المصدر: Journal of Medicinal Chemistry. 49:4183-4195
مصطلحات موضوعية: Models, Molecular, Erythrocytes, Plasmodium falciparum, In Vitro Techniques, Antimalarials, Structure-Activity Relationship, chemistry.chemical_compound, DUTP pyrophosphatase, Drug Discovery, Animals, Humans, Structure–activity relationship, Pyrophosphatases, Uracil, ADME, chemistry.chemical_classification, biology, Nucleosides, Stereoisomerism, Trityl Compounds, biology.organism_classification, Deoxyuridine, Enzyme, chemistry, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b71bba426ce4e5a34a71b03d41dc1c34Test
https://doi.org/10.1021/jm060126sTest -
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المؤلفون: Alison Jayne Foster, Andrew Owen, Neill J. Liptrott, Paul Curley, Phill Roberts, James Long, Alessandro Schipani, Philip Martin, Marco Giardiello, Darren Smith, Tom O. McDonald, Saye Khoo, Marco Siccardi, Steven Paul Rannard
المصدر: Advanced healthcare materials. 3(3)
مصطلحات موضوعية: Drug, Cyclopropanes, Male, Materials science, Efavirenz, Polymers, media_common.quotation_subject, Biomedical Engineering, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Biological Availability, Pharmacology, Biomaterials, chemistry.chemical_compound, Pharmacokinetics, Oral administration, In vivo, medicine, Animals, Humans, Particle Size, Rats, Wistar, media_common, Reverse-transcriptase inhibitor, Bioavailability, Benzoxazines, Rats, chemistry, Alkynes, Nanomedicine, Nanoparticles, Emulsions, Caco-2 Cells, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c31c4b4acf51db41b592ccfad7268457Test
https://pubmed.ncbi.nlm.nih.gov/23997027Test