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المؤلفون: Katharina Korpis, Valentina Dal Col, Patrick J. Bednarski, Stefanie Brune, Dirk Schepmann, Bernhard Wünsch, Frauke Weber, Sabrina Pricl, Erik Laurini
المساهمون: Frauke, Weber, Steffi, Brune, Katharina, Korpi, Patrick J., Bednarski, Laurini, Erik, DAL COL, Valentina, Pricl, Sabrina, Dirk, Schepmann, Bernhard, Wünsch
المصدر: Journal of Medicinal Chemistry. 57:2884-2894
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Guinea Pigs, sigma receptors, computer assisted drug design, Antineoplastic Agents, Apoptosis, Plasma protein binding, Molecular Dynamics Simulation, Piperazines, Structure-Activity Relationship, Neoplasms, Drug Discovery, Tumor Cells, Cultured, Animals, Humans, Receptors, sigma, Structure–activity relationship, Homology modeling, sigma receptor, Receptor, Molecular Structure, Chemistry, Brain, Ligand (biochemistry), Affinities, Cell culture, Molecular Medicine, Chromatography, Thin Layer, Protein Binding
وصف الملف: STAMPA
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::de21ded4a7d95a96339e4c5711ed5b77Test
https://doi.org/10.1021/jm401707tTest -
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المؤلفون: Carsten Lange, Frauke Weber, Patrick J. Bednarski, Maurizio Fermeglia, Bernhard Wünsch, Dirk Schepmann, Frederik Börgel, Stefanie Brune, Erik Laurini, Sabrina Pricl, Katharina Korpis
المصدر: Journal of Medicinal Chemistry. 59:5505-5519
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Stereochemistry, Guinea Pigs, Antineoplastic Agents, Apoptosis, Ligands, Heterocyclic Compounds, 2-Ring, Piperazines, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Receptors, sigma, Structure–activity relationship, Receptor, Cell Proliferation, Sigma-1 receptor, Dose-Response Relationship, Drug, Molecular Structure, Bicyclic molecule, Cell growth, Chemistry, Ligand, Biological activity, 030104 developmental biology, Mechanism of action, 030220 oncology & carcinogenesis, Thermodynamics, Molecular Medicine, Drug Screening Assays, Antitumor, medicine.symptom
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dcf03d726ba597ffbd869cae9faec2cbTest
https://doi.org/10.1021/acs.jmedchem.6b00585Test -
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المؤلفون: Antonio Donaire, Alicia Buceta, Gorakh S. Yellol, Christoph Janiak, Piotr Szumlas, Jyoti G. Yellol, Sergio A. Pérez, José Ruiz, Arturo Espinosa, Patrick J. Bednarski, Gamall Makhloufi
المصدر: Journal of medicinal chemistry. 58(18)
مصطلحات موضوعية: Models, Molecular, Benzimidazole, Stereochemistry, chemistry.chemical_element, Neovascularization, Physiologic, Angiogenesis Inhibitors, Antineoplastic Agents, Apoptosis, Ring (chemistry), Crystallography, X-Ray, Iridium, Ruthenium, chemistry.chemical_compound, Hydrolysis, Mice, Structure-Activity Relationship, Coordination Complexes, Cell Line, Tumor, Drug Discovery, Human Umbilical Vein Endothelial Cells, Molecule, Structure–activity relationship, Animals, Humans, Chelation, Serum Albumin, Molecular Structure, Caspase 3, Cell Cycle Checkpoints, 3. Good health, Enzyme Activation, chemistry, Drug Resistance, Neoplasm, Molecular Medicine, Benzimidazoles, Cisplatin, Drug Screening Assays, Antitumor, Reactive Oxygen Species, Hydrophobic and Hydrophilic Interactions
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::400275ebd8f51af862ca1e60cf781b8dTest
https://pubmed.ncbi.nlm.nih.gov/26313136Test