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المؤلفون: Steven C. Kim, Yongbo Hu, Nancy Torres, Dan Maarten Berger, Ariamala Gopalsamy, Kyung-Hee Kim, Weixin Xu, Donald Wojciechowicz, Larry Feldberg, Jeremy I. Levin, Dennis Powell, James M. Wilhelm, Greg Ciszewski, Eileen Frommer, Karen Collins, Minu Dutia, Robert Mallon
المصدر: Bioorganicmedicinal chemistry letters. 19(23)
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Crystallography, X-Ray, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Transferase, Structure–activity relationship, Molecular Biology, Protein Kinase Inhibitors, Trifluoromethyl, Molecular Structure, Kinase, Chemistry, Aryl, Organic Chemistry, Stereoisomerism, Pyrimidines, Benzamides, Molecular Medicine, Pyrazoles
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e8c93c7ce2c3fcc01d9a845c40838c5cTest
https://pubmed.ncbi.nlm.nih.gov/19864136Test -
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المؤلفون: Karen Collins, Steven C. Kim, Donald Wojciechowicz, Larry Feldberg, Frederick Lee, Eileen Frommer, Yongbo Hu, Robert Mallon, Ariamala Gopalsamy, Greg Ciszewski
المصدر: Bioorganicmedicinal chemistry letters. 19(10)
مصطلحات موضوعية: Proto-Oncogene Proteins B-raf, Pyrimidine, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Humans, Computer Simulation, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, biology, Kinase, Organic Chemistry, Small molecule, In vitro, Enzyme, Pyrimidines, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Signal transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fd8e36f6b9ef3c487a3b1c921c05d988Test
https://pubmed.ncbi.nlm.nih.gov/19362830Test -
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المصدر: Biochimica et biophysica acta. 1649(1)
مصطلحات موضوعية: Stereochemistry, Peptidomimetic, Biophysics, Peptide, Biochemistry, Binding, Competitive, Analytical Chemistry, Substrate Specificity, Serine, Proto-Oncogene Proteins p21(ras), Scissile bond, Methionine, Endopeptidases, Animals, Humans, Protease Inhibitors, Amino Acid Sequence, Isoleucine, Molecular Biology, Peptide sequence, chemistry.chemical_classification, Valine, Peptide Fragments, Recombinant Proteins, chemistry, Cysteine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d2fb1ae58c7d11d5579df85c4b2144a6Test
https://pubmed.ncbi.nlm.nih.gov/12818187Test -
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المؤلفون: Raymond J. Andersen, David E. Williams, Irwin Hollander, Akbar Tahir, Donald Wojciechowicz, Rob W. M. Van Soest, Karen Collins, Eileen Frommer, Robert Mallon, Kyle S. Craig
المساهمون: Systematische en Geografische Dierkunde (inactive) (IBED, FNWI)
المصدر: Tetrahedron Letters, 43, 4801-4804. Elsevier
مصطلحات موضوعية: Protease, biology, Chemistry, Stereochemistry, medicine.medical_treatment, Organic Chemistry, biology.organism_classification, Biochemistry, Terpenoid, Hippospongia, Sponge, Drug Discovery, medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5e95a66fa3ad03ea43b70cac32f6a62bTest
https://dare.uva.nl/personal/pure/en/publications/novel-sesterterpenoid-and-norsesterterpenoid-rceprotease-inhibitors-isolated-from-the-marine-sponge-hippospongia-spTest(43f45c56-7e33-4056-859f-ba243dd10e1d).html -
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المؤلفون: Wang Xiaolun, Levin I. Jeremy, Nancy Torres, Donald Wojciechowicz, Edward J. Salaski, Yongbo Hu, Eileen Frommer, Dan Maarten Berger, Dennis Powell, Karen Collins
المصدر: Molecular Cancer Therapeutics. 8:A85-A85
مصطلحات موضوعية: chemistry.chemical_classification, Cancer Research, Kinase, Cell, Wild type, Biology, Serine, Enzyme, medicine.anatomical_structure, Oncology, Biochemistry, chemistry, Cell culture, medicine, Signal transduction, Protein kinase A
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::524814e839cb0deb10ba60886cd95053Test
https://doi.org/10.1158/1535-7163.targ-09-a85Test