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1
المؤلفون: Fara Brasó-Maristany, Mònica Sánchez-Guixé, Andreu Ódena, Aleix Prat, Olga Rodriguez, Yasir H. Ibrahim, Alejandra Bruna, Elza C. de Bruin, Barry R. Davies, Alan Barnicle, Laia Monserrat, Judit Grueso, Carlos Caldas, Guillermo Villacampa, Nicholas C. Turner, Avinash Reddy, Paolo Nuciforo, Albert Gris-Oliver, Joaquín Arribas, Violeta Serra, Gordon B. Mills, Maurizio Scaltriti, Caroline S. Hirst, Mafalda Oliveira, Gaia Schiavon, Cristina Saura, Marta Guzman, Marta Palafox, Pedram Razavi, Mireia Parés, Rodrigo Dienstmann
المصدر: Clin Cancer Res
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Paclitaxel, Class I Phosphatidylinositol 3-Kinases, DNA Mutational Analysis, AKT1, P70-S6 Kinase 1, Breast Neoplasms, Tuberous Sclerosis Complex 1 Protein, Article, 03 medical and health sciences, Mice, 0302 clinical medicine, Breast cancer, Antineoplastic Combined Chemotherapy Protocols, medicine, Biomarkers, Tumor, PTEN, Animals, Humans, Pyrroles, Breast, Protein kinase B, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Mastectomy, biology, Fulvestrant, business.industry, TOR Serine-Threonine Kinases, Ribosomal Protein S6 Kinases, 70-kDa, medicine.disease, Prognosis, Metastatic breast cancer, Xenograft Model Antitumor Assays, 030104 developmental biology, Pyrimidines, Oncology, Chemotherapy, Adjuvant, Drug Resistance, Neoplasm, 030220 oncology & carcinogenesis, Mutation, biology.protein, Cancer research, Female, business, Proto-Oncogene Proteins c-akt, medicine.drug, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ef93ddf12491d1bbf7d5667c25fa96d7Test
https://pubmed.ncbi.nlm.nih.gov/32220884Test -
2
المؤلفون: A. Robert MacLeod, Kazuhiro Yoshikawa, Kazuko Sakai, Youngsoo Kim, Hayley Campbell, Koichi Sugimoto, Stephanie Klein, Marco A. De Velasco, Yurie Kura, Barry R. Davies, Yuji Hatanaka, Hirotsugu Uemura, Kazuto Nishio
المصدر: JCI Insight. 4
مصطلحات موضوعية: Male, 0301 basic medicine, medicine.drug_class, Antineoplastic Agents, Castration resistant, urologic and male genital diseases, Antiandrogen, Mice, Phosphatidylinositol 3-Kinases, 03 medical and health sciences, Prostate cancer, 0302 clinical medicine, Pharmacotherapy, Antisense Oligonucleotide Therapy, Animals, Humans, Medicine, Pyrroles, Protein kinase B, PI3K/AKT/mTOR pathway, Mice, Knockout, business.industry, Prostatic Neoplasms, General Medicine, Oligonucleotides, Antisense, medicine.disease, Gene Expression Regulation, Neoplastic, Mice, Inbred C57BL, Androgen receptor, Disease Models, Animal, Prostatic Neoplasms, Castration-Resistant, Pyrimidines, 030104 developmental biology, Drug Resistance, Neoplasm, Receptors, Androgen, 030220 oncology & carcinogenesis, Cancer research, Transcriptome, business, Proto-Oncogene Proteins c-akt, Research Article, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa8cf2bddeac4732db473566c0ff7ec1Test
https://doi.org/10.1172/jci.insight.122688Test -
3
المؤلفون: Stephen Green, Sylvie Guichard, Robert McEwen, Barry R. Davies, Urszula M. Polanska, Zoe Howard, Teresa Klinowska, Celina M. D'Cruz, Michael Grondine, Christine M. Chresta, Teeru Bihani, Graham Bigley, James W.T. Yates, Kurt Gordon Pike, Jon Curwen, Sabina Cosulich, Oona Delpuech, Martin Pass
المصدر: Molecular Cancer Therapeutics. 14:2508-2518
مصطلحات موضوعية: Cancer Research, Morpholines, Immunoblotting, Breast Neoplasms, Mechanistic Target of Rapamycin Complex 2, Mice, SCID, mTORC1, Mechanistic Target of Rapamycin Complex 1, Biology, Pharmacology, mTORC2, Drug Administration Schedule, Mice, Inbred NOD, Cell Line, Tumor, Antineoplastic Combined Chemotherapy Protocols, medicine, Animals, Humans, Fulvestrant, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Cell Proliferation, Mice, Knockout, Serine/threonine-specific protein kinase, Estradiol, Cell growth, TOR Serine-Threonine Kinases, Xenograft Model Antitumor Assays, Tumor Burden, HEK293 Cells, Pyrimidines, Receptors, Estrogen, Oncology, Multiprotein Complexes, Benzamides, MCF-7 Cells, Hormonal therapy, Female, Signal Transduction, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::689b8ba235f8b435652d9591e5d9196fTest
https://doi.org/10.1158/1535-7163.mct-15-0365Test -
4
المؤلفون: Lindsay C, Spender, G John, Ferguson, Gareth D, Hughes, Barry R, Davies, Frederick W, Goldberg, Blanca, Herrera, Richard G, Taylor, Lauren S, Strathearn, Owen J, Sansom, Simon T, Barry, Gareth J, Inman
المصدر: Molecular pharmacology. 95(2)
مصطلحات موضوعية: Receptor, Transforming Growth Factor-beta Type I, Smad2 Protein, Cell Line, DNA-Binding Proteins, Mice, Bone Morphogenetic Proteins, NIH 3T3 Cells, Animals, Neoplasm Metastasis, Phosphorylation, Activin Receptors, Type I, Protein Kinase Inhibitors, Cell Proliferation, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=pmid________::450dfb12551ade5dad0de67c197e09c5Test
https://pubmed.ncbi.nlm.nih.gov/30459156Test -
5
المؤلفون: Claire Crafter, Lillian Castriotta, Stephen Green, Martina Fitzek, Cath Trigwell, Donald J. Ogilvie, Steve Powell, Rebecca Ellston, Mandy Lawson, Urs Hancox, Lyndsey Hanson, Barry R. Davies, Lara Ward, Hannah Dry, Sabina Cosulich, Marie Cumberbatch, Celina M. D'Cruz, Stephen R. Wedge, Barlaam Bernard Christophe, Carol Lenaghan, Elizabeth A. Harrington, Paul D. Smith, Emily Foster, Simon T. Barry
المصدر: Molecular Cancer Therapeutics. 14:48-58
مصطلحات موضوعية: Male, Cancer Research, medicine.medical_treatment, Antineoplastic Agents, Triple Negative Breast Neoplasms, Docetaxel, Pharmacology, Mice, Prostate cancer, Prostate, Cell Line, Tumor, Antineoplastic Combined Chemotherapy Protocols, medicine, Animals, Humans, PTEN, PI3K/AKT/mTOR pathway, Cell Proliferation, Phosphoinositide-3 Kinase Inhibitors, Chemotherapy, Aniline Compounds, biology, Cell growth, PTEN Phosphohydrolase, Prostatic Neoplasms, Drug Synergism, medicine.disease, Xenograft Model Antitumor Assays, medicine.anatomical_structure, Oncology, Chromones, Tumor progression, biology.protein, Female, Taxoids, Signal Transduction, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d0de79ea05648a8f13f0ac9f05b31f90Test
https://doi.org/10.1158/1535-7163.mct-14-0406Test -
6
المؤلفون: Diana Tuskova, James T. Lynch, German Ott, Kevin Hudson, Wolfgang E. Berdel, Myroslav Zapukhlyak, Barry R. Davies, Simon T. Barry, Matthias Pfeifer, Jan Molinsky, Peter Lenz, Michele Mayo, Kristian Erdmann, Michael Grau, Petra Vockova, Pavel Klener, Marek Trneny, Annette M. Staiger, Daniela Schwammbach, Beiying Dai, Tabea Erdmann, Francisco Cruzalegui, Georg Lenz, Urszula M. Polanska, Michael Grondine
المصدر: Blood. 130(3)
مصطلحات موضوعية: 0301 basic medicine, Apoptosis, Pharmacology, Biochemistry, Tyrosine-kinase inhibitor, chemistry.chemical_compound, Mice, Phosphatidylinositol 3-Kinases, 0302 clinical medicine, Piperidines, hemic and lymphatic diseases, Agammaglobulinaemia Tyrosine Kinase, Phosphoinositide-3 Kinase Inhibitors, Oxadiazoles, biology, NF-kappa B, Drug Synergism, Hematology, Protein-Tyrosine Kinases, Gene Expression Regulation, Neoplastic, Drug Combinations, Organ Specificity, 030220 oncology & carcinogenesis, Ibrutinib, Lymphoma, Large B-Cell, Diffuse, Signal transduction, Signal Transduction, medicine.drug_class, Immunology, Antineoplastic Agents, Proto-Oncogene Proteins c-myc, 03 medical and health sciences, medicine, Animals, Humans, Pyrroles, Protein kinase B, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Phosphoinositide 3-kinase, Akt inhibitor AZD5363, Adenine, PTEN Phosphohydrolase, Germinal center, Cell Biology, Xenograft Model Antitumor Assays, 030104 developmental biology, Pyrimidines, chemistry, biology.protein, Cancer research, Pyrazoles, Drug Screening Assays, Antitumor, Proto-Oncogene Proteins c-akt
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::15b7729777f360eff7908ecbecbfbd4dTest
https://pubmed.ncbi.nlm.nih.gov/28729335Test -
7
المؤلفون: Michael Ittmann, Peter S. Nelson, Paul D. Smith, Barry R. Davies, Shu Feng, Longjiang Shao, Ilsa Coleman, Patricia Castro
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, MAPK/ERK pathway, Male, STAT3 Transcription Factor, medicine.medical_specialty, kinase inhibitor, Mice, SCID, Fibroblast growth factor, Piperazines, 03 medical and health sciences, Internal medicine, Cell Line, Tumor, Antineoplastic Combined Chemotherapy Protocols, medicine, Animals, Humans, Pyrroles, Receptor, Fibroblast Growth Factor, Type 1, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Protein kinase B, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Cell Proliferation, Dose-Response Relationship, Drug, Kinase, business.industry, Fibroblast growth factor receptor 1, AKT, fibroblast growth factors, Prostatic Neoplasms, prostate cancer, Xenograft Model Antitumor Assays, 3. Good health, Tumor Burden, 030104 developmental biology, Endocrinology, Pyrimidines, Oncology, Fibroblast growth factor receptor, Benzamides, Cancer research, Pyrazoles, Signal transduction, business, Proto-Oncogene Proteins c-akt, signal transduction, Research Paper
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a286cbf59b00d90c15d81932e9cb0d4eTest
https://pubmed.ncbi.nlm.nih.gov/28008155Test -
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المؤلفون: Colin P.N. Dinney, Barry R. Davies, David J. McConkey, Giovanni Nitti, Ashish M. Kamat, Rian J. Dickstein
المصدر: Cancer Biology & Therapy. 13:1325-1338
مصطلحات موضوعية: Cancer Research, Class I Phosphatidylinositol 3-Kinases, Apoptosis, Biology, Phosphatidylinositol 3-Kinases, chemistry.chemical_compound, Cell Line, Tumor, Autophagy, Humans, Propidium iodide, Phosphorylation, Protein Kinase Inhibitors, Protein kinase B, PI3K/AKT/mTOR pathway, Cell Proliferation, Sirolimus, Pharmacology, Cell growth, TOR Serine-Threonine Kinases, RPTOR, Urinary Bladder Neoplasms, Oncology, chemistry, Mutation, Cancer cell, Cancer research, Molecular Medicine, Signal transduction, Apoptosis Regulatory Proteins, Proto-Oncogene Proteins c-akt, Signal Transduction, Research Paper
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::da8b688b9e0129cfacdcee7b88f76f91Test
https://doi.org/10.4161/cbt.21793Test -
9
المؤلفون: Robert Shaw, Dawn Baker, Margaret Veldman-Jones, Jonathan R. Dry, Dennis Wang, Claire Rooney, Pei Zhang, Sarah Cross, Michael Dymond, Oona Delpuech, Lorraine Mooney, Barry R. Davies, Joanne Wilson, Paul D. Smith, Elaine Kilgour
المصدر: Molecular cancer therapeutics. 15(11)
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, FGFR Inhibition, EGR1, Antineoplastic Agents, Biology, Piperazines, 03 medical and health sciences, Mice, Cell Line, Tumor, Animals, Cluster Analysis, Humans, Protein kinase B, PI3K/AKT/mTOR pathway, Regulation of gene expression, Gene Expression Profiling, Gene Amplification, Reproducibility of Results, Molecular biology, Receptors, Fibroblast Growth Factor, Gene expression profiling, Disease Models, Animal, 030104 developmental biology, Oncology, Gene Expression Regulation, Benzamides, Cancer research, Phosphorylation, Heterografts, Pyrazoles, Female, Signal transduction, Transcriptome, Biomarkers, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a7f5322a34a71f41b2d372c212f670f1Test
https://pubmed.ncbi.nlm.nih.gov/27550940Test -
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المؤلفون: Sylvie Guichard, Robert W. Wilkinson, Sarah L. Fenton, Yi-Long Wu, Paul D. Smith, Jingchuan Zhang, Barry R. Davies, Armelle Logie, Sarah V. Holt, Sarah Runswick, D Alferez, Yi Gu, Christine M. Chresta
المصدر: Cancer Research. 72:1804-1813
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, Lung Neoplasms, MAP Kinase Signaling System, Morpholines, Apoptosis, mTORC1, Mitogen-activated protein kinase kinase, Biology, mTORC2, Proto-Oncogene Proteins p21(ras), Mice, Carcinoma, Non-Small-Cell Lung, Proto-Oncogene Proteins, Animals, Humans, Protein Kinase Inhibitors, Protein kinase B, PI3K/AKT/mTOR pathway, Mitogen-Activated Protein Kinase Kinases, Gene Expression Profiling, TOR Serine-Threonine Kinases, RPTOR, Neoplasms, Experimental, Xenograft Model Antitumor Assays, Oncology, Mutation, ras Proteins, Cancer research, Selumetinib, Benzimidazoles, Female, Colorectal Neoplasms, Signal Transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::72dae4cf385b4a4e49a80db38ebb80b8Test
https://doi.org/10.1158/0008-5472.can-11-1780Test