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المؤلفون: Katherine Hopkins, Daniel Hoyer, Soumya Mukherjee, Jonathan E. Mangum, Dalia Ponce, Laura H. Jacobson
المصدر: Medicine in Drug Discovery, Vol 11, Iss, Pp 100102-(2021)
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, Mass spectrometry, Chemistry, Neuropeptide, Orexin, Triple quadrupole mass spectrometer, Animal models, RS1-441, Orexin-A, Sleep deprivation, Mice, Cerebrospinal fluid, Targeted mass spectrometry, Endocrinology, Pharmacy and materia medica, Internal medicine, Drug Discovery, medicine, Pharmacology (medical), Circadian rhythm, medicine.symptom, Arousal, Orexins/hypocretins, Sleep
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ea3fc5213706014db381fb39cdf5d7a7Test
http://www.sciencedirect.com/science/article/pii/S2590098621000233Test -
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المؤلفون: Tetsuya Shiga, Yusuke Osakabe, Sho Horikoshi, Hiroshi Hoshino, Hirooki Yabe, Kazuko Kanno, Itaru Miura, Haruka Ochiai
المصدر: Journal of psychopharmacology (Oxford, England). 35(12)
مصطلحات موضوعية: Adult, Male, Side effect, medicine.drug_class, Mismatch negativity, Pharmacology, Lorazepam, 03 medical and health sciences, Benzodiazepines, Young Adult, 0302 clinical medicine, Discrimination, Psychological, Medicine, Humans, Pharmacology (medical), Cognitive Dysfunction, 030212 general & internal medicine, Cognitive decline, Benzodiazepine, business.industry, Suvorexant, Antagonist, Electroencephalography, Azepines, Triazoles, Event-Related Potentials, P300, Orexin receptor, Psychiatry and Mental health, Tolerability, Auditory Perception, Evoked Potentials, Auditory, Female, Orexin Receptor Antagonists, business, 030217 neurology & neurosurgery
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::67dee48dc49baa60fe2b41d5127f1512Test
https://pubmed.ncbi.nlm.nih.gov/34330170Test -
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المؤلفون: Muneto Izuhara, Shoko Miura, Koji Otsuki, Michiharu Nagahama, Maiko Hayashida, Sadayuki Hashioka, Hiroya Asou, Hajime Kitagaki, Masatoshi Inagaki
المصدر: Frontiers in Psychiatry, Vol 12 (2021)
Frontiers in Psychiatryمصطلحات موضوعية: glia, insomnia, ventral tegmental area, RC435-571, Pharmacology, Creatine, chemistry.chemical_compound, mental disorders, Medicine, Premovement neuronal activity, Original Research, Psychiatry, psychiatric patients, business.industry, Dopaminergic, Suvorexant, Antagonist, suvorexant, magnetic resonance spectroscopy, Orexin receptor, Orexin, Ventral tegmental area, Psychiatry and Mental health, medicine.anatomical_structure, chemistry, nervous system, orexin, business, psychological phenomena and processes
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04734ffe5c6f2011c00194c7a16c49a2Test
https://www.frontiersin.org/articles/10.3389/fpsyt.2021.714376/fullTest -
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المؤلفون: Fabio Arturo Iannotti, Fabiana Piscitelli, Pietro Amodeo, Rosa Maria Vitale, Vincenzo Di Marzo, Ranjev Savopoulos, Luigia Cristino, Aniello Schiano Moriello, Royston A. Gray, Luciano De Petrocellis, Lea Tunisi
المصدر: Biomolecules, Vol 11, Iss 1134, p 1134 (2021)
Biomolecules
Volume 11
Issue 8
Biomolecules 11 (2021). doi:10.3390/biom11081134
info:cnr-pdr/source/autori:Vitale R.M.; Iannotti F.A.; Moriello A.S.; Tunisi L.; Piscitelli F.; Savopoulos R.; Cristino L.; De Petrocellis L.; Amodeo P.; Gray R.; Di Marzo V./titolo:Identification and characterization of cannabidiol as an ox1r antagonist by computational and in vitro functional validation/doi:10.3390%2Fbiom11081134/rivista:Biomolecules/anno:2021/pagina_da:/pagina_a:/intervallo_pagine:/volume:11مصطلحات موضوعية: Protein Conformation, alpha-Helical, 0301 basic medicine, Gene Expression, Pharmacology, Biochemistry, Radioligand Assay, cannabidiol, 0302 clinical medicine, Transgenes, Receptor, media_common, Chemistry, calcium mobilization assay, Ligand (biochemistry), calcium influx assay, Orexin receptor, QR1-502, Molecular Imaging, Molecular Docking Simulation, calcium imaging, Anticonvulsants, Orexin Receptor Antagonists, Protein Binding, medicine.drug, Drug, orexin receptors, OX1R, media_common.quotation_subject, CHO Cells, Microbiology, Article, 03 medical and health sciences, Cricetulus, medicine, Animals, Humans, Protein Interaction Domains and Motifs, Molecular Biology, Orexins, Binding Sites, Antagonist, antagonist, molecular docking, In vitro, molecular dynamics, Orexin, Kinetics, 030104 developmental biology, Anti-Anxiety Agents, Calcium, Protein Conformation, beta-Strand, Cannabidiol, 030217 neurology & neurosurgery
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::774e5847c77075e8bf23ab08f2e5ffadTest
https://www.mdpi.com/2218-273X/11/8/1134Test -
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المؤلفون: William Stoops, Justin C. Strickland, Kevin W. Hatton, Lon R. Hays, Abner O. Rayapati, Joshua A. Lile, Craig R. Rush
المصدر: Pharmacology Biochemistry and Behavior. 220:173466
مصطلحات موضوعية: Pharmacology, History, Orexins, Polymers and Plastics, Clinical Biochemistry, Azepines, Triazoles, Toxicology, Biochemistry, Industrial and Manufacturing Engineering, Behavioral Neuroscience, Cocaine, Orexin Receptors, Animals, Humans, Orexin Receptor Antagonists, Business and International Management, Biological Psychiatry
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b3c0b1724bdf9a32e3407294960b420eTest
https://doi.org/10.1016/j.pbb.2022.173466Test -
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المؤلفون: Maryam Majidinezhad, Haleh Amirteymouri, Saeideh Karimi-haghighi, Masoumeh Kourosh-Arami, Abbas Haghparast
المصدر: European journal of pharmacology. 930
مصطلحات موضوعية: Pharmacology, Orexins, Reward, Orexin Receptors, Ventral Tegmental Area, Animals, Rats, Wistar, Methamphetamine, Rats
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::df5ad154c4e8d1c2e9a16417c46145ccTest
https://pubmed.ncbi.nlm.nih.gov/35921956Test -
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المصدر: Neuropharmacology
مصطلحات موضوعية: Pharmacology, Male, Hypothalamo-Hypophyseal System, Orexins, Corticotropin-Releasing Hormone, Pituitary-Adrenal System, Self Administration, Receptors, Corticotropin-Releasing Hormone, Article, Rats, Cellular and Molecular Neuroscience, Orexin Receptors, Animals, Rats, Wistar
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a7c504bb3bbf47eb74e25227faba9695Test
https://europepmc.org/articles/PMC9176217Test/ -
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المؤلفون: Larisa Reyderman, Jagadeesh Aluri, Kenya Nakai, Bojan Lalovic, Margaret Moline, Ishani Landry, Takashi Ueno, Satish Dayal, Yukiko Miyajima, Nancy Hall, Gleb Filippov
المصدر: Clinical Pharmacology in Drug Development
مصطلحات موضوعية: Adult, Male, CYP2B6, Pyridines, Itraconazole, CYP3A, orexin receptor antagonists, Cmax, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, Young Adult, 03 medical and health sciences, 0302 clinical medicine, drug‐drug interaction, Pharmacokinetics, Cytochrome P-450 CYP3A, Humans, Medicine, Drug Interactions, Pharmacology (medical), Cytochrome P-450 Enzyme Inducers, Bupropion, business.industry, Brief Report, Middle Aged, Cytochrome P-450 CYP2B6, Pyrimidines, Area Under Curve, 030220 oncology & carcinogenesis, Cytochrome P-450 CYP3A Inhibitors, Midazolam, Female, Brief Reports, business, pharmacokinetics, Fluconazole, lemborexant, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1bcf08514e8d52bbf289e88aa00268bcTest
https://doi.org/10.1002/cpdd.915Test -
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المصدر: Drug Alcohol Depend
مصطلحات موضوعية: Male, medicine.medical_specialty, Evening, medicine.medical_treatment, Toxicology, Article, Methamphetamine, Internal medicine, Acetamides, medicine, Animals, Pharmacology (medical), Morning, Pharmacology, business.industry, Antagonist, Isoquinolines, Macaca mulatta, Orexin receptor, Orexin, Stimulant, Psychiatry and Mental health, Endocrinology, Female, Orexin Receptor Antagonists, Almorexant, business, Sleep, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8aadc10f2ed736bdb3ef384bbeebcc96Test
https://europepmc.org/articles/PMC8464508Test/ -
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المؤلفون: Martine Gehin, Jolanta Wierdak, Jasper Dingemanse, Giancarlo Sabattini, Patricia N. Sidharta
المصدر: British journal of clinical pharmacologyREFERENCES. 88(2)
مصطلحات موضوعية: Male, Efavirenz, Pyrrolidines, Cmax, Pharmacology, chemistry.chemical_compound, Pharmacokinetics, Medicine, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), Drug Interactions, Prospective Studies, CYP3A4, business.industry, Antagonist, Imidazoles, Cytochrome P-450 CYP3A Inducers, Hydrogen-Ion Concentration, Famotidine, Orexin receptor, Tolerability, chemistry, Area Under Curve, Orexin Receptor Antagonists, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::43f316bb390a8f0097914f56d1a5ca2dTest
https://pubmed.ncbi.nlm.nih.gov/34371524Test