-
1
المؤلفون: Eirik Sundby, Kristin G. Nørsett, Bård Helge Hoff, Silje Henriksen, Jin Han
المصدر: European Journal of Medicinal Chemistry
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, hERG, Pharmacology, Cell Line, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Stability, Drug Discovery, medicine, Humans, Potency, Pyrroles, Epidermal growth factor receptor, Cell Proliferation, ADME, EGFR inhibitors, chemistry.chemical_classification, biology, Organic Chemistry, General Medicine, EGFR, Pyrrolopyrimidine, SAR, Metabolism, Erlotinib, ErbB Receptors, Pyrimidines, 030104 developmental biology, Enzyme, Biochemistry, chemistry, Drug Design, 030220 oncology & carcinogenesis, biology.protein, Efflux, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1c170e443e60845774e85f6d7385051eTest
https://doi.org/10.1016/j.ejmech.2016.08.068Test -
2
المؤلفون: Kristin G. Nørsett, Eirik Sundby, Sondre Nervik, Bård Helge Hoff, Jin Han, Svein Jacob Kaspersen
المصدر: European Journal of Medicinal Chemistry. 119:278-299
مصطلحات موضوعية: Protein Conformation, Stereochemistry, Stereoisomerism, 01 natural sciences, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Protein structure, Drug Discovery, medicine, Structure–activity relationship, Moiety, Amines, Protein Kinase Inhibitors, EGFR inhibitors, Pharmacology, 010405 organic chemistry, Kinase, Aryl, Organic Chemistry, General Medicine, 0104 chemical sciences, ErbB Receptors, Molecular Docking Simulation, Kinetics, Pyrimidines, chemistry, 030220 oncology & carcinogenesis, Erlotinib, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9efcd7efaa05464b58400b33c79f8fb6Test
https://doi.org/10.1016/j.ejmech.2016.04.054Test -
3
المؤلفون: Eirik Sundby, Ann Christin Reiersølmoen, Bård Helge Hoff, Jin Han
المصدر: European Journal of Medicinal Chemistry
مصطلحات موضوعية: 0301 basic medicine, Cell Survival, Retinoic acid, Peripheral blood mononuclear cell, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, Humans, Secretion, Mode of action, Interleukin 5, Pharmacology, Orphan receptor, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Interleukin-17, Organic Chemistry, General Medicine, Molecular biology, HEK293 Cells, Pyrimidines, 030104 developmental biology, chemistry, Leukocytes, Mononuclear, Interleukin 17
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::893671f4e99ae7a07853be2354389cbeTest
http://hdl.handle.net/11250/2599282Test -
4
المؤلفون: Eli Kjøbli, Eirik Sundby, Svein Jacob Kaspersen, Geir Bjørkøy, Line Rydså, Steffen Bugge, Jin Han, Bård Helge Hoff, Kristin G. Nørsett
المصدر: European Journal of Pharmaceutical Sciences. 59:69-82
مصطلحات موضوعية: Models, Molecular, Pharmaceutical Science, Antineoplastic Agents, Pharmacology, Colony stimulating factor 1 receptor, Structure-Activity Relationship, Cell Line, Tumor, medicine, Humans, Pyrroles, Epidermal growth factor receptor, Amines, Protein Kinase Inhibitors, Cell Proliferation, chemistry.chemical_classification, biology, Chemistry, Kinase, Cell growth, ErbB Receptors, Pyrimidines, src-Family Kinases, Enzyme, Biochemistry, Cell culture, biology.protein, Erlotinib, Proto-oncogene tyrosine-protein kinase Src, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aeba3f7c0964eaed544adc926510e6b6Test
https://doi.org/10.1016/j.ejps.2014.04.011Test -
5
المؤلفون: Ina Stuen, Lene Østby, Arne Reimers, Eirik Sundby
المصدر: European Journal of Drug Metabolism and Pharmacokinetics
مصطلحات موضوعية: medicine.medical_specialty, UGT1A4, Glucuronosyltransferase, Clinical chemistry, Placenta, Blotting, Western, Biology, Lamotrigine, Isozyme, Gene Expression Regulation, Enzymologic, Western blot, Pregnancy, Microsomes, Internal medicine, medicine, Humans, Pharmacology (medical), reproductive and urinary physiology, Pharmacology, Original Paper, Epilepsy, medicine.diagnostic_test, Triazines, medicine.disease, Pregnancy Complications, Endocrinology, medicine.anatomical_structure, Case-Control Studies, embryonic structures, Microsome, biology.protein, Anticonvulsants, Female, UGT
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aed616be8c95f1f1abca6231b3ccba3aTest
https://doi.org/10.1007/s13318-010-0021-xTest -
6
المؤلفون: Bård Helge Hoff, Jin Han, Eirik Sundby, Svein Jacob Kaspersen
المصدر: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences. 80
مصطلحات موضوعية: Lung Neoplasms, Pharmaceutical Science, Antineoplastic Agents, Breast Neoplasms, Pharmacology, In Vitro Techniques, Lapatinib, Erlotinib Hydrochloride, Cell Line, Tumor, medicine, Cytochrome P-450 Enzyme Inhibitors, Humans, Pyrroles, IC50, ADME, Cell Proliferation, Ovarian Neoplasms, Dose-Response Relationship, Drug, Chemistry, Dasatinib, ErbB Receptors, Pyrimidines, Female, Efflux, Erlotinib, Caco-2 Cells, Tyrosine kinase, Drug metabolism, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9430425cf4f2b1dd47dcebd5690e1496Test
https://pubmed.ncbi.nlm.nih.gov/26296860Test -
7
المؤلفون: Bård Helge Hoff, Ingri Ullestad Moen, Kent-Ove Kragseth Sylte, Steffen Bugge, Eirik Sundby
المصدر: European journal of medicinal chemistry. 94
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Models, Molecular, Chemistry, Stereochemistry, Organic Chemistry, Stereoisomerism, General Medicine, Combinatorial chemistry, ErbB Receptors, Structure-Activity Relationship, Activity measurements, Enzyme, Gefitinib, Pyrimidines, Binding efficiency, Drug Discovery, Retrospective analysis, medicine, Moiety, Protein Kinase Inhibitors, EGFR inhibitors, Epidermal growth factor receptor tyrosine kinase, medicine.drug, Retrospective Studies
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2da781867991cd3c09d954f90888555dTest
https://pubmed.ncbi.nlm.nih.gov/25768701Test -
8
المؤلفون: Eirik Sundby, Synne Larsen, Unni Nonstad, Bård Helge Hoff, Geir Bjørkøy, Steffen Bugge, Svein Jacob Kaspersen
المصدر: European journal of medicinal chemistry. 75
مصطلحات موضوعية: Models, Molecular, Benzylamines, Pyrimidine, Stereochemistry, Mutant, Antineoplastic Agents, chemistry.chemical_compound, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Potency, Humans, IC50, Protein Kinase Inhibitors, EGFR inhibitors, Pharmacology, Chemistry, Organic Chemistry, General Medicine, In vitro, ErbB Receptors, Pyrimidines, Biochemistry, Cell culture, Erlotinib, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::076e87fc8ead7a1f45de3cc07f6b5422Test
https://pubmed.ncbi.nlm.nih.gov/24556149Test -
9
مصطلحات موضوعية: Antifungal, Benzylamines, Antifungal Agents, medicine.drug_class, Stereochemistry, Microbial Sensitivity Tests, Trichophyton rubrum, Naphthalenes, Trichophyton mentagrophytes, Trichophyton, Drug Discovery, medicine, Amines, Terbinafine, Antifungal agents, Pharmacology, Cryptococcus neoformans, Molecular Structure, biology, Lipase B from Candida antarctica, Chemistry, Squalene epoxidase, Organic Chemistry, Stereoisomerism, General Medicine, biology.organism_classification, In vitro, VDP::Medisinske Fag: 700::Basale medisinske, odontologiske og veterinærmedisinske fag: 710::Medisinsk biokjemi: 726, Medisinske Fag: 700::Basale medisinske, odontologiske og veterinærmedisinske fag: 710::Medisinsk biokjemi: 726 [VDP]
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6edde9fbf4ae67fd305c5d08a70f8636Test
https://hdl.handle.net/10642/1899Test -
10
المؤلفون: Veronica Willassen, Erik Fuglseth, Christopher Sørum, Eirik Sundby, Bård Helge Hoff, Svein Jacob Kaspersen, Geir Bjørkøy, Eli Kjøbli
المصدر: European journal of medicinal chemistry. 46(12)
مصطلحات موضوعية: Models, Molecular, Pyrimidine, Stereochemistry, media_common.quotation_subject, chemistry.chemical_element, Antineoplastic Agents, Electrophilic aromatic substitution, HeLa, chemistry.chemical_compound, Structure-Activity Relationship, Neoplasms, Drug Discovery, Structure–activity relationship, Humans, Pyrroles, Internalization, Protein Kinase Inhibitors, media_common, Pharmacology, biology, Chemistry, Aryl, Organic Chemistry, General Medicine, biology.organism_classification, ErbB Receptors, Pyrimidines, Tyrosine kinase, Palladium, HeLa Cells
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a87f7fc879a7117e56673ee5831cf8e7Test
https://pubmed.ncbi.nlm.nih.gov/22018877Test