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المؤلفون: Victor Moreno, Noelia Nebot, Emmanuel Bouillaud, Dung-Yang Lee, Eva Muñoz-Couselo, Christina S. Won, Eduard Gasal
المساهمون: Institut Català de la Salut, [Nebot N, Lee DY, Gasal E] Novartis Pharmaceuticals Corporation, East Hanover, New Jersey, USA. [Won CS] Novartis Institutes for BioMedical Research, East Hanover, New Jersey, USA. [Moreno V] START Madrid-FJD, Hospital Universitario Fundación Jiménez Díaz, Madrid, Spain. [Muñoz-Couselo E] Vall d’Hebron Institute of Oncology (VHIO), Barcelona, Spain. Vall d’Hebron Hospital Universitari, Barcelona, Spain. [Bouillaud E] Novartis Pharma AG, Basel, Switzerland, Vall d'Hebron Barcelona Hospital Campus
المصدر: Clinical Pharmacology in Drug Development
Scientiaمصطلحات موضوعية: Male, CYP3A4, CYP3A, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, fenómenos fisiológicos::fenómenos farmacológicos y toxicológicos::fenómenos farmacológicos::interacciones farmacológicas [FENÓMENOS Y PROCESOS], 0302 clinical medicine, Oximes, Medicine, fenómenos fisiológicos::fenómenos farmacológicos y toxicológicos::farmacocinética [FENÓMENOS Y PROCESOS], Cytochrome P-450 CYP3A, Pharmacology (medical), Drug Interactions, Rosuvastatin Calcium, OATP, Liver-Specific Organic Anion Transporter 1, Imidazoles, Articles, Middle Aged, Other subheadings::/pharmacology [Other subheadings], Physiological Phenomena::Pharmacological and Toxicological Phenomena::Pharmacokinetics [PHENOMENA AND PROCESSES], 030220 oncology & carcinogenesis, Area Under Curve, Female, pharmacokinetics, medicine.drug, Adult, Midazolam, Cmax, Original Manuscript, transporters, Chemical Actions and Uses::Pharmacologic Actions::Molecular Mechanisms of Pharmacological Action::Enzyme Inhibitors::Protein Kinase Inhibitors [CHEMICALS AND DRUGS], 03 medical and health sciences, Solute Carrier Organic Anion Transporter Family Member 1B3, Pharmacokinetics, Humans, Rosuvastatin, dabrafenib, Protein Kinase Inhibitors, drug interaction, Farmacocinètica, business.industry, acciones y usos químicos::acciones farmacológicas::mecanismos moleculares de acción farmacológica::inhibidores enzimáticos::inhibidores de proteínas cinasas [COMPUESTOS QUÍMICOS Y DROGAS], Dabrafenib, Drug interaction, Medicaments - Interacció, Proteïnes quinases - Inhibidors, Physiological Phenomena::Pharmacological and Toxicological Phenomena::Pharmacological Phenomena::Drug Interactions [PHENOMENA AND PROCESSES], Otros calificadores::/farmacología [Otros calificadores], business
وصف الملف: application/pdf
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7adef14bde6abca56c9d91bfe2b8074dTest
http://europepmc.org/articles/PMC8453865Test -
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المؤلفون: Tycho Heimbach, Handan He, Christina S. Won, Felix Huth, Kenichi Umehara
المصدر: Biopharmaceutics & Drug Disposition. 39:152-163
مصطلحات موضوعية: Pharmacology, Physiologically based pharmacokinetic modelling, CYP3A4, business.industry, Cmax, virus diseases, Pharmaceutical Science, General Medicine, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, immune system diseases, In vivo, 030220 oncology & carcinogenesis, medicine, heterocyclic compounds, Pharmacology (medical), Ketoconazole, Ritonavir, Dosing, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_________::25adfea51b5124afbaf648ccb44a0773Test
https://doi.org/10.1002/bdd.2122Test -
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المؤلفون: Handan He, Heidi J. Einolf, Christina S. Won, Lai Wang, Helen Gu, Wen Lin, Dung Yu Chun, James B. Mangold
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 45(12)
مصطلحات موضوعية: Physiologically based pharmacokinetic modelling, Indoles, medicine.drug_class, Midazolam, Pharmaceutical Science, Pharmacology, Hydroxamic Acids, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, In vivo, Panobinostat, medicine, Cytochrome P-450 CYP3A, Cytochrome P-450 Enzyme Inhibitors, Humans, Drug Interactions, Chemistry, Histone deacetylase inhibitor, Area under the curve, Gastric Acidity Determination, Drug interaction, Cytochrome P-450 CYP2C19, Histone Deacetylase Inhibitors, 030220 oncology & carcinogenesis, Enzyme Induction, Microsomes, Liver, Ketoconazole, Rifampin, Oxidation-Reduction, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::38cd9dac1e23d8ca3898d85896f59acaTest
https://pubmed.ncbi.nlm.nih.gov/28912253Test -
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المؤلفون: Christina S. Won, Lai Wang, Jocelyn Zhou, Sam Rebello, Heidi J. Einolf
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 45(4)
مصطلحات موضوعية: Drug, Adult, Male, Physiologically based pharmacokinetic modelling, Time Factors, CYP3A, Metabolic Clearance Rate, Pyridines, media_common.quotation_subject, Cmax, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, Models, Biological, Sonidegib, 03 medical and health sciences, chemistry.chemical_compound, Young Adult, 0302 clinical medicine, Pharmacokinetics, Neoplasms, Medicine, Cytochrome P-450 CYP3A, Humans, Computer Simulation, Drug Interactions, Dosing, media_common, business.industry, Biphenyl Compounds, Cytochrome P-450 CYP3A Inducers, Middle Aged, Smoothened Receptor, Healthy Volunteers, Ketoconazole, chemistry, 030220 oncology & carcinogenesis, Cytochrome P-450 CYP3A Inhibitors, Female, Rifampin, business, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::19413d02d53b18c1ea6a8a9c3fe17ae9Test
https://pubmed.ncbi.nlm.nih.gov/28122787Test -
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المؤلفون: Mary F. Paine, Yolanda Scarlett, Christina S. Won, Tian Lan, Karen M. VanderMolen, Nicholas H. Oberlies, Wilbur W. Widmer, Paul A. Dawson
المصدر: The Journal of Clinical Pharmacology. 53:982-990
مصطلحات موضوعية: Pharmacology, food.ingredient, Fexofenadine, Organic anion transporter 1, biology, Chemistry, food and beverages, Grapefruit juice, Organic anion-transporting polypeptide, chemistry.chemical_compound, food, Citrus paradisi, Pharmacokinetics, biology.protein, medicine, Pharmacology (medical), Terfenadine, Naringin, medicine.drug
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::eec4d131d51f2a686430075ba6f6d988Test
https://doi.org/10.1002/jcph.136Test -
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المؤلفون: Mary F. Paine, Nicholas H. Oberlies, Christina S. Won
المصدر: Pharmacology & Therapeutics. 136:186-201
مصطلحات موضوعية: Drug, media_common.quotation_subject, In silico, Pharmacology, Article, law.invention, Beverages, Food-Drug Interactions, Pharmacokinetics, In vivo, law, Animals, Cytochrome P-450 CYP3A, Humans, Pharmacology (medical), Glucuronosyltransferase, Intestinal Mucosa, media_common, Clinical pharmacology, biology, Chemistry, Clinical study design, Cytochrome P450, Biological Transport, Arylsulfotransferase, biology.protein, Citrus paradisi
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4cbae2c75d3094de0bc1451461793236Test
https://doi.org/10.1016/j.pharmthera.2012.08.001Test -
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المؤلفون: Mary F. Paine, Christina S. Won, Nicholas H. Oberlies
مصطلحات موضوعية: Drug, media_common.quotation_subject, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmacology, Biology, Intestinal absorption, Article, Food-Drug Interactions, Pharmacokinetics, Intestinal mucosa, Animals, Humans, Prodrugs, Intestinal Mucosa, Biotransformation, media_common, Mechanism (biology), Membrane Transport Proteins, Biological Transport, Intestines, Drug development, Intestinal Absorption, Pharmaceutical Preparations, Research Design, Drug metabolism
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e227a0ba0720d06c22153261ae842d63Test
https://europepmc.org/articles/PMC3034088Test/