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المؤلفون: Yongbo Hu, Karen Collins, Edward J. Salaski, Nancy Torres, Eileen Frommer, Dennis Powell, Wang Xiaolun, Jeremy I. Levin, Donald Wojciechowicz, Dan Maarten Berger
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:6571-6574
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Substrate Specificity, Structure-Activity Relationship, Pyrimidine analogue, Drug Discovery, Protein Kinase Inhibitors, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Kinase, Organic Chemistry, In vitro, Pyrimidines, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Pyrazoles, Molecular Medicine, Signal transduction
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::981acddc510eaf8186f924c43131f046Test
https://doi.org/10.1016/j.bmcl.2009.10.030Test -
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المؤلفون: Rob Van Soest, Akbar Tahir, Robert Mallon, Irwin Hollander, David E. Williams, Raymond J. Andersen, Larry Feldberg, Eileen Frommer
المصدر: Journal of Natural Products. 72:1106-1109
مصطلحات موضوعية: Sesterterpenes, Stereochemistry, medicine.medical_treatment, Pharmaceutical Science, Marine Biology, Tumor cells, Biology, Animal origin, Analytical Chemistry, Carteriospongia foliascens, Endopeptidases, Drug Discovery, medicine, Animals, Humans, Protease Inhibitors, Pharmacology, Protease, Molecular Structure, Extramural, Organic Chemistry, biology.organism_classification, Porifera, Sponge, Complementary and alternative medicine, Biochemistry, Indonesia, Molecular Medicine
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bd31a3b2af8ada25421ea61a271139b4Test
https://doi.org/10.1021/np900042rTest -
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المؤلفون: Edward J. Salaski, Wang Xiaolun, Dennis Powell, Donald Wojciechowicz, Eileen Frommer, Dan M. Berger, Karen Collins, Yongbo Hu
المصدر: Bioorganicmedicinal chemistry letters. 21(23)
مصطلحات موضوعية: Models, Molecular, Niacinamide, Proto-Oncogene Proteins B-raf, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Isoindoles, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Potency, Enzyme Inhibitors, Molecular Biology, Molecular Structure, Chemistry, Kinase, Phenylurea Compounds, Organic Chemistry, Benzenesulfonates, Imidazoles, Isoindoline, Sorafenib, Combinatorial chemistry, Enzyme Activation, Drug Design, Molecular Medicine, Structure based, Phthalazines, Selectivity
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cc2b84f81a40df7101d2b4f6a8635c87Test
https://pubmed.ncbi.nlm.nih.gov/22024030Test -
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المؤلفون: Steven C. Kim, Yongbo Hu, Nancy Torres, Dan Maarten Berger, Ariamala Gopalsamy, Kyung-Hee Kim, Weixin Xu, Donald Wojciechowicz, Larry Feldberg, Jeremy I. Levin, Dennis Powell, James M. Wilhelm, Greg Ciszewski, Eileen Frommer, Karen Collins, Minu Dutia, Robert Mallon
المصدر: Bioorganicmedicinal chemistry letters. 19(23)
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Crystallography, X-Ray, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Transferase, Structure–activity relationship, Molecular Biology, Protein Kinase Inhibitors, Trifluoromethyl, Molecular Structure, Kinase, Chemistry, Aryl, Organic Chemistry, Stereoisomerism, Pyrimidines, Benzamides, Molecular Medicine, Pyrazoles
الوصول الحر: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e8c93c7ce2c3fcc01d9a845c40838c5cTest
https://pubmed.ncbi.nlm.nih.gov/19864136Test